Jumpei Aida

Nonbisphosphonate inhibitors of Plasmodium falciparum FPPS/GGPPS.

Stephanie C. Kabeche, Michael J. Pulkoski-Gross, Mark Smith, 2021, Bioorganic & medicinal chemistry letters.

Amine-free melanin-concentrating hormone receptor 1 antagonists: Novel 1-(1H-benzimidazol-6-yl)pyridin-2(1H)-one derivatives and design to avoid CYP3A4 time-dependent inhibition.

Masaharu Nakayama, S. Okuda, Masashi Takahashi, 2016, Bioorganic & medicinal chemistry.

Design, Synthesis, and Evaluation of [18F]T-914 as a Novel Positron-Emission Tomography Tracer for Lysine-Specific Demethylase 1.

G. Tamagnan, O. Barret, C. Sandiego, 2021, Journal of medicinal chemistry.

Amine-free melanin-concentrating hormone receptor 1 antagonists: Novel non-basic 1-(2H-indazole-5-yl)pyridin-2(1H)-one derivatives and mitigation of mutagenicity in Ames test.

Masaharu Nakayama, S. Okuda, Masashi Takahashi, 2016, Bioorganic & medicinal chemistry.

Design and Synthesis of Novel Spiro Derivatives as Potent and Reversible Monoacylglycerol Lipase (MAGL) Inhibitors: Bioisosteric Transformation from 3-Oxo-3,4-dihydro-2H-benzo[b][1,4]oxazin-6-yl Moiety.

L. Qin, S. Gay, D. Dougan, 2021, Journal of medicinal chemistry.

Melanin-Concentrating Hormone Receptor 1 Antagonists Lacking an Aliphatic Amine: Synthesis and Structure-Activity Relationships of Novel 1-(Imidazo[1,2-a]pyridin-6-yl)pyridin-2(1H)-one Derivatives.

Masaharu Nakayama, Masashi Takahashi, H. Hirabayashi, 2016, Journal of medicinal chemistry.

Design, Synthesis, and Evaluation of Piperazinyl Pyrrolidin-2-ones as a Novel Series of Reversible Monoacylglycerol Lipase Inhibitors.

M. Fushimi, S. Sogabe, Kazunobu Aoyama, 2018, Journal of medicinal chemistry.

Melanin-Concentrating Hormone Receptor 1 Antagonists Lacking an Aliphatic Amine: Synthesis and Structure-Activity Relationships of Novel 1-(Imidazo[1,2-a]pyridin-6-yl)pyridin-2(1H)-one Derivatives.

Masaharu Nakayama, Masashi Takahashi, H. Hirabayashi, 2016, Journal of Medicinal Chemistry.

Design and Identification of a GPR40 Full Agonist (SCO-267) Possessing a 2-Carbamoylphenyl Piperidine Moiety.

Mitsugi Ookawara, Masanori Watanabe, Y. Moritoh, 2020, Journal of medicinal chemistry.