Haolun Jin

发表

Conformationally Constrained Tricyclic HIV Integrase Inhibitors

James M. Chen, Xiaowu Chen, M. Tsiang, 2011 .

Interactive design and synthesis of a novel antibacterial agent

S. Wolfe, Haolun Jin, K. Yang, 1994 .

Investigation of novel fumagillin analogues as angiogenesis inhibitors.

C. Kim, J. Tario, M. Fardis, 2004, Bioorganic & medicinal chemistry letters.

Highly potent HCV NS4B inhibitors with activity against multiple genotypes.

Huiling Yang, W. Delaney, Ruby Z Cai, 2014, Journal of medicinal chemistry.

Discovery of a Potent and Orally Bioavailable Cyclophilin Inhibitor Derived from the Sanglifehrin Macrocycle.

J. Chiva, R. Mackman, T. Appleby, 2018, Journal of medicinal chemistry.

Preclinical Evaluation of GS-9160, a Novel Inhibitor of Human Immunodeﬁciency Virus Type 1 Integrase (cid:1) †

R. Geleziunas, Xiaowu Chen, M. Tsiang, 2009 .

Preclinical Evaluation of GS-9160, a Novel Inhibitor of Human Immunodeficiency Virus Type 1 Integrase

R. Geleziunas, Xiaowu Chen, M. Tsiang, 2008, Antimicrobial Agents and Chemotherapy.

Design, synthesis, and SAR studies of novel and highly active tri-cyclic HIV integrase inhibitors.

James M. Chen, Ruby Z Cai, Xiaowu Chen, 2006, Bioorganic & medicinal chemistry letters.

Discovery of GS-9688 (Selgantolimod), as a Potent and Selective Oral Toll-like Receptor 8 Agonist for the Treatment of Chronic Hepatitis B.

Helen Yu, R. Mackman, T. Appleby, 2020, Journal of medicinal chemistry.

Antiviral Properties of a Series of 1,6-Naphthyridine and 7,8-Dihydroisoquinoline Derivatives Exhibiting Potent Activity against Human Cytomegalovirus

L. Chan, L. L'Heureux, J. Bédard, 2000, Antimicrobial Agents and Chemotherapy.

A practical synthesis of trans-iodoolefins

W. Christ, Y. Kishi, Haolun Jin, 1986 .

On Cardioactive Steroids. XVI. Stereoselective β-Glycosylation of Digitoxose: The Synthesis of Digitoxin†

Haolun Jin, T. Y. Tsai, K. Wiesner, 1985 .

Effect of substitution on novel tricyclic HIV-1 integrase inhibitors.

Ruby Z Cai, M. Tsiang, C. Kim, 2006, Bioorganic & medicinal chemistry letters.

Diastereoselective Synthesis of the Potent Antiviral Agent (-)-2'-Deoxy-3'-thiacytidine and Its Enantiomer

P. Ravenscroft, T. Mansour, M. Siddiqui, 1995 .

Catalytic effect of nickel(II) chloride and palladium(II) acetate on chromium(II)-mediated coupling reaction of iodo olefins with aldehydes

W. Christ, Y. Kishi, J. Uenishi, 1986 .

Total synthesis of a fully protected palytoxin carboxylic acid

J. B. White, M. Martinelli, W. Christ, 1989 .

Total Synthesis of Palytoxin Carboxylic Acid and Palytoxin Amide

W. Christ, R. W. Armstrong, H. Fujioka, 1989 .

ON CARDIOACTIVE STEROIDS. XVI. STEREOSELECTIVE β-GLYCOSYLATION OF DIGITOXOSE: THE SYNTHESIS OF DIGITOXIN

Haolun Jin, T. Y. Tsai, K. Wiesner, 1985 .

Tricyclic HIV integrase inhibitors V. SAR studies on the benzyl moiety.

Xiaowu Chen, M. Tsiang, Rachael Lansdown, 2009, Bioorganic & medicinal chemistry letters.

Tricyclic HIV integrase inhibitors: VI. SAR studies of 'benzyl flipped' C3-substituted pyrroloquinolines.

Xiaowu Chen, M. Tsiang, Rachael Lansdown, 2009, Bioorganic & medicinal chemistry letters.

Tricyclic HIV integrase inhibitors: potent and orally bioavailable C5-aza analogs.

Ruby Z Cai, Xiaowu Chen, M. Tsiang, 2008, Bioorganic & medicinal chemistry letters.

Effect of Substitution on Novel Tricyclic HIV‐1 Integrase Inhibitors.

Ruby Z Cai, M. Tsiang, C. Kim, 2006 .

Composes inhibant l'integrase

Rachael Lansdown, C. Kim, M. Mish, 2006 .

Design, synthesis, and biological evaluation of novel tricyclic HIV-1 integrase inhibitors by modification of its pyridine ring.

M. Tsiang, C. Kim, Sammy Metobo, 2006, Bioorganic & medicinal chemistry letters.

Unexpected effects of Lewis acids in the synthesis of optically pure 2′-deoxy-3′-oxacytidine nucleoside analogues

P. Ravenscroft, T. Mansour, J. Payne, 1993 .

(1′R,2′S,5′R)-Menthyl-(5R)-acetoxy-1,3-oxathiolan-(2R)-carboxylate: Synthesis and isomeric purity determination by HPLC

T. Mansour, M. Siddiqui, Haolun Jin, 1994 .

Expeditious preparation of (−)-2′-deoxy-3′-thiacytidine (3TC)

T. Mansour, J. Payne, Haolun Jin, 1992 .

Catalytic Effect of Nickel(II) Chloride and Palladium(II) Acetate on Chromium(II)-Mediated Coupling Reaction of Iodo Olefins with Aldehydes.

W. Christ, Y. Kishi, J. Uenishi, 1987 .

Design, synthesis and evaluation of a series of novel fumagillin analogues.

B. Hicke, L. Green, C. Kim, 2003, Bioorganic & medicinal chemistry.

Antiviral Activity of Bictegravir (GS-9883), a Novel Potent HIV-1 Integrase Strand Transfer Inhibitor with an Improved Resistance Profile

K. White, Helen Yu, G. Kukolj, 2016, Antimicrobial Agents and Chemotherapy.