H. Naito

发表

Design, synthesis and SAR of novel ethylenediamine and phenylenediamine derivatives as factor Xa inhibitors.

K. Uoto, Makoto Suzuki, A. Mochizuki, 2011, Bioorganic & medicinal chemistry letters.

Design, synthesis, and biological activity of piperidine diamine derivatives as factor Xa inhibitor.

K. Uoto, Yumi Nakamoto, A. Mochizuki, 2008, Bioorganic & medicinal chemistry letters.

Discovery of EP300/CBP histone acetyltransferase inhibitors through scaffold hopping of 1,4-oxazepane ring.

Y. Tominaga, Mizuki Takahashi, O. Ubukata, 2022, Bioorganic & medicinal chemistry letters.

Bystander killing effect of DS‐8201a, a novel anti‐human epidermal growth factor receptor 2 antibody–drug conjugate, in tumors with human epidermal growth factor receptor 2 heterogeneity

T. Agatsuma, K. Hagihara, H. Naito, 2016, Cancer science.

Studies on glycosphingolipids in larvae of the green-bottle fly, Lucilia caesar: two neutral glycosphingolipids having large straight oligosaccharide chains with eight and nine sugars.

F. Inagaki, H. Naito, M. Sugita, 1990, Journal of biochemistry.

Novel antibody drug conjugates containing exatecan derivative-based cytotoxic payloads.

Shinji Ashida, K. Morita, Hideki Miyazaki, 2016, Bioorganic & medicinal chemistry letters.

Cyclomaltodextrin Glucanotransferase-Catalyzed Transglycosylation from Dextrin to Alkanol Maltosides

Minoru Izumi, N. Baba, S. Nakajima, 2008, Bioscience, biotechnology, and biochemistry.

Syntheses and differentiating action of vitamin D endoperoxides. Singlet oxygen adducts of vitamin D derivatives in human myeloid leukemia cells (HL-60).

M. Ohmori, T. Suzuki, S. Yamada, 1985, Journal of medicinal chemistry.

Synthesis and mechanism of action of novel pyrimidinyl pyrazole derivatives possessing antiproliferative activity.

Y. Koiso, Y. Hashimoto, M. Minami, 2002, Bioorganic & medicinal chemistry letters.

Synthesis and antitumor activity of novel pyrimidinyl pyrazole derivatives. III. Synthesis and antitumor activity of 3-phenylpiperazinyl-1-trans-propenes.

M. Minami, R. Atsumi, H. Naito, 2005, Chemical & pharmaceutical bulletin.

Synthesis and antitumor activity of novel pyrimidinyl pyrazole derivatives.

Y. Nakamura, M. Sugimori, H. Naito, 1999, Chemical & pharmaceutical bulletin.

The First Total Synthesis of (+)-Bullatacin, a Potent Antitumor Annonaceous Acetogenin, and (+)-(15,24)-bisepi-Bullatacin

S. Sasaki, M. Maeda, E. Kawahara, 1995 .

Synthesis and antitumor activity of novel pyrimidinyl pyrazole derivatives. II. Optimization of the phenylpiperazine moiety of 1-[5-methyl-1-(2-pyrimidinyl)-4-pyrazolyl]-3-phenylpiperazinyl-1-trans-propenes.

M. Minami, M. Sugimori, Yoshihide Nakamura, 2002, Chemical & pharmaceutical bulletin.

Stereoselective synthesis of (E)-α-hydroxy-1,3-dienes via the reaction of 2,5-dihydrothiophene S,S-dioxides with carbonyl compounds

S. Yamada, T. Nomoto, H. Takayama, 1987 .

Design, synthesis, and SAR of cis-1,2-diaminocyclohexane derivatives as potent factor Xa inhibitors. Part I: exploration of 5-6 fused rings as alternative S1 moieties.

Hiroyuki Naito, Tsutomu Nagata, Kengo Watanabe, 2009, Bioorganic & medicinal chemistry.

NOVEL ACYCLIC LIGANDS FOR METAL CATIONS BASED ON THE ADJACENT BISTETRAHYDROFURAN AS ANALOGS OF NATURAL ANNONACEOUS ACETOGENINS

S. Sasaki, M. Maeda, E. Kawahara, 1998 .

The First Total Synthesis of (+)-Bullatacin (V), a Potent Antitumor Annonaceous Acetogenin, and (+)-(15,24)-bisepi-Bullatacin (VI).

S. Sasaki, M. Maeda, E. Kawahara, 1995 .

Copper-catalyzed 1,2-double amination of 1-halo-1-alkynes. Concise synthesis of protected tetrahydropyrazines and related heterocyclic compounds.

Yasuhiro Fukudome, H. Urabe, H. Naito, 2008, Journal of the American Chemical Society.

Discovery of DS-5272 as a promising candidate: A potent and orally active p53-MDM2 interaction inhibitor.

Masaki Miyazaki, Mayumi Kitagawa, K. Uoto, 2015, Bioorganic & medicinal chemistry.

New calcium-selective electrodes based on Annonaceous acetogenins and their analogs with neighboring bistetrahydrofuran

H. Sugihara, S. Sasaki, K. Hiratani, 1995 .

Novel calcium ionophores: Supramolecular complexation by the hydroxylated-bistetrahydrofuran skeleton of potent antitumor Annonaceous acetogenins

S. Sasaki, M. Maeda, E. Kawahara, 1994 .

Facile preparation of N-protected 2-alkylidene-1,3-imidazolidines

H. Urabe, H. Naito, T. Hata, 2008 .

In vitro antitumor activities of new synthetic bistetrahydrofuran derivatives as analogs of Annonaceous acetogenins.

S. Sasaki, M. Maeda, E. Kawahara, 1998, Chemical & pharmaceutical bulletin.

Diffusion of oxide ions in LaFeO3 single crystal

J. Mizusaki, S. Yamauchi, K. Fueki, 1984 .

Selective deprotection of methanesulfonamides to amines.

H. Urabe, H. Naito, T. Hata, 2010, Organic letters.

Synthesis and evaluation of novel orally active p53-MDM2 interaction inhibitors.

Keisuke Yoshida, Hiroyuki Naito, Takahiko Seki, 2013, Bioorganic & medicinal chemistry.

Lead optimization of novel p53-MDM2 interaction inhibitors possessing dihydroimidazothiazole scaffold.

Masaki Miyazaki, Mayumi Kitagawa, T. Soga, 2013, Bioorganic & medicinal chemistry letters.

Discovery of novel dihydroimidazothiazole derivatives as p53-MDM2 protein-protein interaction inhibitors: synthesis, biological evaluation and structure-activity relationships.

Masaki Miyazaki, Mayumi Kitagawa, T. Soga, 2012, Bioorganic & medicinal chemistry letters.

The Reactions of Silicon Phosphate with Alkaline Earth Metal Oxides at High Temperatures

E. Narita, H. Naito, Kazuhiro Sango, 1985 .

FTR1335 is a novel synthetic inhibitor of Candida albicans N-myristoyltransferase with fungicidal activity.

Masataka Nakamura, H. Naito, K. Nakazawa, 2005, Biological & pharmaceutical bulletin.

The Formation and Thermal Decomposition of Hydrous Lead(II) Oxide Prepared by the Alkoxide Method

E. Narita, Makito Kobayashi, H. Naito, 1983 .

Vertical distribution of components in a polymer blend with the aid of the secondary ion mass spectroscopy

T. Nishi, T. Adachi, H. Naito, 1983 .

Discovery of DS-9300: A Highly Potent, Selective, and Once-Daily Oral EP300/CBP Histone Acetyltransferase Inhibitor.

H. Ogiwara, T. Kohno, Y. Tominaga, 2022, Journal of Medicinal Chemistry.

Kinetic Study on Hydrolysis of Silicon Phosphate in Aqueous Alkaline Solutions

E. Narita, H. Naito, T. Saeki, 1984 .