A. Bolasco

发表

Synthesis, semipreparative HPLC separation, biological evaluation, and 3D-QSAR of hydrazothiazole derivatives as human monoamine oxidase B inhibitors.

T. Langer, S. Carradori, J. Kirchmair, 2010, Bioorganic & medicinal chemistry.

Anti-inflammatory, analgesic and antipyretic 4,6-disubstituted 3-cyano-2-aminopyridines

W. Filippelli, A. Filippelli, F. Manna, 1999 .

S. Carradori, D. Secci, A. Bolasco, 2012, Expert opinion on therapeutic patents.

Synthesis and inhibitory activity against human monoamine oxidase of N1-thiocarbamoyl-3,5-di(hetero)aryl-4,5-dihydro-(1H)-pyrazole derivatives.

S. Carradori, D. Secci, M. Yáñez, 2010, European journal of medicinal chemistry.

Synthesis and Selective Inhibitory Activity Against Human COX‐1 of Novel 1‐(4‐Substituted‐thiazol‐2‐yl)‐3,5‐di(hetero)aryl‐pyrazoline Derivatives

C. De Monte, S. Carradori, D. Secci, 2012, Archiv der Pharmazie.

Synthesis and selective human monoamine oxidase inhibition of 3-carbonyl, 3-acyl, and 3-carboxyhydrazido coumarin derivatives.

S. Carradori, D. Secci, S. Alcaro, 2011, European journal of medicinal chemistry.

Enantiomers of C(5)-chiral 1-acetyl-3,5-diphenyl-4,5-dihydro-(1H)-pyrazole derivatives: Analytical and semipreparative HPLC separation, chiroptical properties, absolute configuration, and inhibitory activity against monoamine oxidase.

D. Secci, R. Cirilli, R. Ferretti, 2004, Chirality.

Monoamine oxidase isoform-dependent tautomeric influence in the recognition of 3,5-diaryl pyrazole inhibitors.

D. Secci, S. Alcaro, F. Ortuso, 2007, Journal of medicinal chemistry.

Synthesis and molecular modelling studies of prenylated pyrazolines as MAO-B inhibitors.

A. Vitali, S. Alcaro, M. Yáñez, 2010, Bioorganic & medicinal chemistry letters.

A chromatographic study on the exceptional enantioselectivity of cellulose tris(4-methylbenzoate) towards C5-chiral 4,5-dihydro-(1H)-pyrazole derivatives.

S. Alcaro, R. Cirilli, R. Ferretti, 2011, Journal of chromatography. A.

Synthesis and biological evaluation of N-substituted-3,5-diphenyl-2-pyrazoline derivatives as cyclooxygenase (COX-2) inhibitors.

S. Alcaro, R. Cirilli, F. Orallo, 2010, European journal of medicinal chemistry.

Simple Extraction and HPLC Determination of UV-A and UV-B Filters in Sunscreen Products

D. Tonelli, D. Orsi, A. Bolasco, 2006 .

Synthesis, stereochemical identification, and selective inhibitory activity against human monoamine oxidase-B of 2-methylcyclohexylidene-(4-arylthiazol-2-yl)hydrazones.

S. Carradori, D. Secci, S. Alcaro, 2008, Journal of medicinal chemistry.

Selective inhibitory activity against MAO and molecular modeling studies of 2-thiazolylhydrazone derivatives.

D. Secci, S. Alcaro, F. Ortuso, 2007, Journal of medicinal chemistry.

Synthesis and in vitro activity of 2-thiazolylhydrazone derivatives compared with the activity of clotrimazole against clinical isolates of Candida spp.

S. Carradori, D. Secci, E. Maccioni, 2007, Bioorganic & medicinal chemistry letters.

Polymerization of P-diethynylbiphenyl via oxidative or catalytic reactions

M. Russo, A. Frezza, G. Ortaggi, 1992 .

Synthesis, anti-Candida activity, and cytotoxicity of new (4-(4-iodophenyl)thiazol-2-yl)hydrazine derivatives.

S. Carradori, L. Polletta, D. Secci, 2012, European journal of medicinal chemistry.

Synthesis of a novel series of thiazole-based histone acetyltransferase inhibitors.

S. Carradori, C. Canzonetta, P. Ballario, 2014, Bioorganic & medicinal chemistry.

Synthesis and evaluation of 4-acyl-2-thiazolylhydrazone derivatives for anti-Toxoplasma efficacy in vitro.

S. Carradori, D. Secci, L. Jones-Brando, 2009, Journal of medicinal chemistry.

Selective MAO-B inhibitors: a lesson from natural products

S. Carradori, D. Secci, A. Bolasco, 2014, Molecular Diversity.

Conventional and Microwave-Assisted Synthesis of Benzimidazole Derivatives and Their In Vitro Inhibition of Human Cyclooxygenase

S. Carradori, D. Secci, M. Yáñez, 2012 .

Anti-inflammatory, analgesic and antipyretic 4,6-disubstituted 3-cyanopyridine-2-ones and 3-cyano-2-aminopyridines

W. Filippelli, A. Filippelli, F. Manna, 1992 .

Chalcones: a valid scaffold for monoamine oxidases inhibitors.

D. Secci, S. Alcaro, M. Yáñez, 2009, Journal of medicinal chemistry.

Synthesis and in vitro selective anti-Helicobacter pylori activity of N-substituted-2-oxo-2H-1-benzopyran-3-carboxamides.

S. Carradori, D. Secci, A. Granese, 2006, European journal of medicinal chemistry.

Synthesis of some pyrazole derivatives and preliminary investigation of their affinity binding to P-glycoprotein.

G. Scambia, C. Ferlini, D. Secci, 2005, Bioorganic & medicinal chemistry letters.

Discovery and optimization of pyrazoline derivatives as promising monoamine oxidase inhibitors.

S. Carradori, D. Secci, E. Maccioni, 2012, Current topics in medicinal chemistry.

The state of the art of pyrazole derivatives as monoamine oxidase inhibitors and antidepressant/anticonvulsant agents.

S. Carradori, D. Secci, A. Bolasco, 2011, Current medicinal chemistry.

Synthesis and Molecular Modelling of Novel Substituted‐4,5‐dihydro‐(1H)‐pyrazole Derivatives as Potent and Highly Selective Monoamine Oxidase‐A Inhibitors

D. Secci, S. Alcaro, F. Ortuso, 2006, Chemical biology & drug design.

Design, synthesis and biological characterization of thiazolidin-4-one derivatives as promising inhibitors of Toxoplasma gondii.

C. De Monte, S. Carradori, D. Secci, 2014, European journal of medicinal chemistry.

Synthesis and anti-Helicobacter pylori Activity of 4-(Coumarin-3-yl)thiazol-2-ylhydrazone Derivatives.

S. Carradori, D. Secci, F. Sisto, 2011 .

Synthesis and anti-Helicobacter pylori activity of 4-(coumarin-3-yl)thiazol-2-ylhydrazone derivatives

S. Carradori, D. Secci, F. Sisto, 2010 .

Synthesis and biological evaluation of novel conjugated coumarin‐thiazole systems

S. Carradori, D. Secci, A. Granese, 2009 .

Synthesis, selective anti-Helicobacter pylori activity, and cytotoxicity of novel N-substituted-2-oxo-2H-1-benzopyran-3-carboxamides.

S. Carradori, D. Secci, A. Zicari, 2010, Bioorganic & medicinal chemistry letters.

A novel class of selective anti-Helicobacter pylori agents 2-oxo-2H-chromene-3-carboxamide derivatives.

S. Carradori, D. Secci, A. Zicari, 2007, Bioorganic & medicinal chemistry letters.

Synthesis and in vitro selective anti-Helicobacter pylori activity of pyrazoline derivatives.

D. Secci, A. Granese, F. Manna, 2005, Bioorganic & medicinal chemistry letters.

High-performance liquid chromatographic separation of enantiomers and diastereomers of 2-methylcyclohexanone thiosemicarbazone, and determination of absolute configuration and configurational stability.

S. Carradori, D. Secci, R. Cirilli, 2007, Journal of chromatography. A.

Investigations on the 2-thiazolylhydrazyne scaffold: synthesis and molecular modeling of selective human monoamine oxidase inhibitors.

S. Carradori, D. Secci, S. Alcaro, 2010, Bioorganic & medicinal chemistry.

Synthesis, molecular modeling, and selective inhibitory activity against human monoamine oxidases of 3-carboxamido-7-substituted coumarins.

Stefano Alcaro, Francesco Ortuso, Adriana Bolasco, 2009, Journal of medicinal chemistry.

Microwave and ultrasound-assisted synthesis of thiosemicarbazones and their corresponding (4,5-substituted-thiazol-2-yl)hydrazines

S. Carradori, D. Secci, A. Bolasco, 2014 .

LC Determination of Coumarin-3-Acyl Derivatives for Evaluation of the Stability and Monoamine Oxidase Inhibition Mechanism

D. Secci, A. Granese, D. Orsi, 2005 .

Synthesis and beta-adrenoreceptor blocking activity of [[3-(alkylamine)-2-hydroxypropyl]oximino]pyridines and O[3-(alkylamine)-2-hydroxypropyl]methylpyridine ketone oximes derivatives.

M. Fontana, A. Filippelli, F. Manna, 1996, Farmaco.

Synthesis and cytotoxicity of novel (thiazol-2-yl)hydrazine derivatives as promising anti-Candida agents.

S. Carradori, D. Secci, L. Lotti, 2013, European journal of medicinal chemistry.

Recent advances in the development of selective human MAO-B inhibitors: (hetero)arylidene-(4-substituted-thiazol-2-yl)hydrazines.

S. Carradori, D. Secci, R. Nescatelli, 2012, European journal of medicinal chemistry.

Synthesis, molecular modeling studies, and selective inhibitory activity against monoamine oxidase of 1-thiocarbamoyl-3,5-diaryl-4,5-dihydro-(1H)- pyrazole derivatives.

D. Secci, S. Alcaro, R. Cirilli, 2005, Journal of medicinal chemistry.

Synthesis and biological evaluation of novel 2,4-disubstituted-1,3-thiazoles as anti-Candida spp. agents.

S. Carradori, D. Secci, A. Granese, 2011, European journal of medicinal chemistry.

A novel histone acetyltransferase inhibitor modulating Gcn5 network: cyclopentylidene-[4-(4'-chlorophenyl)thiazol-2-yl)hydrazone.

S. Carradori, P. Ballario, P. Filetici, 2009, Journal of medicinal chemistry.

Anti-inflammatory, analgesic and antipyretic N-acetyl-Δ2-pyrazolines and dihydrothienocoumarines

E. Marmo, M. D'Amico, F. Manna, 1992 .

Selective MAO-B inhibitors: a lesson from natural products

S. Carradori, D. Secci, A. Bolasco, 2013, Molecular Diversity.

Homoisoflavonoids: natural scaffolds with potent and selective monoamine oxidase-B inhibition properties.

S. Alcaro, M. Yáñez, F. Orallo, 2011, Journal of medicinal chemistry.

Synthesis, molecular modeling studies and selective inhibitory activity against MAO of N1-propanoyl-3,5-diphenyl-4,5-dihydro-(1H)-pyrazole derivatives.

D. Secci, S. Alcaro, F. Ortuso, 2008, European journal of medicinal chemistry.

Inhibition of amine oxidases activity by 1-acetyl-3,5-diphenyl-4,5-dihydro-(1H)-pyrazole derivatives.

B. Mondovì, D. Secci, A. Tafi, 2002, Bioorganic & medicinal chemistry letters.

Synthesis and inhibitory activity against human monoamine oxidase of N1-thiocarbamoyl-3,5-di(hetero)aryl-4,5-dihydro-(1H)-pyrazole derivatives.

S. Carradori, D. Secci, M. Yáñez, 2010, European journal of medicinal chemistry.

Synthesis and selective inhibitory activity of 1-acetyl-3,5-diphenyl-4,5-dihydro-(1H)-pyrazole derivatives against monoamine oxidase.

B. Mondovì, D. Secci, R. Cirilli, 2004, Journal of medicinal chemistry.

Inhibitory effect of 1,3,5-triphenyl-4,5-dihydro-(1H)-pyrazole derivatives on activity of amine oxidases.

B. Mondovì, P. Pietrangeli, F. Manna, 1998, Journal of enzyme inhibition.

Inhibition of monoamine oxidases by coumarin-3-acyl derivatives: biological activity and computational study.

D. Secci, S. Alcaro, F. Ortuso, 2004, Bioorganic & medicinal chemistry letters.

Anti-Candida activity and cytotoxicity of a large library of new N-substituted-1,3-thiazolidin-4-one derivatives.

C. De Monte, S. Carradori, A. Mollica, 2016, European journal of medicinal chemistry.

Analytical and semipreparative high performance liquid chromatography enantioseparation of new substituted 1-thiocarbamoyl-3,5-diaryl-4,5-dihydro-(1H)-pyrazoles on polysaccharide-based chiral stationary phases in normal-phase, polar organic and reversed-phase conditions.

D. Secci, R. Cirilli, R. Ferretti, 2006, Journal of chromatography. A.

Synthesis of New Diethynylbenzene Derivatives

D. Secci, A. Granese, F. Chimenti, 2004 .

Organometallic Platinum(II) and Palladium(II) Polymers Containing 2,6-Diethynyl-4-nitroaniline Bridging Spacer and Related Dinuclear Model Complexes

M. Russo, G. Polzonetti, I. Fratoddi, 2004 .

Synthesis and characterization of new 3‐acyl‐7‐hydroxy‐6,8‐substituted‐coumarin and 3‐acyl‐7‐benzyloxy‐6,8‐substituted‐coumarin derivatives

S. Carradori, D. Secci, A. Granese, 2010 .

A new series of flavones, thioflavones, and flavanones as selective monoamine oxidase-B inhibitors.

D. Secci, S. Alcaro, R. Cirilli, 2010, Bioorganic & Medicinal Chemistry.

Focusing on new monoamine oxidase inhibitors

S. Carradori, R. Fioravanti, A. Bolasco, 2010, Expert opinion on therapeutic patents.

Synthesis and selective inhibition of human monoamine oxidases of a large scaffold of (4,5-substituted-thiazol-2-yl)hydrazones

S. Carradori, D. Secci, M. Yáñez, 2010 .

Synthesis, stereochemical separation, and biological evaluation of selective inhibitors of human MAO-B: 1-(4-arylthiazol-2-yl)-2-(3-methylcyclohexylidene)hydrazines.

S. Carradori, D. Secci, R. Cirilli, 2010, Journal of medicinal chemistry.

Recent development of monoamine oxidase inhibitors

S. Carradori, R. Fioravanti, A. Bolasco, 2005 .

Antiinflammatory, analgesic and antipyretic 4,6-disubstituted 3-cyanopyridine-2-ones and 3-cyano-2-aminopyridines

W. Filippelli, A. Filippelli, F. Chimenti, 1992 .

CPTH6, a Thiazole Derivative, Induces Histone Hypoacetylation and Apoptosis in Human Leukemia Cells

L. Ricci-Vitiani, S. Carradori, D. Trisciuoglio, 2011, Clinical Cancer Research.

Quercetin as the active principle of Hypericum hircinum exerts a selective inhibitory activity against MAO-A: extraction, biological analysis, and computational study.

Stefano Alcaro, Francesco Ortuso, Adriana Bolasco, 2006, Journal of natural products.

Synthesis, biological evaluation and 3D-QSAR of 1,3,5-trisubstituted-4,5-dihydro-(1H)-pyrazole derivatives as potent and highly selective monoamine oxidase A inhibitors.

T. Langer, D. Secci, S. Alcaro, 2006, Current Medicinal Chemistry.

HPLC Determination of 6-Methylcoumarin and 3-Pyridine Methanol in Toiletries for Oral Hygiene

D. Tonelli, D. Orsi, A. Bolasco, 2000 .

Environmental geology problems in the Tyrrhenian coastal area of Santa Marinella, province of Rome, central Italy

G. Patrizi, A. Bolasco, F. Manna, 1997 .

Synthesis and biological assessment of novel 2-thiazolylhydrazones and computational analysis of their recognition by monoamine oxidase B.

Stefano Alcaro, Gerhard Wolber, Johannes Kirchmair, 2012, European journal of medicinal chemistry.

Synthesis, molecular modeling studies, and selective inhibitory activity against monoamine oxidase of N,N'-bis[2-oxo-2H-benzopyran]-3-carboxamides.

S. Carradori, D. Secci, S. Alcaro, 2006, Bioorganic & medicinal chemistry letters.

Computer-Aided Molecular Design of Asymmetric Pyrazole Derivatives with Exceptional Enantioselective Recognition toward the Chiralcel OJ-H Stationary Phase

Stefano Alcaro, Francesco Ortuso, Adriana Bolasco, 2012, J. Chem. Inf. Model..

Identification and quantification of hydroquinone and some of its ethers in cosmetic products by reversed-phase high-performance liquid chromatography.

D. Tonelli, F. Chimenti, A. Bolasco, 1987, Journal of chromatography.

Antiinflammatory, Analgesic and Antipyretic 4,6-Disubstituted 3-Cyano-2-aminopyridines.

W. Filippelli, A. Filippelli, F. Manna, 1999 .

Synthesis of a novel series of thiazole-based histone acetyltransferase inhibitors.

S. Carradori, C. Canzonetta, P. Ballario, 2014, Bioorganic & medicinal chemistry.

Pyrrolnitrin analogues. XI--Synthesis and microbiological activity of new 1,4- and 1,5-diarylpyrroles.

N. Simonetti, M. Biava, S. Panico, 1985, Il Farmaco; edizione scientifica.