G. Cirrincione

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Synthesis of a new class of pyrrolo[3,4-h]quinazolines with antimitotic activity.

P. Brun, O. Issinger, P. Diana, 2014, European journal of medicinal chemistry.

Synthesis of the new ring system 6,8-dihydro-5H-pyrrolo[3,4-h]quinazoline

P. Diana, V. Spanò, P. Barraja, 2009 .

Three‐Membered Heterocyclic Rings and Their Fused Derivatives

P. Diana, G. Cirrincione, 2015 .

2-Diazoindoles: building blocks for the synthesis of antineoplastic agents.

A. M. Almerico, A. Lauria, P. Diana, 2002, Farmaco.

Pyrrolo[2,1-d][1,2,3,5]tetrazinones deaza analogues of temozolomide with potent antitumor activity.

A. M. Almerico, A. Lauria, P. Diana, 2000, Farmaco.

2-Triazenopyrroles: synthesis and biological activity

A. M. Almerico, A. Lauria, P. Diana, 1999 .

Quality characteristics and in vitro digestibility study of barley flour enriched ditalini pasta

L. Tesoriere, A. Attanzio, M. A. Livrea, 2016 .

The potential of neurotrophic tyrosine kinase (NTRK) inhibitors for treating lung cancer

E. Giovannetti, A. Russo, C. Rolfo, 2016, Expert opinion on investigational drugs.

Synthesis and Antitumor Activity of 3‐(2‐Phenyl‐1,3‐thiazol‐4‐yl)‐1H‐indoles and 3‐(2‐Phenyl‐1,3‐thiazol‐4‐yl)‐1H‐7‐azaindoles

N. Zaffaroni, M. Pennati, P. Diana, 2011, ChemMedChem.

Synthesis of 5H-pyrido[3,2-b]pyrrolizin-5-one tripentone analogs with antitumor activity.

P. Diana, L. Tesoriere, A. Attanzio, 2018, European journal of medicinal chemistry.

New Tripentone Analogs with Antiproliferative Activity

P. Diana, L. Tesoriere, A. Attanzio, 2017, Molecules.

New Imidazo[2,1-b][1,3,4]Thiadiazole Derivatives Inhibit FAK Phosphorylation and Potentiate the Antiproliferative Effects of Gemcitabine Through Modulation of the Human Equilibrative Nucleoside Transporter-1 in Peritoneal Mesothelioma

E. Giovannetti, G. Peters, N. Zaffaroni, 2020, AntiCancer Research.

Synthesis and Antiproliferative Activity of 2,5-bis(3′-Indolyl)pyrroles, Analogues of the Marine Alkaloid Nortopsentin

A. Maier, H. Fiebig, P. Diana, 2013, Marine drugs.

Synthesis and antiproliferative mechanism of action of pyrrolo[3',2':6,7] cyclohepta[1,2-d]pyrimidin-2-amines as singlet oxygen photosensitizers.

P. Diana, S. Richter, M. Nadai, 2016, European journal of medicinal chemistry.

Synthesis and photocytotoxic activity of [1,2,3]triazolo[4,5-h][1,6]naphthyridines and [1,3]oxazolo[5,4-h][1,6]naphthyridines.

P. Diana, S. Richter, M. Nadai, 2019, European journal of medicinal chemistry.

Synthesis, antitumor activity and CDK1 inhibiton of new thiazole nortopsentin analogues.

P. Diana, L. Tesoriere, A. Attanzio, 2017, European journal of medicinal chemistry.

3-(6-Phenylimidazo [2,1-b][1,3,4]thiadiazol-2-yl)-1H-Indole Derivatives as New Anticancer Agents in the Treatment of Pancreatic Ductal Adenocarcinoma

E. Giovannetti, N. Funel, G. Peters, 2020, Molecules.

Eight-Membered Rings With Two Heteroatoms 1,3

P. Diana, G. Cirrincione, 2021, Reference Module in Chemistry, Molecular Sciences and Chemical Engineering.

Biological Evaluation of the Antiproliferative and Anti-migratory Activity of a Series of 3-(6-Phenylimidazo[2,1-b][1,3,4]thiadiazol-2-yl)-1H-indole Derivatives Against Pancreatic Cancer Cells*

E. Giovannetti, G. Peters, D. Carbone, 2019, Anticancer Research.

Nucleophilic substitutions in the isoindole series as a valuable tool to synthesize derivatives with antitumor activity

P. Diana, A. Martorana, A. Montalbano, 2011 .

Imidazo[2,1-b] [1,3,4]thiadiazoles with antiproliferative activity against primary and gemcitabine-resistant pancreatic cancer cells.

E. Giovannetti, N. Funel, G. Peters, 2020, European journal of medicinal chemistry.

New tricyclic systems of biological interest. Annelated 1,2,3-triazolo[1,5-a]pyrimidines through domino reaction of 3-azidopyrroles and methylene active nitriles

A. M. Almerico, A. Lauria, P. Diana, 2002 .

3-Triazenoindoles. Synthesis and antileukemic activity

A. M. Almerico, P. Diana, P. Barraja, 1994 .

Pharmaceutical Approaches to Target Antibiotic Resistance Mechanisms.

P. Diana, V. Spanò, A. Montalbano, 2017, Journal of medicinal chemistry.

New 1,2,4-Oxadiazole Nortopsentin Derivatives with Cytotoxic Activity

Simona Musella, P. Diana, L. Tesoriere, 2019, Marine drugs.

Synthesis of isoindolo[1,4]benzoxazinone and isoindolo[1,5]benzoxazepine: two new ring systems of pharmaceutical interest

C. Ciancimino, P. Diana, V. Spanò, 2015 .

Aza-isoindolo and isoindolo-azaquinoxaline derivatives with antiproliferative activity.

M. Palumbo, P. Diana, L. Tesoriere, 2015, European journal of medicinal chemistry.

Water-soluble isoindolo[2,1-a]quinoxalin-6-imines: in vitro antiproliferative activity and molecular mechanism(s) of action.

P. Mátyus, N. Zaffaroni, M. Palumbo, 2015, European journal of medicinal chemistry.

Synthesis of [1,2]oxazolo[5,4-e]indazoles as antitumour agents

P. Diana, V. Spanò, A. Montalbano, 2013 .

Synthesis of the new oligopeptide pyrrole derivative isonetropsin and its one pyrrole unit analogue

P. Diana, V. Spanò, A. Montalbano, 2013 .

Synthesis and Antiproliferative Activity of the Ring System [1,2]Oxazolo[4,5‐g]indole

P. Diana, V. Spanò, A. Montalbano, 2012, ChemMedChem.

An efficient synthesis of pyrrolo[3′,2′:4,5]thiopyrano[3,2-b]pyridin-2-one: a new ring system of pharmaceutical interest

P. Diana, V. Spanò, A. Montalbano, 2012 .

Synthesis of Triazenoazaindoles: a New Class of Triazenes with Antitumor Activity

P. Brun, O. Issinger, P. Diana, 2011, ChemMedChem.

Synthesis and antitumor activity of 2,5-bis(3'-indolyl)-furans and 3,5-bis(3'-indolyl)-isoxazoles, nortopsentin analogues.

H. Fiebig, P. Diana, G. Kelter, 2010, Bioorganic & medicinal chemistry.

Pyrano[2,3-e]isoindol-2-ones, new angelicin heteroanalogues.

G. Viola, Alessia Salvador, F. Dall'acqua, 2009, Bioorganic & medicinal chemistry letters.

Isoindolo[2,1-a]quinoxaline derivatives, novel potent antitumor agents with dual inhibition of tubulin polymerization and topoisomerase I.

G. Basso, G. Viola, P. Diana, 2008, Journal of medicinal chemistry.

Synthesis and photochemotherapeutic activity of thiopyrano[2,3-e]indol-2-ones.

G. Basso, A. M. Almerico, A. Lauria, 2005, Bioorganic & medicinal chemistry letters.

Pyrrolo[2,3-h]quinolinones: synthesis and photochemotherapic activity.

A. M. Almerico, A. Lauria, G. Viola, 2003, Bioorganic & medicinal chemistry letters.

Novel 1H-pyrrolo[2,3-b]pyridine derivative nortopsentin analogues: synthesis and antitumor activity in peritoneal mesothelioma experimental models.

N. Zaffaroni, M. Pennati, P. Diana, 2013, Journal of medicinal chemistry.

Eight-Membered Rings With Two Heteroatoms 1,2

P. Diana, G. Cirrincione, 2021, Reference Module in Chemistry, Molecular Sciences and Chemical Engineering.

1,2,4-Oxadiazole topsentin analogs as staphylococcal biofilm inhibitors targeting the bacterial transpeptidase sortase A.

E. Giovannetti, D. Carbone, Simona Musella, 2020, European journal of medicinal chemistry.

Quality, functional and sensory evaluation of pasta fortified with extracts from Opuntia ficus-indica cladodes.

P. Diana, L. Tesoriere, A. Attanzio, 2019, Journal of the science of food and agriculture.

Synthesis and antitumor activities of 1,2,3-triazines and their benzo- and heterofused derivatives.

P. Diana, V. Spanò, A. Montalbano, 2017, European journal of medicinal chemistry.

Eight-membered Rings with Two Heteroatoms 1,5

P. Diana, G. Cirrincione, 2008 .

Synthesis and antiproliferative activity of [1,2,4]triazino [4,3-a] indoles.

A. M. Almerico, A. Lauria, P. Diana, 2004, Anticancer research.

Pyrrolo[2,1-c][1,2,4]triazines from 2-diazopyrroles: synthesis and antiproliferative activity.

A. M. Almerico, A. Lauria, P. Diana, 2002, European journal of medicinal chemistry.

11H-Pyrido[3',2':4,5]pyrrolo[3,2-c]cinnoline and pyrido[3',2':4,5]pyrrolo[1,2-c][1,2,3]benzotriazine: two new ring systems with antitumor activity.

P. Diana, Alessia Salvador, D. Vedaldi, 2014, Journal of medicinal chemistry.

Polycondensed nitrogen heterocycles. Part 13. Pyrrolo[3,2-b]indole by intramolecular nucleophilic substitution reaction in the pyrrole series†

G. Cirrincione, G. Dattolo, E. Aiello, 1984 .

Reaction of amino substituted heterocycles with one heteroatom in a five‐membered ring as enamines. A revision

P. Diana, F. Mingoia, S. Grimaudo, 1995 .

Determination of copper and zinc levels in human hair

G. Allegri, C. Costa, A. Bertazzo, 1996, Biological Trace Element Research.

Pyrrolo[3,4-h]quinolinones a new class of photochemotherapeutic agents.

G. Basso, G. Viola, P. Diana, 2011, Bioorganic & medicinal chemistry.

Isoindolo[2,1-c]benzo[1,2,4]triazines: a new ring system with antiproliferative activity.

A. Lauria, P. Diana, A. Martorana, 2007, Bioorganic & medicinal chemistry.

Polycondensed nitrogen heterocycles. Part 27. Indolo[3,2-c]cinnoline. Synthesis and antileukemic activity.

P. Diana, P. Barraja, F. Mingoia, 1995, Farmaco.

Polycondensed nitrogen heterocycles. XXII. A new synthesis of 5,6-dihydro-7H-pyrazolo[1,5-d][1,4]benzodiazepin-6-ones†

G. Cirrincione, G. Dattolo, E. Aiello, 1982 .

Synthetic small molecules as anti-biofilm agents in the struggle against antibiotic resistance.

E. Giovannetti, P. Diana, I. Carnevale, 2019, European journal of medicinal chemistry.

Synthesis and antitumor properties of 2,5-bis(3'-indolyl)thiophenes: analogues of marine alkaloid nortopsentin.

O. Gia, L. Dalla Via, P. Diana, 2007, Bioorganic & medicinal chemistry letters.

An overview on the recent developments of 1,2,4-triazine derivatives as anticancer compounds.

P. Diana, V. Spanò, A. Montalbano, 2017, European journal of medicinal chemistry.

3-Diazopyrroles. Part 6. Mutagenic activity of 3-diazopyrroles in Streptomyces coelicolor A3(2) during various phases of growth.

P. Diana, P. Barraja, F. Mingoia, 1996, Farmaco.

3-Diazopyrroles. Part 5 (1). Antibacterial activity of 3-diazo-2-phenylpyrroles.

P. Diana, S. Grimaudo, G. Cirrincione, 1992, Farmaco.

1-Methyl-3H-pyrazolo[1,2-a]benzo[1,2,3,4]tetrazin-3-ones. Design, synthesis, and biological activity of new antitumor agents.

A. Lauria, P. Diana, A. Montalbano, 2005, Journal of medicinal chemistry.

Glycosidopyrroles. Part 3. Effect of the benzocondensation on acyclic derivatives: 1-(2-hydroxyethoxy) methylindoles as potential antiviral agents.

G. Perra, P. Diana, M. Marongiu, 1998, Farmaco.

Pyrrolo[3,2‐h]quinazolines as Photochemotherapeutic Agents

P. Brun, P. Diana, Alessia Salvador, 2011, ChemMedChem.

Rarrangements of N-ureidopyrroles : a case of mononuclear heterocyclic rearrangement involving an aromatic heterocycle as carbon-nitrogen-nitrogen sequence

P. Diana, G. Cirrincione, G. Macaluso, 1991 .

NUCLEOPHILIC REACTIONS IN THE PYRROLE SERIES : DISPLACEMENT OF HALOGEN AS A TOOL TO FUNCTIONALIZE THE PYRROLE NUCLEUS

P. Diana, F. Mingoia, G. Cirrincione, 1997 .

Thiopyrano[2,3-e]indol-2-ones: angelicin heteroanalogues with potent photoantiproliferative activity.

G. Viola, P. Diana, Alessia Salvador, 2008, Bioorganic & medicinal chemistry.

3,5-bis(3'-indolyl)pyrazoles, analogues of marine alkaloid nortopsentin: synthesis and antitumor properties.

O. Gia, P. Diana, A. Martorana, 2007, Bioorganic & medicinal chemistry letters.

Thiazoles, Their Benzofused Systems, and Thiazolidinone Derivatives: Versatile and Promising Tools to Combat Antibiotic Resistance

E. Giovannetti, D. Carbone, P. Diana, 2020, Journal of medicinal chemistry.

Therapeutic Strategies To Counteract Antibiotic Resistance in MRSA Biofilm‐Associated Infections

E. Giovannetti, D. Carbone, P. Diana, 2020, ChemMedChem.

Pyrazolo[3,4-h]quinolines promising photosensitizing agents in the treatment of cancer.

P. Brun, P. Diana, Alessia Salvador, 2015, European journal of medicinal chemistry.

2,6-Disubstituted imidazo[2,1-b][1,3,4]thiadiazole derivatives as potent staphylococcal biofilm inhibitors.

E. Giovannetti, Simona Musella, P. Diana, 2019, European journal of medicinal chemistry.

Synthesis and antiproliferative activity of 2-triazenothiophenes.

A. Lauria, P. Diana, P. la Colla, 1999, Anticancer research.

Seven‐, Eight‐Membered and Larger Heterocyclic Rings and Their Fused Derivatives

P. Diana, G. Cirrincione, 2015 .

Reactivity of aminopyrroles: Protonation

P. Diana, P. Barraja, F. Mingoia, 1996 .

Protonation of 3-aminopyrroles

R. Jones, G. Cirrincione, G. Dattolo, 1987 .

Six‐Membered Rings, and Their Fused Derivatives

P. Diana, G. Cirrincione, 2015 .

3-[4-(1H-Indol-3-yl)-1,3-thiazol-2-yl]-1H-pyrrolo[2,3-b]pyridines, Nortopsentin Analogues with Antiproliferative Activity

C. Ciancimino, P. Diana, L. Tesoriere, 2015, Marine drugs.

Synthesis and antiproliferative activity of substituted 3[2-(1H-indol-3-yl)- 1,3-thiazol-4-yl]-1H-pyrrolo[3,2-b]pyridines, marine alkaloid nortopsentin analogues.

N. Zaffaroni, M. Pennati, P. Diana, 2014, Current medicinal chemistry.

Synthesis of the new ring system pyrrolizino[2,3-b]indol-4(5H)-one

P. Diana, A. Montalbano, P. Barraja, 2011 .

New synthesis of condensed heterocycles from isoxazole derivatives VI. 2,5‐Dimethyl‐3‐aeetyl‐7‐amino‐1H‐pyrrolo[3,2‐b] pyridine

G. Cirrincione, G. Daidone, G. Dattolo, 1978 .

New syntheses of condensed heterocycles from isoxazole derivatives. V. Pyrrolo[3,4-b ]pyridin-4-ones

G. Cirrincione, G. Daidone, G. Dattolo, 1977 .

Polycondensed nitrogen heterocycles. X. 5,6,7,8-Tetrahydropyrrolo[1,2-e][1,5]benzodiazocin-7-ones. A new ring system†‡

G. Cirrincione, G. Dattolo, E. Aiello, 1981 .

Pyrrolo[2,1-d][1,2,3,5]tetrazine-4(3H)-ones, a new class of azolotetrazines with potent antitumor activity.

A. Lauria, P. Diana, A. Montalbano, 2003, Bioorganic & medicinal chemistry.

Biosynthesis of Heterocycles: From Isolation to Gene Cluster

P. Diana, G. Cirrincione, 2015 .

Synthesis of the new ring system 2-oxo-[1,4]oxazino[3,2-e]indole, heteroanalogue of Angelicin

P. Diana, A. Martorana, A. Montalbano, 2009 .

Polycondensed nitrogen heterocycles. Part 8. Pyrrolo[3,2-b]indole

G. Cirrincione, G. Dattolo, E. Aiello, 1981 .

Pyrrolo[2,3-d][1,2,3]triazoles as Potential Antineoplastic Agents

A. Lauria, P. Diana, P. Barraja, 1998 .

Pyrrolo[2,3-h]quinolinones: a new ring system with potent photoantiproliferative activity.

G. Viola, P. Diana, F. Dall'acqua, 2006, Bioorganic & medicinal chemistry.

1,3,5-Triazines: A promising scaffold for anticancer drugs development.

P. Diana, V. Spanò, A. Montalbano, 2017, European journal of medicinal chemistry.

Synthesis of pyrrolo[3,2-h]quinolinones with good photochemotherapeutic activity and no DNA damage.

P. Brun, G. Palù, P. Diana, 2010, Bioorganic & medicinal chemistry.

Derivatives of the new ring system indolo[1,2-c]benzo[1,2,3]triazine with potent antitumor and antimicrobial activity.

A. Lauria, P. Diana, P. la Colla, 1999, Journal of Medicinal Chemistry.

Polycondensed nitrogen heterocycles. Part 22. Pyrrolo[3,4-d]-1,2,3-triazines: A new ring system as potential antineoplastic agent †

G. Cirrincione, G. Dattolo, E. Aiello, 1989 .

Synthesis and Antiproliferative Activity of Thiazolyl-bis-pyrrolo[2,3-b]pyridines and Indolyl-thiazolyl-pyrrolo[2,3-c]pyridines, Nortopsentin Analogues

P. Diana, L. Tesoriere, A. Attanzio, 2015, Marine drugs.

Nucleophilic reactions in the indole series: displacement of bromine under phase transfer catalysis

P. Diana, P. Barraja, A. Carbone, 2008 .

A synthetic approach to new polycyclic ring system of biological interest through domino reaction: indolo[2,3-e][1,2,3]triazolo[1,5-a]pyrimidine

A. Lauria, P. Diana, A. Montalbano, 2006 .

Annelated pyrrolo-pyrimidines from amino-cyanopyrroles and BMMAs as leads for new DNA-interactive ring systems.

A. Lauria, P. Diana, A. Montalbano, 2005, Bioorganic & medicinal chemistry.

Pyrrolo[3,4‐e][1,2,3]triazolo[1,5‐a]pyrimidine and pyrrolo[3,4‐d] [1,2,3]triazolo[1,5‐a]pyrimidine. New tricyclic ring systems of biological interest

A. Lauria, P. Diana, P. Barraja, 2000 .

Pyrrolotetrazinones deazaanalogues of temozolomide induce apoptosis in Jurkat cell line: involvement of tubulin polymerization inhibition

P. Brun, G. Basso, G. Viola, 2009, Cancer Chemotherapy and Pharmacology.

[1,2]Oxazolo[5,4-e]isoindoles as promising tubulin polymerization inhibitors.

N. Zaffaroni, M. Pennati, P. Diana, 2016, European journal of medicinal chemistry.

Preclinical Activity of New [1,2]Oxazolo[5,4-e]isoindole Derivatives in Diffuse Malignant Peritoneal Mesothelioma.

N. Zaffaroni, M. Pennati, P. Diana, 2016, Journal of medicinal chemistry.

Pyrrolo[3',2':6,7]cyclohepta[1,2-b]pyridines with potent photo-antiproliferative activity.

P. Diana, Alessia Salvador, S. Richter, 2017, European journal of medicinal chemistry.

Itraconazole inhibits nuclear delivery of extracellular vesicle cargo by disrupting the entry of late endosomes into the nucleoplasmic reticulum

G. Vistoli, D. Corbeil, P. Diana, 2021, Journal of extracellular vesicles.

2-Triazenoazaindoles: A novel class of triazenes inducing transcriptional down-regulation of EGFR and HER-2 in human pancreatic cancer cells

O. Issinger, B. Guerra, D. Litchfield, 2011, International journal of oncology.

Pyrrolo[2,1-d][1,2,3,5]tetrazine-4(3H)-ones with Potent Antitumor Activity

G. Cirrincione, 2003 .

CHK1 inhibitor sensitizes resistant colorectal cancer stem cells to nortopsentin

M. Todaro, G. Stassi, I. Screpanti, 2021, iScience.

Eight-membered heterocycles with two heteroatoms in a 1,2-relationship of interest in medicinal chemistry

D. Carbone, P. Diana, B. Parrino, 2021 .

Bacterial Biofilm Inhibition in the Development of Effective Anti-Virulence Strategy

P. Diana, B. Parrino, G. Cirrincione, 2018, The open medicinal chemistry journal.

Nanostructured Lipid Carriers-Containing Anticancer Compounds: Preparation, Characterization, and Cytotoxicity Studies

G. Giammona, P. Diana, M. Bondì, 2007, Drug delivery.

New Thiazole Nortopsentin Analogues Inhibit Bacterial Biofilm Formation

P. Diana, V. Spanò, A. Montalbano, 2018, Marine drugs.

Interleukin 3- receptor targeted exosomes inhibit in vitro and in vivo Chronic Myelogenous Leukemia cell growth

Stefania Raimondo, Stefano Forte, Patrizia Diana, 2017, Theranostics.

An overview of recent molecular dynamics applications as medicinal chemistry tools for the undruggable site challenge.

Ugo Perricone, Alessandro Padova, Maria Rita Gulotta, 2018, MedChemComm.

Preparation of monohalopyrroles

G. Cirrincione, G. Dattolo, E. Aiello, 1982 .

Polycondensed nitrogen heterocycles. Part 23. Pyrrolo[3,2-c]cinnolines by a japp-klingemann type reaction†

G. Cirrincione, G. Dattolo, E. Aiello, 1990 .

Polycondensed nitrogen heterocycles. Part 19. Pyrrolo[1,2‐f]phenanthridines by pschorr‐type cyclization brought about by hypophosphorous acid

G. Cirrincione, G. Dattolo, E. Aiello, 1986 .

Studies on the synthesis of heterocyclic compounds. Part I. The pschorr reaction in the pyrazole series

G. Cirrincione, G. Daidone, G. Dattolo, 1978 .

A Multivariate Analysis of HIV-1 Protease Inhibitors and Resistance Induced by Mutation

Anna Maria Almerico, Antonino Lauria, Marco Tutone, 2006, J. Chem. Inf. Model..

Metabolomics-assisted discovery of a new anticancer GLS-1 inhibitor chemotype from a nortopsentin-inspired library: From phenotype screening to target identification.

A. Bertamino, P. Campiglia, D. Carbone, 2022, European journal of medicinal chemistry.

1,2,4-Amino-triazine derivatives as pyruvate dehydrogenase kinase inhibitors: Synthesis and pharmacological evaluation.

S. Moro, D. Carbone, V. Gandin, 2023, European journal of medicinal chemistry.

Thiazole Analogues of the Marine Alkaloid Nortopsentin as Inhibitors of Bacterial Biofilm Formation

D. Carbone, P. Diana, A. Carbone, 2020, Molecules.

Pyrido[2’,3’:4,5]pyrrolo[2,1-d][1,2,3,5]tetrazine-4(3H)-ones, a new class of temozolomide heteroanalogues

P. Diana, A. Martorana, A. Montalbano, 2009 .

On the preparation of 1-aryl-2-heteroaryl- and 2-aryl-1-heteroaryl-pyrroles as useful building blocks for biologically interesting heterocycles

A. Lauria, P. Diana, A. Montalbano, 2002 .

Techniques for Biosynthesis

P. Diana, G. Cirrincione, 2015 .

Discovery of the 3-Amino-1,2,4-triazine-Based Library as Selective PDK1 Inhibitors with Therapeutic Potential in Highly Aggressive Pancreatic Ductal Adenocarcinoma

S. Moro, D. Carbone, V. Gandin, 2023, International journal of molecular sciences.

1,2,4‐Oxadiazole Topsentin Analogs with Antiproliferative Activity against Pancreatic Cancer Cells, Targeting GSK3β Kinase

E. Giovannetti, D. Carbone, Simona Musella, 2020, ChemMedChem.

Structural Manipulations of Marine Natural Products Inspire a New Library of 3-Amino-1,2,4-Triazine PDK Inhibitors Endowed with Antitumor Activity in Pancreatic Ductal Adenocarcinoma.

S. Moro, D. Carbone, V. Gandin, 2023, Marine drugs.

Biosynthesis of Heterocycles: Diana/Biosynthesis of Heterocycles

P. Diana, G. Cirrincione, 2015 .

Eight-membered heterocycles with two heteroatoms in a 1,5-relationship of interest in medicinal chemistry

D. Carbone, P. Diana, B. Parrino, 2020 .

Synthesis of the New Ring System Bispyrido[4',3':4,5]pyrrolo[1,2-a:1',2'-d]pyrazine and Its Deaza Analogue

P. Diana, V. Spanò, A. Montalbano, 2014, Molecules.

Protonation of Aminoindoles

A. Lauria, P. Diana, P. Barraja, 2000 .

Eight-membered heterocycles with two heteroatoms in a 1,3-relationship of interest in medicinal chemistry

D. Carbone, P. Diana, B. Parrino, 2021 .

‘Interrupted’ diazotization of 3-aminoindoles and 3-aminopyrroles

P. Mátyus, P. Diana, V. Spanò, 2014 .

Convenient synthesis of pyrrolo[3,4-g]indazole

P. Diana, V. Spanò, A. Montalbano, 2013 .

2-triazenoindoles: synthesis and biological activity.

A. Lauria, P. Diana, A. Montalbano, 2002, Anticancer research.

Synthesis of 3-Triazenopyrroles

P. Diana, S. Grimaudo, G. Cirrincione, 1993 .

3-Triazenopyrroles: synthesis and antineoplastic activity.

P. Diana, M. Tolomeo, S. Grimaudo, 1993, Farmaco.

Synthesis and Antitumor Activity of New Thiazole Nortopsentin Analogs

P. Diana, L. Tesoriere, A. Attanzio, 2016, Marine drugs.

Inhibitors of antibiotic resistance mechanisms: clinical applications and future perspectives.

D. Carbone, P. Diana, B. Parrino, 2020, Future medicinal chemistry.

HIV-1-induced nuclear invaginations mediated by VAP-A, ORP3, and Rab7 complex explain infection of activated T cells

D. Carbone, D. Corbeil, P. Diana, 2023, Nature communications.

Polycondensed nitrogen heterocycles. IX. 5,6-dihydro-7H-pyrrolo[1,2-d][1,4]benzodiazepin-6-one

G. Cirrincione, G. Dattolo, E. Aiello, 1980 .

A Multivariate Analysis on Non-nucleoside HIV-1 Reverse Transcriptase Inhibitors and Resistance Induced by Mutation

M. Tutone, A. Lauria, P. Diana, 2003 .

marine drugs

S. Moro, D. Carbone, V. Gandin, 2022 .

Triazole derivatives inhibit the VOR complex-mediated nuclear transport of extracellular particles: Potential application in cancer and HIV-1 infection.

D. Carbone, P. Diana, B. Parrino, 2024, Bioorganic chemistry.

About the synthesis of N-1-substituted 3-aminopyrroles. A comparison †

G. Cirrincione, G. Dattolo, E. Aiello, 1989 .