Teresa A. Martin

The SERM/SERD Bazedoxifene Disrupts ESR1 Helix 12 to Overcome Acquired Hormone Resistance in Breast Cancer Cells

Myles A Brown, S. Chandarlapaty, E. Tajkhorshid, 2018, bioRxiv.

Licorice root components in dietary supplements are selective estrogen receptor modulators with a spectrum of estrogenic and anti-estrogenic activities

B. Katzenellenbogen, J. Katzenellenbogen, K. Carlson, 2016, Steroids.

Mechanisms enforcing the estrogen receptor β selectivity of botanical estrogens

B. Katzenellenbogen, J. Katzenellenbogen, I. Khan, 2013, FASEB journal : official publication of the Federation of American Societies for Experimental Biology.

A mutant form of ERα associated with estrogen insensitivity affects the coupling between ligand binding and coactivator recruitment

R. Houtman, J. Katzenellenbogen, K. Korach, 2020, Science Signaling.

Cyclic Ketoximes as Estrogen Receptor β Selective Agonists

J. Katzenellenbogen, K. Carlson, T. Tuccinardi, 2016, ChemMedChem.

Selective Human Estrogen Receptor Partial Agonists (ShERPAs) for Tamoxifen-Resistant Breast Cancer.

J. Katzenellenbogen, G. Thatcher, D. Tonetti, 2016, Journal of medicinal chemistry.

Estrogen receptor alpha somatic mutations Y537S and D538G confer breast cancer endocrine resistance by stabilizing the activating function-2 binding conformation

Sarat Chandarlapaty, Emad Tajkhorshid, Patrick R Griffin, 2016, eLife.

The SERM/SERD bazedoxifene disrupts ESR1 helix 12 to overcome acquired hormone resistance in breast cancer cells

S. Chandarlapaty, E. Tajkhorshid, J. Nwachukwu, 2018, bioRxiv.

Neural-Network Scoring Functions Identify Structurally Novel Estrogen-Receptor Ligands

Rommie E. Amaro, Jacob D. Durrant, Tavina L. Offutt, 2015, J. Chem. Inf. Model..

The SERM / SERD Bazedoxifene Disrupts ESR 1 Helix 12 to Overcome Acquired Hormone 1 Resistance in Breast Cancer Cells 2

S. Chandarlapaty, E. Tajkhorshid, J. Nwachukwu, 2022 .

Licorice root components in dietary supplements are selective estrogen receptor modulators with a spectrum of estrogenic and anti-estrogenic activities

B. Katzenellenbogen, J. Katzenellenbogen, K. Carlson, 2016, Steroids.