Peter ‘t Hart

发表

Hot-spot guided design of macrocyclic inhibitors of the LSD1-CoREST1 interaction

H. Waldmann, H. Adihou, Peter ‘t Hart, 2019, Tetrahedron.

A combined solid- and solution-phase approach provides convenient access to analogues of the calcium-dependent lipopeptide antibiotics.

J. Kemmink, N. Martin, S. F. Oppedijk, 2014, Organic & biomolecular chemistry.

Semisynthetic Lipopeptides Derived from Nisin Display Antibacterial Activity and Lipid II Binding on Par with That of the Parent Compound.

E. Breukink, A. Hendrickx, T. Wood, 2015, Journal of the American Chemical Society.

New Insights into Nisin's Antibacterial Mechanism Revealed by Binding Studies with Synthetic Lipid II Analogues.

E. Breukink, N. Martin, S. F. Oppedijk, 2016, Biochemistry.

Development of Macrocyclic PRMT5–Adaptor Protein Interaction Inhibitors

H. Waldmann, R. Prudent, C. Peter, 2022, Journal of medicinal chemistry.

Oseltamivir analogues bearing N-substituted guanidines as potent neuraminidase inhibitors.

C. D. de Haan, N. Martin, Linda Quarles van Ufford, 2014, Journal of medicinal chemistry.

Weak coupling between magnetically inequivalent spins: The deceptively simple, complicated spectrum of a 13C-labeled trimethylated amine.

H. van Ingen, N. Martin, Peter ‘t Hart, 2017, Journal of magnetic resonance.

Peptidic Partial Bisubstrates as Inhibitors of the Protein Arginine N‐Methyltransferases

Ted M. Lakowski, Dylan Thomas, A. Frankel, 2011, Chembiochem : a European journal of chemical biology.

Nη-substituted arginyl peptide inhibitors of protein arginine N-methyltransferases.

Ted M. Lakowski, C. Ahern, A. Frankel, 2010, ACS chemical biology.

RNA-Binding Macrocyclic Peptides

Sunit Pal, Peter ‘t Hart, 2022, Frontiers in Molecular Biosciences.

Total Synthesis of Laspartomycin C and Characterization of Its Antibacterial Mechanism of Action.

E. Breukink, J. Kemmink, N. Martin, 2016, Journal of medicinal chemistry.

Rationally designed stapled peptides allosterically inhibit PTBP1–RNA-binding

Peter ‘t Hart, Joseph Openy, Gulshan Amrahova, 2023, Chemical science.

A translational repression reporter assay for the analysis of RNA-binding protein consensus sites

Benjamin C. Buchmuller, Peter ‘t Hart, D. Schiller, 2022, bioRxiv.

Semisynthetic Lipopeptides Derived from Nisin Display Antibacterial Activity and Lipid II Binding on Par with That of the Parent Compound.

E. Breukink, A. Hendrickx, T. Wood, 2015, Journal of the American Chemical Society.