K. Kumura

发表

Synthesis and structure–activity relationships of novel lincomycin derivatives. Part 2. Synthesis of 7(S)-7-deoxy-7-(4-morpholinocarbonylphenylthio)lincomycin and its 3-dimensional analysis with rRNA

K. Ajito, Yoshinari Wakiyama, K. Kumura, 2015, The Journal of Antibiotics.

Synthesis and structure–activity relationships of novel lincomycin derivatives. Part 1. Newly generated antibacterial activities against Gram-positive bacteria with erm gene by C-7 modification

K. Ajito, Yoshinari Wakiyama, K. Kumura, 2015, The Journal of Antibiotics.

Synthesis and antibacterial activity of novel lincomycin derivatives. III. Optimization of a phenyl thiadiazole moiety

K. Ajito, Yoshinari Wakiyama, K. Kumura, 2017, The Journal of Antibiotics.

Synthesis and antibacterial activity of novel lincomycin derivatives. IV. Optimization of an N-6 substituent

Keiko Yamada, K. Ajito, Yoshinari Wakiyama, 2017, The Journal of Antibiotics.

Synthesis and antibacterial activity of novel lincomycin derivatives. II. Exploring (7S)-7-(5-aryl-1,3,4-thiadiazol-2-yl-thio)-7-deoxylincomycin derivatives

K. Ajito, Yoshinari Wakiyama, K. Kumura, 2016, The Journal of Antibiotics.

Synthesis and antibacterial activity of novel lincomycin derivatives. I. Enhancement of antibacterial activities by introduction of substituted azetidines

K. Ajito, Yoshinari Wakiyama, K. Kumura, 2016, The Journal of Antibiotics.

A Novel Synthesis of 2,3-Disubstituted-4-pyridones from 4-Methoxypyridine

K. Kumura, H. Kitagawa, K. Atsumi, 2006 .

Characterization of compound A, a novel lincomycin derivative active against methicillin-resistant Staphylococcus aureus

K. Maebashi, K. Ajito, Keiko Yamada, 2020, The Journal of Antibiotics.

4-Pyridone derivatives as new inhibitors of bacterial enoyl-ACP reductase FabI.

K. Kumura, M. Iida, H. Kitagawa, 2007, Bioorganic & medicinal chemistry.

Synthesis and SARs of novel lincomycin derivatives Part 5: optimization of lincomycin analogs exhibiting potent antibacterial activities by chemical modification at the 6- and 7-positions

Y. Hayashi, K. Ajito, Yoshinari Wakiyama, 2017, The Journal of Antibiotics.

Synthesis and structure–activity relationships of novel lincomycin derivatives. Part 4: synthesis of novel lincomycin analogs modified at the 6- and 7-positions and their potent antibacterial activities

Keiko Yamada, K. Ajito, T. Okutomi, 2017, The Journal of Antibiotics.

Synthesis and structure–activity relationships of novel lincomycin derivatives part 3: discovery of the 4-(pyrimidin-5-yl)phenyl group in synthesis of 7(S)-thiolincomycin analogs

K. Ajito, Yoshinari Wakiyama, K. Kumura, 2016, The Journal of Antibiotics.

Discovery of 4-Pyridone Derivatives as Specific Inhibitors of Enoyl-Acyl Carrier Protein Reductase (FabI) with Antibacterial Activity against Staphylococcus aureus

K. Kumura, M. Iida, H. Kitagawa, 2007, The Journal of Antibiotics.