Tatsuya Urushima

发表

The direct and enantioselective, one-pot, three-component, cross-mannich reaction of aldehydes.

Y. Hayashi, M. Shoji, K. Sakai, 2003, Angewandte Chemie.

Asymmetric Mannich reaction of imines derived from aliphatic and aromatic aldehydes catalyzed by diarylprolinol silyl ether.

Y. Hayashi, H. Ishikawa, Tatsuya Urushima, 2011, Chemistry.

Highly diastereo- and enantioselective direct aldol reactions in water.

Y. Hayashi, H. Gotoh, M. Shoji, 2006 .

Direct organocatalytic mannich reaction of acetaldehyde: an improved catalyst and mechanistic insight from a computational study.

Tsubasa Okano, T. Uchimaru, Y. Hayashi, 2008, Angewandte Chemie.

The Direct, Enantioselective, One-Pot, Three-Component, Cross-Mannich Reaction of Aldehydes: The Reason for the Higher Reactivity of Aldimine versus Aldehyde in Proline-Mediated Mannich and Aldol Reactions

T. Uchimaru, Y. Hayashi, M. Shoji, 2005 .

A Highly Active 4‐Siloxyproline Catalyst for Asymmetric Synthesis

D. Hashizume, H. Koshino, Junichiro Yamaguchi, 2004 .

Highly diastereo- and enantioselective direct aldol reactions in water.

Y. Hayashi, H. Gotoh, M. Shoji, 2006, Angewandte Chemie.

One-pot synthesis of chiral aziridines by a domino reaction by using desulfonylative formation on the N-tosyl imine of chloroacetaldehyde with an asymmetric Mannich reaction as a key step.

Y. Hayashi, H. Ishikawa, Tatsuya Urushima, 2011, Chemistry.

Enantio- and diastereoselective synthesis of piperidines by coupling of four components in a "one-pot" sequence involving diphenylprolinol silyl ether mediated Michael reaction.

Y. Hayashi, H. Ishikawa, Tatsuya Urushima, 2010, Organic letters.

The stereoselective synthesis of α-substituted β-amino secondary alcohols based on the proline-mediated, asymmetric, three-component Mannich reaction and its application to the formal total synthesis of nikkomycins B and Bx

Y. Hayashi, M. Shoji, Tatsuya Urushima, 2005 .

Organic solvent-free, enantio- and diastereoselective, direct Mannich reaction in the presence of water.

Tsubasa Okano, Y. Hayashi, Tatsuya Urushima, 2008, Organic letters.

One‐Pot Synthesis of Chiral Aziridines by a Domino Reaction by Using Desulfonylative Formation on the N‐Tosyl Imine of Chloroacetaldehyde with an Asymmetric Mannich Reactions as a Key Step.

Y. Hayashi, H. Ishikawa, Tatsuya Urushima, 2012 .

Enantio- and Diastereoselective Synthesis of Piperidines by Coupling of Four Components in a “One-Pot” Sequence Involving Diphenylprolinol Silyl Ether Mediated Michael Reaction.

Y. Hayashi, H. Ishikawa, Tatsuya Urushima, 2011 .

Asymmetric epoxidation of α-substituted acroleins catalyzed by diphenylprolinol silyl ether.

B. Bondžić, Y. Hayashi, H. Ishikawa, 2010, Organic letters.

L-Proline-catalyzed enantioselective one-pot cross-Mannich reaction of aldehydes

Y. Hayashi, M. Shoji, Wataru Tsuboi, 2007, Nature Protocols.

Polymeric ethyl glyoxylate in an asymmetric aldol reaction catalyzed by diarylprolinol.

Y. Hayashi, H. Ishikawa, Tatsuya Urushima, 2010, Organic letters.

The Stereoselective Synthesis of α‐Substituted β‐Amino Secondary Alcohols Based on the Proline‐Mediated, Asymmetric, Three‐Component Mannich Reaction and Its Application to the Formal Total Synthesis of Nikkomycins B and Bx.

Y. Hayashi, M. Shoji, Tatsuya Urushima, 2006 .

Organic solvent-free, enantio- and diastereoselective, direct Mannich reaction in the presence of water.

Tsubasa Okano, Y. Hayashi, Tatsuya Urushima, 2008, Organic letters.

Fragment-to-Lead Medicinal Chemistry Publications in 2019.

Paul N. Mortenson, W. Jahnke, I. D. de Esch, 2020, Journal of medicinal chemistry.

Fragments: where are we now?

Harren Jhoti, James Osborne, Stanislava Panova, 2020, Biochemical Society transactions.

AzoCholine Enables Optical Control of Alpha 7 Nicotinic Acetylcholine Receptors in Neural Networks.

A. Gottschalk, D. Trauner, W. Kummer, 2015, ACS chemical neuroscience.