J. Balsells

发表

A case of remote asymmetric induction in the peptide-catalyzed desymmetrization of a bis(phenol).

Scott J. Miller, R. Reamer, J. Gustafson, 2008, Journal of the American Chemical Society.

Photoredox Catalysis for Silyl-Mediated C-H Alkylation of Heterocycles with Non-Activated Alkyl Bromides

Jeffrey W Schubert, E. Streckfuss, J. Balsells, 2020, European Journal of Organic Chemistry.

Silyl-mediated photoredox-catalyzed Giese reaction: addition of non-activated alkyl bromides† †Electronic supplementary information (ESI) available. See DOI: 10.1039/c8sc02253d

J. Balsells, Abdellatif ElMarrouni, Casey B Ritts, 2018, Chemical science.

Synthesis of bis-macrocyclic HCV protease inhibitor MK-6325 via intramolecular sp²-sp³ Suzuki-Miyaura coupling and ring closing metathesis.

Jeremy P. Scott, L. Tan, Cheng-yi Chen, 2015, Organic letters.

Synthesis of Sitagliptin

Feng Xu, Edward J. J. Grabowski, Shane W. Krska, 2009 .

Highly efficient asymmetric synthesis of sitagliptin.

Feng Xu, Andrew Clausen, Shane W. Krska, 2009, Journal of the American Chemical Society.

Synthesis of a CGRP Receptor Antagonist via an Asymmetric Synthesis of 3-Fluoro-4-aminopiperidine.

Manuel de Lera Ruiz, L. Tan, Jiahui Chen, 2019, The Journal of organic chemistry.

Copper-Catalyzed Synthesis of 5-Carboxyl-4-perfluoroalkyl Triazoles.

J. Balsells, Robert Panish, Tho V. Thieu, 2021, Organic letters.

Toward the total synthesis of variecolin.

G. Molander, J. Balsells, M. Quirmbach, 2001, Organic letters.

Enantioselective Synthesis of (1R,2S)-1-Amino-2-vinylcyclopropanecarboxylic Acid Ethyl Ester (Vinyl-ACCA-OEt) by Asymmetric Phase-Transfer Catalyzed Cyclopropanation of (E)-N-Phenylmethyleneglycine Ethyl Ester

Cheng-yi Chen, P. Bulger, Jingjun Yin, 2010 .

Discovery of novel oxazolidinedione derivatives as potent and selective mineralocorticoid receptor antagonists.

J. Lisnock, A. Crespo, Gaochao Zhou, 2013, Bioorganic & medicinal chemistry letters.

Careful Navigation of the Crystallographic Landscape of MK-8970: A Racemic Acetal Carbonate Prodrug of Raltegravir

Jimmy O. DaSilva, R. Ball, R. Reamer, 2015 .

Discovery of MK‐8970: An Acetal Carbonate Prodrug of Raltegravir with Enhanced Colonic Absorption

Q. Dang, Jing Li, P. Coleman, 2015, ChemMedChem.

Use of achiral and meso ligands to convey asymmetry in enantioselective catalysis.

P. Walsh, Alice E. Lurain, J. Balsells, 2003, Chemical reviews.

Temperature‐dependent nonlinear effects and catalyst evolution in the asymmetric addition of diethylzinc to benzaldehyde

P. Walsh, Anna M. Costa, J. Balsells, 2001 .

First Generation Process for the Preparation of the DPP-IV Inhibitor Sitagliptin

Edward J. J. Grabowski, Spencer D. Dreher, J. Armstrong, 2005 .

New Method for the General Synthesis of [1,2,4]Triazolo[1,5‐a]pyridines

J. Balsells, Elliott W. D. Huntsman, 2005 .

Synthesis of 2-amino-5-substituted-1,3,4-oxadiazoles using 1,3-dibromo-5,5-dimethylhydantoin as oxidant

J. Balsells, K. Hansen, N. Rivera, 2006 .

Optimization of asymmetric catalysts using achiral ligands: metal geometry-induced ligand asymmetry.

P. Carroll, P. Walsh, J. Balsells, 2001, Organic letters.

Achiral tetrahydrosalen ligands for the synthesis of C(2)-symmetric titanium complexes: a structure and diastereoselectivity study.

P. Carroll, P. Walsh, J. Balsells, 2001, Inorganic chemistry.

Insight into the mechanism of the asymmetric addition of alkyl groups to aldehydes catalyzed by titanium-BINOLate species.

P. Carroll, P. Walsh, J. Balsells, 2002, Journal of the American Chemical Society.

Snapshots of titanium BINOLate complexes with diverse solid state structures.

P. Carroll, P. Walsh, J. Balsells, 2001, Organic letters.

Synthesis of 4-Alkylated Isocoumarins via Pd-Catalyzed α-Arylation Reaction.

S. Kuduk, S. Plunkett, Lindsey G. DeRatt, 2020, Organic letters.

Highly selective and efficient conversion of aryl bromides to t-butyl benzoates with di-t-butyl dicarbonate

Hongmei Li, J. Balsells, 2008 .

An efficient catalyst for Pd-catalyzed carbonylation of aryl arenesulfonates.

Yong-kui Sun, J. McWilliams, J. Balsells, 2006, Organic letters.

Toward the understanding of the mechanism and enantioselectivity of the PausonKhand reaction. Theoretical and experimental studies

A. Riera, A. Moyano, X. Verdaguer, 2002 .

Synthesis of [1,2,4]Triazolo[4,3-α]piperazines via Highly Reactive Chloromethyloxadiazoles

J. Armstrong, Jinchu Liu, J. Balsells, 2005 .

New Method for the General Synthesis of [1,2,4]Triazolo[1,5‐a]pyridines.

J. Balsells, Elliott W. D. Huntsman, 2005 .

Synthesis of chiral sulfonamide/Schiff base ligands

R. Somanathan, G. Aguirre, P. Walsh, 1998 .

Synthesis of 2-Amino-5-substituted-1,3,4-oxadiazoles Using 1,3-Dibromo-5,5-dimethylhydantoin as Oxidant.

J. Balsells, K. Hansen, N. Rivera, 2006 .

Remote desymmetrization at near-nanometer group separation catalyzed by a miniaturized enzyme mimic.

Scott J. Miller, R. Reamer, David Pollard, 2006, Journal of the American Chemical Society.

Highly selective synthesis of 2-substituted-5-hydroxy-6-oxo-1,6-dihydropyrimidine-4-carboxylic acid derivatives using a novel protected dihydroxyfumarate

J. Armstrong, D. Mathre, T. Novak, 2004 .

Tandem Aminocarbonylation/Pauson-Khand Reaction of Haloacetylenes

A. Riera, A. Moyano, M. A. Pericàs, 1999 .

An improved preparation and a new application of trichloromethylcarbinols from enolizable ketones

T. Itoh, J. Balsells, Brenden P. Derstine, 2014 .

Efficient synthesis of chiral acetylene dithioethers in enantiomerically pure form

A. Riera, A. Moyano, M. A. Pericàs, 1997 .

Practical cleavage of trifluoroacetamides with p-toluensulfonic acid

Hongmei Li, J. Balsells, C. Spencer, 2009 .

Probing the Conformation of Flexible Catalysts in Solution

P. Walsh, J. Balsells, J. M. Betancort, 2000 .

The Use of Achiral Ligands to Convey Asymmetry: Chiral Environment Amplification.

P. Walsh, J. Balsells, 2000 .

Preparation of t‐Butyl‐3‐Bromo‐5‐Formylbenzoate Through Selective Metal‐Halogen Exchange Reactions

Hongmei Li, J. Balsells, J. Arredondo, 2014 .

Discovery of 6-(Fluoro-(18)F)-3-(1H-pyrrolo[2,3-c]pyridin-1-yl)isoquinolin-5-amine ([(18)F]-MK-6240): A Positron Emission Tomography (PET) Imaging Agent for Quantification of Neurofibrillary Tangles (NFTs).

Talakad G. Lohith, S. Melquist, L. Gantert, 2016, Journal of medicinal chemistry.

Discovery of benzimidazole oxazolidinediones as novel and selective nonsteroidal mineralocorticoid receptor antagonists.

J. Lisnock, A. Crespo, Gaochao Zhou, 2015, ACS medicinal chemistry letters.

Design of Prodrugs to Enhance Colonic Absorption by Increasing Lipophilicity and Blocking Ionization

Q. Dang, P. Coleman, A. Templeton, 2014, Pharmaceuticals.

Mineralocorticoid receptor antagonists: identification of heterocyclic amide replacements in the oxazolidinedione series.

J. Lisnock, A. Crespo, Gaochao Zhou, 2014, Bioorganic & medicinal chemistry letters.