V. Straniero

发表

Targeting Bacterial Cell Division: A Binding Site-Centered Approach to the Most Promising Inhibitors of the Essential Protein FtsZ

A. Casiraghi, Lorenzo Suigo, E. Valoti, 2020, Antibiotics.

2,6‐Difluorobenzamide Inhibitors of Bacterial Cell Division Protein FtsZ: Design, Synthesis, and Structure–Activity Relationships

S. Duga, L. Straniero, A. Casiraghi, 2017, ChemMedChem.

3-(Benzodioxan-2-ylmethoxy)-2,6-difluorobenzamides bearing hydrophobic substituents at the 7-position of the benzodioxane nucleus potently inhibit methicillin-resistant Sa and Mtb cell division.

M. Pallavicini, M. Sanguinetti, G. Delogu, 2016, European journal of medicinal chemistry.

Benzodioxane-benzamides as new bacterial cell division inhibitors.

M. Pallavicini, M. Bissa, E. Valoti, 2015, European journal of medicinal chemistry.

Stressed degradation studies of domiphen bromide by LC‐ESI‐MS/MS identify a novel promising antimicrobial agent

G. Aldini, G. Vistoli, L. Regazzoni, 2018, Journal of pharmaceutical and biomedical analysis.

Thiazole- and imidazole-containing peptidomimetic inhibitors of protein farnesyltransferase.

M. Pallavicini, A. Corsini, N. Ferri, 2011, Bioorganic & medicinal chemistry letters.

Methylphenidate Analogues as a New Class of Potential Disease-Modifying Agents for Parkinson’s Disease: Evidence from Cell Models and Alpha-Synuclein Transgenic Mice

A. Newman, A. Gianoncelli, G. Ribaudo, 2022, Pharmaceutics.

Illuminating the norepinephrine transporter: fluorescent probes based on nisoxetine and talopram.

H. Sitte, G. Schütz, A. Newman, 2021, RSC medicinal chemistry.

Identification of 1-butyl-3-(1-(4-methyl)naphtoyl)indole detected for the first time in "herbal high" products on the Italian market.

M. Pallavicini, G. Roda, E. Casagni, 2012, Forensic science international.

From 2-aminomethyl-1,4-benzodioxane enantiomers to unichiral 2-cyano- and 2-carbonyl-substituted benzodioxanes via dichloroamine.

M. Pallavicini, E. Valoti, V. Straniero, 2014, The Journal of organic chemistry.

Farnesyltransferase inhibitors: CAAX mimetics based on different biaryl scaffolds.

M. Pallavicini, A. Corsini, N. Ferri, 2014, Bioorganic & medicinal chemistry letters.

One-Pot Racemization Process of 1-Phenyl-1,2,3,4-tetrahydroisoquinoline: A Key Intermediate for the Antimuscarinic Agent Solifenacin

M. Pallavicini, E. Valoti, V. Straniero, 2013 .

(3-Methylene-2,3-dihydronaphtho[2,3-b][1,4]dioxin-2-yl)methanol

Lorenzo Suigo, E. Valoti, V. Straniero, 2022, Molbank.

Oral Bioavailability and Pharmacokinetics of Nonanimal Chondroitin Sulfate and Its Constituents in Healthy Male Volunteers

F. Galeotti, N. Volpi, D. Bianchi, 2018, Clinical pharmacology in drug development.

Enantiomerically Pure Dibenzyl Esters of l-Aspartic and l-Glutamic Acid

M. Pallavicini, E. Valoti, V. Straniero, 2015 .

Staphylococcus aureus RnpA Inhibitors: Computational-Guided Design, Synthesis and Initial Biological Evaluation

V. Sebastián-Pérez, P. Dunman, A. Casiraghi, 2021, Antibiotics.

Exploring the space of histidine containing dipeptides in search of novel efficient RCS sequestering agents.

B. Testa, G. Aldini, M. Pallavicini, 2013, European journal of medicinal chemistry.

Benzodioxane‐Benzamides as Antibacterial Agents: Computational and SAR Studies to Evaluate the Influence of the 7‐Substitution in FtsZ Interaction

V. Sebastián-Pérez, M. Hrast, I. Zdovc, 2019, ChemMedChem.

Benzamide Derivatives Targeting the Cell Division Protein FtsZ: Modifications of the Linker and the Benzodioxane Scaffold and Their Effects on Antimicrobial Activity

V. Sebastián-Pérez, M. Hrast, I. Zdovc, 2020, Antibiotics.

6-methoxy-7-benzofuranoxy and 6-methoxy-7-indolyloxy analogues of 2-[2-(2,6-Dimethoxyphenoxy)ethyl]aminomethyl-1,4-benzodioxane (WB4101):1 discovery of a potent and selective α1D-adrenoceptor antagonist.

M. Gobbi, R. Budriesi, A. Chiarini, 2013, Journal of medicinal chemistry.

How Reaction Conditions May Influence the Regioselectivity in the Synthesis of 2,3-Dihydro-1,4-benzoxathiine Derivatives.

A. Casiraghi, Lorenzo Suigo, E. Valoti, 2018, The Journal of organic chemistry.

Affinity and activity profiling of unichiral 8-substituted 1,4-benzodioxane analogues of WB4101 reveals a potent and selective α1B-adrenoceptor antagonist.

M. Gobbi, R. Budriesi, A. Chiarini, 2012, European journal of medicinal chemistry.

Resolution via diastereomeric amides of enantiopure 1,4‐benzoxathian‐2‐ and 3‐carboxylic acids and determination of their configuration

Lorenzo Suigo, E. Valoti, V. Straniero, 2022, Chirality.

Computational Design and Development of Benzodioxane-Benzamides as Potent Inhibitors of FtsZ by Exploring the Hydrophobic Subpocket

V. Sebastián-Pérez, W. Margolin, M. Hrast, 2021, Antibiotics.

How do reaction conditions affect the enantiopure synthesis of 2-substituted-1,4-benzodioxane derivatives?

A. Casiraghi, E. Valoti, V. Straniero, 2018, Chirality.

Obtainment of Threo and Erythro Isomers of the 6-Fluoro-3-(2,3,6,7,8,9-hexahydronaphtho[2,3-b][1,4]dioxin-2-yl)-2,3-dihydrobenzo[b][1,4]dioxine-5-carboxamide

Lorenzo Suigo, E. Valoti, V. Straniero, 2023, Molbank.

Design and Synthesis of Fluorescent Methylphenidate Analogues for a FRET‐Based Assay of Synapsin III Binding

A. Newman, A. Casiraghi, E. Valoti, 2020, ChemMedChem.

Alpha-synuclein/synapsin III pathological interplay boosts the motor response to methylphenidate

F. Benfenati, M. Spillantini, C. Missale, 2020, Neurobiology of Disease.

Predicting the physicochemical profile of diastereoisomeric histidine-containing dipeptides by property space analysis.

B. Testa, M. Pallavicini, G. Vistoli, 2012, Chirality.

From pregabalin to rac-3-cyano-5-methylhexanoic acid: an easy conversion which valorizes waste pregabalin enantiomer

M. Pallavicini, O. Piccolo, E. Valoti, 2012 .

Benzodioxane-benzamides as promising inhibitors of Escherichia coli FtsZ.

G. Rivas, W. Margolin, C. Alfonso, 2023, International journal of biological macromolecules.