K. Brands

发表

Crystallization-induced diastereomer transformations.

Karel M J Brands, Antony J Davies, A. Davies, 2006, Chemical reviews.

Crystallization‐Induced Diastereomer Transformations

A. Davies, K. Brands, 2006 .

An expedient one-pot synthesis for protected 2-thia-5-azabicyclo[2.2.1]heptan-3-ones. Versatile intermediates in the synthesis of carbapenem sidechains

P. Reider, K. Brands, G. Marchesini, 1996 .

Development of a Fit-for-Purpose Large-Scale Synthesis of an Oral PARP Inhibitor

Daniel J. Muzzio, Paul Fernandez, P. Sajonz, 2011 .

The conformational bias of aryl, arylsulfonyl geminally substituted tertiary carbon centers: applications in substrate-based stereocontrol.

Jeremy P. Scott, Jennifer R. Chilenski, S. Oliver, 2006, Organic & biomolecular chemistry.

Synthesis of the homochiral “tricyclic heart” of manzamine A☆

A. Meekel, U. Pandit, K. Brands, 1991 .

Regioselective synthesis of 1,3,5-substituted pyrazoles from acetylenic ketones and hydrazines.

Andrew D. Gibb, B. Bishop, K. Brands, 2003 .

Observations on the DDQ Oxidation of 1-Acyldihydropyridines - A Synthetic Application

D. J. Wallace, Andrew D. Gibb, K. Brands, 2001 .

An efficient one-pot synthesis of annulated pyridines utilising a directed ortho-metallation/transmetallation approach

Cameron J. Cowden, A. Davies, D. Lieberman, 2004 .

Practical Asymmetric Synthesis of a Non-Peptidic αvβ3 Antagonist

Cameron J. Cowden, A. Davies, Gavin W. Stewart, 2005 .

Practical synthesis of the new carbapenem antibiotic ertapenem sodium.

D. Sidler, T. Novak, R. Skerlj, 2005, The Journal of organic chemistry.

Reaction development and mechanistic study of a ruthenium catalyzed intramolecular asymmetric reductive amination en route to the dual Orexin inhibitor Suvorexant (MK-4305).

Timothy J. Wright, R. Reamer, S. Krska, 2011, Journal of the American Chemical Society.

An efficient and stereoselective construction of the core structure of the manzamines via an intramolecular Michael reaction

K. Brands, L. Dimichele, 1998 .

MILD ARYL ETHER FORMATION IN THE SEMISYNTHESIS OF THE NOVEL MACROLIDE IMMUNOSUPPRESSANT L-732,531

J. M. Williams, K. Brands, G. Marchesini, 1998 .

Synthesis of 3-alkoxy-7,8-didehydro-4-hydroxy-N-methylmorphinan-6-ones from morphine. Intermediates for novel A- and C-ring-functionalized morphinans. (Chemistry of opium alkaloids, Part XXII)†

L. Maat, K. Brands, T. Lie, 2010 .

Regioselective Synthesis of 1,3,5‐Substituted Pyrazoles from Acetylenic Ketones and Hydrazines.

Andrew D. Gibb, B. Bishop, K. Brands, 2003 .

Practical routes to the triarylsulfonyl chloride intermediate of a β3 adrenergic receptor agonist

P. Reider, Jinchu Liu, J. Mcnamara, 2003 .

Efficient one-pot synthesis of the 2-aminocarbonylpyrrolidin-4-ylthio-containing side chain of the new broad-spectrum carbapenem antibiotic ertapenem.

P. Reider, R. Reamer, K. Conrad, 2002, The Journal of organic chemistry.

Efficient synthesis of NK(1) receptor antagonist aprepitant using a crystallization-induced diastereoselective transformation.

Jing Li, Paul N Devine, Paul N. Devine, 2003, Journal of the American Chemical Society.

Development of a General Protocol To Prepare 2H-1,3-Benzoxazine Derivatives

S. Oliver, J. Qi, K. Brands, 2017 .

Total Synthesis of (-)-Altemicidin: A Novel Exploitation of the Potier-Polonovski Rearrangement

A. Kende, Kun Liu, K. Brands, 1995 .

The First Large-Scale Synthesis of MK-4305: A Dual Orexin Receptor Antagonist for the Treatment of Sleep Disorder

R. Reamer, D. J. Wallace, Faye J. Sheen, 2011 .

Development of a Phase Transfer Catalyzed Asymmetric Synthesis for an Estrogen Receptor Beta Selective Agonist

Jeremy P. Scott, S. Oliver, Khateeta M. Emerson, 2008 .

An efficient and general synthesis of 3-substituted propionaldehydes using the Suzuki-Miyaura coupling

Cameron J. Cowden, Sarah E. Brewer, A. Davies, 2004 .

Synthesis of the “tricyclic heart” of manzamines

U. Pandit, K. Brands, 1989 .

Synthesis of an optically active tricyclic intermediate for manzamines

U. Pandit, K. Brands, 1990 .

Syntheses of morpholine-2,3-diones and 2-hydroxymorpholin-3-ones: intermediates in the synthesis of aprepitant

M. Huffman, J. Mcnamara, K. Brands, 2004 .

Regioselective synthesis of N-substituted-4-substituted isothiazolidine-1,1-dioxides

Faye J. Sheen, Ed Cleator, M. Bio, 2006 .

Regioselective Synthesis of N-Substituted-4-substituted Isothiazolidine-1,1-dioxides.

Faye J. Sheen, Ed Cleator, M. Bio, 2006 .

Practical asymmetric synthesis of aprepitant, a potent human NK-1 receptor antagonist, via a stereoselective Lewis acid-catalyzed trans acetalization reaction.

P. Reider, E. Grabowski, Guojie Ho, 2002, The Journal of organic chemistry.

Process Development and Large-Scale Synthesis of a c-Met Kinase Inhibitor

Simon E. Hamilton, Jeremy P. Scott, D. J. Wallace, 2010 .

A Practical Synthesis of a ?-Secretase Inhibitor

Jeremy P. Scott, C. McWilliams, A. Davies, 2007 .

Expedient Diels–Alder assembly of 4-aryl-4-phenylsulfonyl cyclohexanones ☆

Jeremy P. Scott, E. M. Beck, A. Davies, 2004 .

Practical asymmetric synthesis of a gamma-secretase inhibitor exploiting substrate-controlled intramolecular nitrile oxide-olefin cycloaddition.

Jeremy P. Scott, R. Reamer, S. Oliver, 2006, The Journal of organic chemistry.

A Practical and Scaleable Synthesis of 1R,5S-Bicyclo[3.1.0]hexan-2-one: The Development of a Catalytic Lithium 2,2,6,6-Tetramethylpiperidide (LTMP) Mediated Intramolecular Cyclopropanation of (R)-1,2-Epoxyhex-5-ene

Ed Cleator, M. Bio, A. Davies, 2007 .

Understanding the Origin of Unusual Stepwise Hydrogenation Kinetics in the Synthesis of the 3-(4-Fluorophenyl)morpholine Moiety of NK1 Receptor Antagonist Aprepitant

Shane W. Krska, E. Corley, R. Reamer, 2006 .

Remote substituent effects on regioselectivity in rhodium(I)-catalyzed hydroborations of norbornenes

A. Kende, K. Brands, 1992 .