S. Gackenheimer

发表

Na+-dependent high affinity binding of [3H]LY515300, a 3,4-dimethyl-4-(3-hydroxyphenyl)piperidine opioid receptor inverse agonist.

P. Emmerson, T. Suter, M. Statnick, 2003, European journal of pharmacology.

Regulation of Endogenous (Male) Rodent GLP-1 Secretion and Human Islet Insulin Secretion by Antagonism of Somatostatin Receptor 5

F. Willard, T. Suter, M. Statnick, 2017, Endocrinology.

Functional autoradiography of neuropeptide Y Y1 and Y2 receptor subtypes in rat brain using agonist stimulated [35S]GTPγS binding

D. Gehlert, J. Shaw, S. Gackenheimer, 2003, Journal of Chemical Neuroanatomy.

Differential distribution of neuropeptide Y Y1 and Y2 receptors in rat and guinea-pig brains

D. Gehlert, S. Gackenheimer, 1996, Neuroscience.

Expression cloning of a human brain neuropeptide Y Y2 receptor

D. Johnson, D. Gehlert, L. Beavers, 1996, Regulatory Peptides.

[125I]Leu31, Pro34-PYY is a High Affinity Radioligand for Rat PP1/Y4 and Y1 Receptors: Evidence for Heterogeneity in Pancreatic Polypeptide Receptors

D. Larhammar, D. Gehlert, L. Beavers, 1997, Peptides.

Potent and selective 1,2,3-trisubstituted indole NPY Y-1 antagonists.

P. Hipskind, S. Iyengar, D. Zimmerman, 1997, Journal of medicinal chemistry.

Synthesis and evaluation of a series of novel 2-[(4-chlorophenoxy)methyl]benzimidazoles as selective neuropeptide Y Y1 receptor antagonists.

P. Hipskind, P. Ornstein, B. Cantrell, 1998, Journal of medicinal chemistry.

Characterization of the neuropeptide Y5 receptor in the human hypothalamus: a lack of correlation between Y5 mRNA levels and binding sites

M. Statnick, D. Gehlert, L. Beavers, 1998, Brain Research.

Structure-activity relationship of a series of diaminoalkyl substituted benzimidazole as neuropeptide Y Y1 receptor antagonists.

P. Hipskind, P. Ornstein, B. Cantrell, 1999, Bioorganic & medicinal chemistry letters.

Pharmacological characterization of (125)I-1229U91 binding to Y1 and Y4 neuropeptide Y/Peptide YY receptors.

M. Heiman, D. Gehlert, S. Gackenheimer, 2000, The Journal of pharmacology and experimental therapeutics.

Characterization of neuropeptide Y Y1-like and Y2-like receptor subtypes in the mouse brain

D. Gehlert, S. Gackenheimer, D. Schober, 2001, Peptides.

Cloning and characterization of Rhesus monkey neuropeptide Y receptor subtypes 1 1 The nucleotide sequences and translated proteins reported in this manuscript have been deposited in the Genbank data base (accession nos. rhNPY-Y1R, AF303089; rhNPY-Y2R, AF3030901 and rhNPY-Y5R, AF30309).

D. Gehlert, M. Baez, L. Beavers, 2001, Peptides.

Distribution of nociceptin and Ro64-6198 activated [35S]-GTPγS binding in the rat brain

D. Gehlert, J. Shaw, S. Gackenheimer, 2006, Neuropeptides.

Localization of rat brain binding sites for [3H]tomoxetine, an enantiomerically pure ligand for norepinephrine reuptake sites

D. Robertson, D. Gehlert, S. Gackenheimer, 1993, Neuroscience Letters.

Autoradiographic localization of subtypes of angiotensin II antagonist binding in the rat brain

D. Gehlert, S. Gackenheimer, D. Schober, 1991, Neuroscience.

Angiotensin II receptor subtypes in rat brain: dithiothreitol inhibits ligand binding to All-1 and enhances binding to All-2

D. Gehlert, S. Gackenheimer, D. Schober, 1991, Brain Research.

Angiotensin II receptor subtypes in rat brain: dithiothreitol inhibits ligand binding to AII-1 and enhances binding to AII-2.

D. Gehlert, S. Gackenheimer, D. Schober, 1991, Brain research.

[Leu31-Pro34] neuropeptide Y identifies a subtype of 125I-labeled peptide YY binding sites in the rat brain

D. Gehlert, S. Gackenheimer, D. Schober, 1992, Neurochemistry International.

Unexpected high density of neuropeptide Y Y1 receptors in the guinea pig spleen

D. Gehlert, S. Gackenheimer, 1996, Peptides.

The neuropeptide Y Y1 receptor selective radioligand, [125I][Leu31,Pro34]peptide YY, is also a high affinity radioligand for human pancreatic polypeptide 1 receptors.

D. Larhammar, D. Gehlert, L. Beavers, 1996, European Journal of Pharmacology.

Localization of opioid receptor antagonist [3H]-LY255582 binding sites in mouse brain: Comparison with the distribution of mu, delta and kappa binding sites

J. Pintar, T. Suter, M. Statnick, 2005, Neuropeptides.

In vitro and ex vivo autoradiography of the NK-1 antagonist [3H]-LY686017 in Guinea pig brain

D. Gehlert, S. Gackenheimer, 2011, Neuropeptides.

Synthesis and evaluation of radioligands for imaging brain nociceptin/orphanin FQ peptide (NOP) receptors with positron emission tomography.

Robert B. Innis, Victor W. Pike, Johannes T. Tauscher, 2011, Journal of medicinal chemistry.

Localization of ATP sensitive potassium channels in the rat brain using a novel radioligand, [125I]iodoglibenclamide.

J. Krushinski, D. Robertson, D. Gehlert, 1990, European journal of pharmacology.

Quantitative autoradiography of the binding sites for [125I] iodoglyburide, a novel high-affinity ligand for ATP-sensitive potassium channels in rat brain.

D. Robertson, D. Gehlert, D. Mais, 1991, The Journal of pharmacology and experimental therapeutics.

[3H]-quinelorane binds to D2 and D3 dopamine receptors in the rat brain.

D. Gehlert, S L Gackenheimer, J M Schaus, 1995, The Journal of pharmacology and experimental therapeutics.

Synthesis and evaluation of [125 I]-(S)-iodozacopride , a high affinity radioligand for 5HT3 receptors

D. Robertson, D. Gehlert, D. Mais, 1993, Neurochemistry International.

Localization of 5-HT3 receptors in the rat brain using [3H]LY278584

D. Wong, D. Robertson, D. Gehlert, 1991, Brain Research.

Autoradiographic comparison of [125I]LSD-labeled 5-HT2A receptor distribution in rat and guinea pig brain

D. Gehlert, S. Watts, Marlene L. Cohen, 1994, Neurochemistry International.

Stress and central Urocortin increase anxiety-like behavior in the social interaction test via the CRF1 receptor.

A. Shekhar, D. Gehlert, J. Shaw, 2005, European journal of pharmacology.

Localization of neuropeptide Y immunoreactivity and [125I]peptide YY binding sites in the human pituitary

W. Millington, B. Chronwall, D. Gehlert, 1994, Peptides.

Autoradiographic localization of [3H]quinpirole binding to dopamine D2 and D3 receptors in rat brain.

P. Seeman, D. Gehlert, P Seeman, 1992, European journal of pharmacology.

Comparison of the distribution of binding sites for the potassium channel ligands [125I]Apamin, [125I]Charybdotoxin and [125I]Iodoglyburide in the rat brain

D. Gehlert, S. Gackenheimer, 1993, Neuroscience.

Autoradiographic localization of [125I]charybdotoxin binding sites in rat brain

D. Robertson, D. Gehlert, S. Gackenheimer, 1992, Neuroscience Letters.

Non-peptide angiotensin II receptor antagonists discriminate subtypes of 125I-angiotensin II binding sites in the rat brain.

D. Gehlert, J. Reel, S. Gackenheimer, 1990, European journal of pharmacology.

Pharmacological characterization of neuropeptide Y-(2-36) binding to neuropeptide Y Y1 and Y2 receptors.

D. Gehlert, S. Gackenheimer, D. Schober, 1996, European journal of pharmacology.