M. Journet

发表

Synthesis of bis-macrocyclic HCV protease inhibitor MK-6325 via intramolecular sp²-sp³ Suzuki-Miyaura coupling and ring closing metathesis.

Jeremy P. Scott, L. Tan, Cheng-yi Chen, 2015, Organic letters.

Synthesis of vaniprevir (MK-7009): lactamization to prepare a 20-membered [corrected] macrocycle.

Paul N. Devine, D. Tellers, D. Zewge, 2011, The Journal of organic chemistry.

Selective Continuous Flow Iodination Guided by Direct Spectroscopic Observation of Equilibrating Aryl Lithium Regioisomers

Anna L. Dunn, Bernie O’Hare, P. Liu, 2018, Organometallics.

Asymmetric Synthesis of N-Boc-(R)-Silaproline via Rh-Catalyzed Intramolecular Hydrosilylation of Dehydroalanine and Continuous Flow N-Alkylation.

John Y. L. Chung, A. Klapars, M. Shevlin, 2016, Organic letters.

Preparation of Methyltriazolo[1,4]benzodiazepine via Oxidative Activation of a Thiolactam for the Synthesis of BET Inhibitor Molibresib.

C. Pink, J. Kowalski, M. Journet, 2021, The Journal of organic chemistry.

A rapid synthesis of 2-aryl-5-substituted-2,3-dihydrobenzofurans.

Jeffrey T. Kuethe, I. Davies, M. Journet, 2005, The Journal of organic chemistry.

A Rapid, Large-Scale Synthesis of a Potent Cholecystokinin (CCK) 1R Receptor Agonist

Jeffrey T. Kuethe, G. Humphrey, M. Journet, 2008 .

Highly efficient synthesis of α,β-acetylenic aldehydes from terminal alkynes using DMF as the formylating reagent

D. Cai, M. Journet, R. Larsen, 1998 .

[3H]benzylpempidine, a new radioligand for probing a putative channel site on nicotinic cholinergic receptors.

S. Sheu, L. Abood, A. Kende, 1997, Life sciences.

An integral topical gel for cellulite reduction: results from a double-blind, randomized, placebo-controlled evaluation of efficacy

E. Loing, M. Journet, É. Dupont, 2014, Clinical, cosmetic and investigational dermatology.

Comparison of flow and batch polymerization processes for production of vinyl ether terpolymers for use in the delivery of siRNA

Benjamin W. Thuronyi, Benjamin W Thuronyi, Fanyu Meng, 2014 .

The Evolving State of Continuous Processing in Pharmaceutical API Manufacturing: A Survey of Pharmaceutical Companies and Contract Manufacturing Organizations

Timothy M. Braden, Ayman D. Allian, S. May, 2018 .

A practical synthesis of a COX-2-specific inhibitor.

K. Rossen, I. Davies, M. Palucki, 2000, The Journal of organic chemistry.

A highly regioselective amination of 6-aryl-2,4-dichloropyrimidine.

Zhihua Peng, G. Humphrey, M. Journet, 2006, Organic letters.

Radical cyclization of bromomethyldimethylsilyl propargyl ethers—VIII. Bimolecular stereoselective hydrogen abstraction by trisubstituted vinyl radicals. A new example of rare (1,4) hydrogen transfer.

M. Malacria, M. Journet, 1992 .

Radical cyclization of (bromomethyl) dimethylsilyl propargyl ethers regioselective intramolecular cyclization of vinyl radicals

M. Malacria, M. Journet, Gilbert Agnel, 1990 .

Radical cyclization of bromomethyldimethylsilyl propargyl ethers; synthesis of a carbocyclic core of steroid skeleton by a tandem radical cyclization

M. Malacria, M. Journet, S. Wu, 1994 .

Kinetic analysis and subambient temperature on-line on-column derivatization of an active aldehyde.

Y. Bereznitski, R. Lobrutto, N. Grinberg, 2003, Journal of chromatography. A.

An improved and practical procedure for the synthesis of substituted phenylacetylpyridines

D. Cai, P. Reider, M. Journet, 1998 .

Highly efficient synthesis of HIV NNRTI doravirine.

T. Itoh, I. Mangion, B. Sherry, 2015, Organic letters.

Asymmetric synthesis of telcagepant, a CGRP receptor antagonist for the treatment of migraine.

Paul N. Devine, T. Itoh, Feng Xu, 2010, The Journal of organic chemistry.

An efficient enzyme-catalyzed kinetic resolution: large-scale preparation of an enantiomerically pure indole-ethyl ester derivative, a key component for the synthesis of a prostaglandin D2 receptor antagonist, an anti-allergic rhinitis drug candidate

R. Volante, E. Corley, E. Grabowski, 2005 .

Asymmetric synthesis of a prostaglandin D2 receptor antagonist.

E. Grabowski, R. Tillyer, K. Campos, 2005, The Journal of organic chemistry.

Development of a Multikilogram Scale Synthesis of a TRPV1 Antagonist

Dalian Zhao, G. Humphrey, M. Journet, 2016 .

A New Rare Example of Cyclopropanation in Free-Radical Chemistry

M. Malacria, M. Journet, 1994 .

Radical cyclization of (bromomethyl)dimethylsilyl propargyl ethers. Regio-, chemo-, and stereoselectivity

M. Malacria, M. Journet, 1992 .

Double Radical Cyclization/β-Fragmentation of Acyclic ω-Yne Vinyl Sulfides. Synthesis of 3-Vinyldihydrothiophene and Dihydrothiopyran Derivatives. A New Example of a 5-endo-trig Radical Cyclization

D. Cai, M. Journet, R. Larsen, 1997 .

Good to excellent diastereoselectivities in asymmetric radical cyclizations of optically pure β-alkoxy vinyl sulfoxides

M. Zahouily, M. Malacria, M. Journet, 1994 .

Diastereoselective triple radical cyclization of a bromomethyldimethylsilyl allyl ether

R. Ball, N. Tsou, A. Kende, 1996 .

Acyclic diastereofacial selection in radical addition

M. Zahouily, M. Malacria, M. Journet, 1991 .

Radical Cyclization of (Bromomethyl)dimethylsilyl Propargyl Ethers; VI. Serial Radical Cyclizations Leading to a Stereoselective Synthesis of Functionalized Diquinane Framework from an Acyclic Substrate1

M. Malacria, M. Journet, W. Smadja, 1990 .

An Improved and Practical Procedure for the Synthesis of Substituted Phenylacetylpyridines.

D. Cai, P. Reider, M. Journet, 2010 .

A general method for the highly diastereoselective, kinetically controlled alkylation of ( )-nopinone

D. Cai, P. Reider, K. Campos, 2002 .

Asymmetric Synthesis of a Potent HIV-1 Integrase Inhibitor.

G. Humphrey, M. Journet, J. Kuethe, 2016, The Journal of organic chemistry.

Preparation of 4-Allylisoindoline via a Kumada Coupling with Allylmagnesium Chloride

Michael J. Zacuto, M. Journet, C. S. Shultz, 2011 .

Oral terbinafine in the treatment of toenail onychomycosis: North American multicenter trial.

J. Leyden, W. Gulliver, N. Shear, 1997, Journal of the American Academy of Dermatology.

Optimization and Scale-Up of a Lipase-Catalyzed Enzymatic Resolution of an Indole Ester Intermediate for a Prostaglandin D2 (DP) Receptor Antagonist Targeting Allergic Rhinitis

M. Truppo, M. Journet, J. C. Moore, 2006 .

Mechanistic aspects of chiral discrimination on an amylose tris(3,5-dimethylphenyl)carbamate.

P. Sajonz, Y. Bereznitski, R. Lobrutto, 2002, Enantiomer.

Functional analysis of the Pseudomonas aeruginosa autoinducer PAI

B. Iglewski, L. Passador, A. Kende, 1996, Journal of bacteriology.

Controlled semihydrogenation of aminoalkynes using ethylenediamine as a poison of Lindlar's catalyst.

D. Cai, P. Reider, K. Campos, 2001, The Journal of organic chemistry.

Radical Cyclization of Bromomethyldimethylsilyl Propargyl Ethers; a General Method for the Stereoselective Synthesis of Variously Substituted Trimethylenemethane (TMM) Precursors

M. Malacria, S. Bogen, M. Journet, 1994 .

Highly Efficient Synthesis of α,β-Acetylenic Aldehydes from Terminal Alkynes Using DMF as the Formylating Reagent.

D. Cai, M. Journet, R. Larsen, 1998 .

NOVEL AG(I)-CATALYSIS OF AN INTRAMOLECULAR 1,3-DIPOLAR CYCLOADDITION

A. Kende, M. Journet, 1995 .

Synthesis of a substance P antagonist : An efficient synthesis of 5-substituted-4-N,N-dimethylamino-1,2,3-triazoles

D. Cai, P. Reider, M. Journet, 2005 .