Yves Depetter

Synthesis of Indoline‐Based Benzhydroxamic Acids as Potential HDAC6 Inhibitors

O. De Wever, K. De Bosscher, S. Gobec, 2019, ChemistrySelect.

Assessment of the trifluoromethyl ketone functionality as an alternative zinc-binding group for selective HDAC6 inhibition.

O. De Wever, Jorick Franceus, T. Desmet, 2018, MedChemComm.

Synthesis of Potent and Selective HDAC6 Inhibitors Bearing a Cyclohexane- or Cycloheptane-Annulated 1,5-Benzothiazepine Scaffold.

L. Van Den Bosch, K. Van Hecke, Jorick Franceus, 2017, Chemistry.

Expedient stereoselective synthesis of new dihydropyrano- and dihydrofuranonaphthoquinones

M. D’hooghe, T. V. Nguyen, H. Nguyen, 2015 .

Synthesis and anticancer properties of new (dihydro)pyranonaphthoquinones and their epoxy analogs.

M. D’hooghe, Chinh Pham The, Tuyet Anh Dang Thi, 2015, Bioorganic & medicinal chemistry letters.

Expedient Synthesis of Lupulones and Their Derivatization to 2,8‐7H‐Dihydrochromen‐7‐ones

K. Van Hecke, M. D’hooghe, Gurkirat Kaur, 2020, ChemistryOpen.

Selective pharmacological inhibitors of HDAC6 reveal biochemical activity but functional tolerance in cancer models

O. De Wever, M. Bracke, M. D’hooghe, 2019, International journal of cancer.

Synthesis and SAR assessment of novel Tubathian analogs in the pursuit of potent and selective HDAC6 inhibitors.

L. Van Den Bosch, T. Verhaeghe, T. Desmet, 2016, Organic & biomolecular chemistry.