Y. Ueda

发表

Envelope Conformational Changes Induced by Human Immunodeficiency Virus Type 1 Attachment Inhibitors Prevent CD4 Binding and Downstream Entry Events

James E. Robinson, R. Colonno, P. Clapham, 2006, Journal of Virology.

Synthesis and antitumor evaluation of 2′-oxycarbonylpaclitaxels (paclitaxel-2′-carbonates)

C. Fairchild, W. Rose, E. Kerns, 1994 .

Michael addition of amines and thiols to dehydroalanine amides: a remarkable rate acceleration in water.

T. Connolly, Y. Ueda, M. Sorenson, 2003, The Journal of organic chemistry.

Organic reactions in frozen water: Michael addition of amines and thiols to the dehydroalanine side chain of nocathiacins

K. S. Lam, T. Connolly, J. Bronson, 2004 .

A catalyst for ester hydrolysis showing electrostatic and hydrophobic binding properties

J. Guthrie, Y. Ueda, 1976 .

Novel water soluble phosphate prodrugs of taxol® possessing in vivo antitumor activity

W. Rose, J. Knipe, A. Casazza, 1993 .

Synthesis and antibacterial activity of nocathiacin I analogues.

K. S. Lam, M. Pucci, T. Connolly, 2006, Bioorganic & medicinal chemistry letters.

Synthesis, in vitro, and in vivo antibacterial activity of nocathiacin I thiol-Michael adducts.

M. Pucci, J. Bronson, Y. Ueda, 2005, Bioorganic & medicinal chemistry letters.

Nocathiacin I analogues: synthesis, in vitro and in vivo biological activity of novel semi-synthetic thiazolyl peptide antibiotics.

K. S. Lam, M. Pucci, T. Connolly, 2004, Bioorganic & medicinal chemistry letters.

Antimicrobial Evaluation of Nocathiacins, a Thiazole Peptide Class of Antibiotics

M. Pucci, L. Discotto, J. Barrett, 2004, Antimicrobial Agents and Chemotherapy.

Synthesis and antibacterial activity of O-substituted nocathiacin I derivatives.

M. Pucci, Xiaofan Zheng, J. Bronson, 2004, Bioorganic & medicinal chemistry letters.

Novel semi-synthetic nocathiacin antibiotics: synthesis and antibacterial activity of bis- and mono-O-alkylated derivatives.

M. Pucci, T. Connolly, Xiaofan Zheng, 2004, Bioorganic & medicinal chemistry letters.

Chemical conversion of nocathiacin I to nocathiacin II and a lactone analogue of glycothiohexide alpha.

J. Leet, M. Pucci, T. Connolly, 2005, Journal of natural products.

Synthesis of novel nocathiacin-class antibiotics. Condensation of glycolaldehyde with primary amides and tandem reductive amination of amadori-rearranged 2-oxoethyl intermediates.

Stella Huang, J. Leet, J. Bronson, 2002, The Journal of organic chemistry.

Mild method for cleavage of dehydroalanine units: highly efficient conversion of nocathiacin I to nocathiacin IV.

A. Regueiro-Ren, Y. Ueda, 2002, The Journal of organic chemistry.

Mild Method for Cleavage of Dehydroalanine Units: Highly Efficient Conversion of Nocathiacin I (Ia) to Nocathiacin IV (Ib).

A. Regueiro-Ren, Y. Ueda, 2003 .

Synthesis and structure-activity relationship of C-3 benzoyloxymethyl cephalosporins exhibiting anti-MRSA activities

J. Russell, Y. Ueda, M. Mansuri, 1997 .

A simple method of preparing trimethylsilyl- and tert-butyldimethylsilyl-enol ethers of α-diazoacetoacetates and their use in the synthesis of a chiral precursor to thienamycin analogs

Y. Ueda, G. Roberge, V. Vinet, 1984 .

An efficient enantioselective synthesis of the carbapenam-2-one system. An approach to (+)-thienamycin and related carbapenems

T. Sowin, A. Meyers, Y. Ueda, 1987 .

Synthesis of phenoxyacetyl-N-(hydroxydioxocyclobutenyl)cycloserines

Y. Ueda, L. B. Crast, A. Mikkilineni, 1991 .

Synthesis of α-(S)-acylamino-N-(hydroxydioxocyclobutenyl)-β-lactams as potential antibiotics

Y. Ueda, A. Mikkilineni, R. Partyka, 1992 .

Cyclocondensation adducts from the lewis acid mediated reaction of 4-acetoxy-2-azetidinone with siloxydienes

Y. Ueda, S. C. Maynard, 1985 .

Nuclear analogs of β-lactam antibiotics. XIX. Syntheses of racemic and enantiomeric p-nitrobenzyl carbapen-2-em-3-carboxylates

C. Damas, Y. Ueda, V. Vinet, 1983 .

Synthesis and in vitro activity of novel quaternary ammonium carbapenems: 2-pyridiniopropyl and 1-pyridinioethyl carbapenems.

Y. Ueda, V. Vinet, 1992, The Journal of antibiotics.

Highly regioselective formation of bromohydrins by reaction of epoxy-azetidinones with MgBr2: An alternative route to 4-bromomethylcarbonylmethyl-2-azetidinone, a key carbapenem precursor

Y. Ueda, S. C. Maynard, 1988 .

Nuclear analogs of β-lactam antibiotics. XVIII: A short synthesis of 2-alkylthiocarbapen-2-em-3-carboxylate

C. Damas, B. Belleau, Y. Ueda, 1983 .

Synthesis and evaluation of C2-carbon-linked heterocyclic-5-hydroxy-6-oxo-dihydropyrimidine-4-carboxamides as HIV-1 integrase inhibitors.

N. Meanwell, Zeyu Lin, M. Krystal, 2015, Bioorganic & medicinal chemistry letters.

Phosphonooxymethyl prodrugs of the broad spectrum antifungal azole, ravuconazole: synthesis and biological properties.

Qi Gao, Mandar Dali, Srini Venkatesh, 2003, Bioorganic & medicinal chemistry letters.

Novel C‐acylated triazole derivatives of ravuconazole, an azole antifungal agent

Stella Huang, J. Bronson, Y. Ueda, 2008 .

Inhibitors of human immunodeficiency virus type 1 (HIV-1) attachment 6. Preclinical and human pharmacokinetic profiling of BMS-663749, a phosphonooxymethyl prodrug of the HIV-1 attachment inhibitor 2-(4-benzoyl-1-piperazinyl)-1-(4,7-dimethoxy-1H-pyrrolo[2,3-c]pyridin-3-yl)-2-oxoethanone (BMS-488043)

N. Meanwell, R. Colonno, K. Yeung, 2012, Journal of medicinal chemistry.

Synthesis and cytostatic activity of the antitumor antibiotic chartreusin derivatives.

K. Kon, N. Yamada, Y. Ueda, 1990, The Journal of antibiotics.

Synthesis and Antitumor Evaluation of 2′-Oxycarbonylpaclitaxels ( Paclitaxel-2′-carbonates).

C. Fairchild, W. Rose, E. Kerns, 1995 .

In Vitro Antiviral Characteristics of HIV-1 Attachment Inhibitor BMS-626529, the Active Component of the Prodrug BMS-663068

N. Meanwell, M. Krystal, J. Kadow, 2012, Antimicrobial Agents and Chemotherapy.

Discovery of the Human Immunodeficiency Virus Type 1 (HIV-1) Attachment Inhibitor Temsavir and Its Phosphonooxymethyl Prodrug Fostemsavir.

N. Meanwell, D. Langley, R. Colonno, 2018, Journal of medicinal chemistry.

SKELETAL REARRANGEMENT IN DEHYDROGENATION OF THUJOPSENE AND ITS CONGENERS

M. Yatagai, K. Endo, Y. Ueda, 1974 .

Synthesis and in vitro antibacterial activity of new semi-synthetic noviosylcoumarin antibiotics: chemical modification at the C-3′ ester

Y. Ueda, J. Fung-Tomc, J. Chuang, 1994 .

Synthesis and in vitro activity of new semi-synthetic coumermycin analogs: chemical modification at the C-3 amide.

Y. Ueda, L. B. Crast, J. Chuang, 1989, The Journal of antibiotics.

A selective cleavage of the oxazole moiety in noviosylcoumarin antibiotics a new process to key intermediates for coumermycin analogue synthesis

Y. Ueda, L. B. Crast, J. Chuang, 1988 .

Synthesis and structure-activity relationship of C-3 quaternary ammonium cephalosporins exhibiting anti-MRSA activities

J. Bronson, Y. Ueda, J. Matiskella, 1997 .

Novel, water-soluble phosphate derivatives of 2′-ethoxy carbonylpaclitaxel as potential prodrugs of paclitaxel: Synthesis and antitumor evaluation

W. Rose, J. Knipe, V. Farina, 1995 .

Discovery and Development of HIV‐1 Entry Inhibitors That Target gp120

N. Meanwell, K. Yeung, J. Kadow, 2011 .

The discovery and preclinical evaluation of BMS-707035, a potent HIV-1 integrase strand transfer inhibitor.

N. Meanwell, Zeyu Lin, M. Krystal, 2018, Bioorganic & medicinal chemistry letters.