P. Glunz

发表

Atropisomer Control in Macrocyclic Factor VIIa Inhibitors.

L. Mueller, D. Cheney, Yan Zou, 2016, Journal of medicinal chemistry.

Design and synthesis of bicyclic pyrimidinone-based HCV NS3 protease inhibitors.

B. Douty, C. Decicco, Peter W Glunz, 2003, Bioorganic & medicinal chemistry letters.

Design and synthesis of bicyclic pyrazinone and pyrimidinone amides as potent TF-FVIIa inhibitors.

Wen Jiang, R. Knabb, A. Rendina, 2013, Bioorganic & medicinal chemistry letters.

Design and synthesis of bicyclic pyrimidinone-based HCV NS3 protease inhibitors.

B. Douty, C. Decicco, P. Glunz, 2003, Bioorganic & medicinal chemistry letters.

Advances in Anticoagulants

J. Smallheer, M. Quan, P. Glunz, 2017 .

Recent encounters with atropisomerism in drug discovery.

P. Glunz, 2018, Bioorganic & medicinal chemistry letters.

Design and synthesis of potent, selective phenylimidazole-based FVIIa inhibitors.

D. Cheney, C. Weigelt, R. Wexler, 2015, Bioorganic & medicinal chemistry letters.

Nonbenzamidine acylsulfonamide tissue factor-factor VIIa inhibitors.

D. Cheney, C. Weigelt, Yan Zou, 2013, Bioorganic & medicinal chemistry letters.

Probing cell-surface architecture through synthesis: an NMR-determined structural motif for tumor-associated mucins.

S. Kuduk, S. Danishefsky, L. Williams, 1999, Proceedings of the National Academy of Sciences of the United States of America.

On the power of chemical synthesis: Immunological evaluation of models for multiantigenic carbohydrate-based cancer vaccines

S. Danishefsky, L. Williams, G. Ragupathi, 2002, Proceedings of the National Academy of Sciences of the United States of America.

Toward optimized carbohydrate-based anticancer vaccines: Epitope clustering, carrier structure, and adjuvant all influence antibody responses to Lewisy conjugates in mice

S. Hintermann, S. Danishefsky, K. Lloyd, 2001, Proceedings of the National Academy of Sciences of the United States of America.

Synthetic and Immunological Studies on Clustered Modes of Mucin-Related Tn and TF O-Linked Antigens: The Preparation of a Glycopeptide-Based Vaccine for Clinical Trials against Prostate Cancer†

S. Kuduk, Xiao-tao Chen, S. Danishefsky, 1998 .

The Semipermeable surface, a new restricted access medium

J. A. Perry, B. Invergo, P. Glunz, 1992 .

Neutral macrocyclic factor VIIa inhibitors.

Brandon L. Parkhurst, Wen Jiang, D. Cheney, 2017, Bioorganic & medicinal chemistry letters.

Synthesis and P1' SAR exploration of potent macrocyclic tissue factor-factor VIIa inhibitors.

Wen Jiang, D. Cheney, Yan Zou, 2016, Bioorganic & medicinal chemistry letters.

P2Y6 Receptor Potentiates Pro-Inflammatory Responses in Macrophages and Exhibits Differential Roles in Atherosclerotic Lesion Development

Rongan Zhang, P. Gargalovic, D. Gordon, 2014, PloS one.

Discovery of a Highly Potent, Selective, and Orally Bioavailable Macrocyclic Inhibitor of Blood Coagulation Factor VIIa-Tissue Factor Complex.

Brandon L. Parkhurst, Wen Jiang, D. Cheney, 2016, Journal of medicinal chemistry.

Design and Synthesis of Phenylpyrrolidine Phenylglycinamides As Highly Potent and Selective TF-FVIIa Inhibitors.

Wen Jiang, D. Cheney, Yan Zou, 2014, ACS medicinal chemistry letters.

The synthesis and evaluation of 12,13-benzodesoxyepothilone B: A highly convergent route

T. Chou, S. Chakravarty, S. Danishefsky, 1999 .

Discovery of a Phenylpyrazole Amide ROCK Inhibitor as a Tool Molecule for in vivo Studies.

David S. Taylor, J. Sack, Chunhong Yan, 2020, Bioorganic & medicinal chemistry letters.

Design and Synthesis of Ley-Bearing Glycopeptides that Mimic Cell Surface Ley Mucin Glycoprotein Architecture

S. Hintermann, S. Kuduk, S. Danishefsky, 2000 .

Probing Cell Surface “Glyco-Architecture” through Total Synthesis. Immunological Consequences of a Human Blood Group Determinant in a Clustered Mucin-like Context

S. Hintermann, S. Kuduk, Xiao-tao Chen, 1999 .

A mild and readily scalable procedure for the N-1-difluoromethylation of ethyl 6-((tert-butyldiphenylsilyl)oxy)-1H-indazole-3-carboxylate and its applications to the N-difluoromethylation of indazole, benzotriazole, imidazole, indole and pyrazole derivatives

A. Mathur, Leon M. Smith, Jianqing Li, 2020, Journal of Fluorine Chemistry.

Principles of mucin architecture: structural studies on synthetic glycopeptides bearing clustered mono-, di-, tri-, and hexasaccharide glycodomains.

S. Kuduk, A. Royyuru, Xiao-tao Chen, 2002, Journal of the American Chemical Society.

A Broadly Applicable Method for the Efficient Synthesis of α-O-Linked Glycopeptides and Clustered Sialic Acid Residues

S. Kuduk, Xiao-tao Chen, S. Danishefsky, 1999 .

A Broadly Applicable Method for the Efficient Synthesis of α‐O‐Linked Glycopeptides and Clustered Sialic Acid Residues.

S. Kuduk, Xiao-tao Chen, S. Danishefsky, 1999 .

New Chemical Synthesis of the Promising Cancer Chemotherapeutic Agent 12,13-Desoxyepothilone B: Discovery of a Surprising Long-Range Effect on the Diastereoselectivity of an Aldol Condensation

K. Savin, S. Kuduk, A. Balog, 1999 .

In pursuit of an anticancer vaccine: a monomolecular construct containing multiple carbohydrate antigens

S. Danishefsky, L. Williams, P. Glunz, 2000 .

Reduction of Sterically Hindered α,α-disubstituted Amino Esters

D. Rich, P. Glunz, 1999 .

Phthalazinone-based lactams and cyclic ureas as ROCK2 selective inhibitors.

Yan Zou, R. Wexler, J. Muckelbauer, 2023, Bioorganic & medicinal chemistry letters.

Synthetic and Immunological Studies on Clustered Modes of Mucin‐Related Tn and TF O‐Linked Antigens: The Preparation of a Glycopeptide‐Based Vaccine for Clinical Trials Against Prostate Cancer.

S. Kuduk, Xiao-tao Chen, S. Danishefsky, 1999 .

The synthesis and evaluation of a novel class of (E)-3-(1-cyclohexyl-1H-pyrazol-3-yl)-2-methylacrylic acid hepatitis C virus polymerase NS5B inhibitors.

Carl T. Bergstrom, B. Beno, Scott W. Martin, 2011, Bioorganic & medicinal chemistry letters.