W. Slusarchyk

发表

Monocyclic β-lactam antibiotics produced by bacteria

J. S. Wells, D. Floyd, K. Bush, 1981, Nature.

Solid-phase synthesis and SAR of 4-carboxy-2-azetidinone mechanism-based tryptase inhibitors.

Malcolm E. Davis, A. Mathur, G. Bisacchi, 2004, Bioorganic & medicinal chemistry letters.

Dual metalloprotease inhibitors: mercaptoacetyl-based fused heterocyclic dipeptide mimetics as inhibitors of angiotensin-converting enzyme and neutral endopeptidase.

N. Trippodo, H. Cheung, R. Misra, 1997, Journal of medicinal chemistry.

A novel series of highly potent benzimidazole-based microsomal triglyceride transfer protein inhibitors.

H. Jamil, D. Gordon, T. Harrity, 2001, Journal of medicinal chemistry.

The structure of a novel lipid from the antibiotic diumycin.

W. Slusarchyk, F. Weisenborn, J. A. Osband, 1970, Journal of the American Chemical Society.

Discovery of nonbenzamidine factor VIIa inhibitors using a biaryl acid scaffold.

D. Cheney, S. Sheriff, E. Liu, 2013, Bioorganic & medicinal chemistry letters.

Diumycin A' and diumycin B', new members of the diumycin family of antibiotics.

W. Slusarchyk, F. Weisenborn, J. L. Bouchard-Ewing, 1973, The Journal of antibiotics.

Chemical and biological aspects of a new family of phosphorus‐containing antibiotics

W. Slusarchyk, 1971, Biotechnology and bioengineering.

Mass Spectrometry in Structural and Stereochemical Problems. XXXI.1 Aporphines and Related Alkaloids2

C. Djerassi, M. Ohashi, M. Shamma, 1963 .

Synthesis of 6-methylthiopenicillins and 7-heteroatom-substituted cephalosporins.

M. Young, P. Funke, J. E. Dolfini, 1973, The Journal of organic chemistry.

BMS-200475, a novel carbocyclic 2′-deoxyguanosine analog with potent and selective anti-hepatitis B virus activity in vitro

O. Kocy, M. Young, R. Colonno, 1997 .

Synthesis of potent and highly selective nonguanidine azetidinone inhibitors of human tryptase.

A. Mathur, G. Bisacchi, W. Meng, 2004, Bioorganic & medicinal chemistry letters.

Synthesis of 2-, 4-, and 7-methylthio-substituted cephalosporins

M. Young, P. Funke, J. E. Dolfini, 1979 .

Synthesis and antiviral activity of enantiomeric forms of cyclobutyl nucleoside analogues.

T. Mitt, J. Clark, C. Cianci, 1991, Journal of medicinal chemistry.

Synthesis of SQ-33,054, a novel cyclobutane nucleoside with potent antiviral activity

M. Young, G. Bisacchi, R. Zahler, 1989 .

Synthesis of 7.alpha.-methoxycephalosporins

J. E. Dolfini, H. Applegate, M. Puar, 1974 .

Dual metalloprotease inhibitors.v. Utilization of bicyclic azepinonethiazolidines and azepinonetetrahydrothiazines in constrained peptidomimetics of mercaptoacyl dipeptides

J. Robl, J. E. Bird, W. Slusarchyk, 1995 .

4-Alkylated monobactams : Chiral synthesis and antibacterial activity

D. Floyd, R. Sykes, J. Pluščec, 1983 .

Monobactams. The conversion of 6-APA to (S)-3-amino-2-oxoazetidine-1-sulfonic acid and its 3 (RS)-methoxy derivative

M. Young, D. Floyd, H. W. Chang, 1982 .

Synthesis of 2-, 4-, and 7-methylthio-substituted cephalosporins

M. Young, P. Funke, J. E. Dolfini, 1979 .

Synthesis and SAR of 4-carboxy-2-azetidinone mechanism-based tryptase inhibitors.

G. Bisacchi, W. Meng, R. Zahler, 2002, Bioorganic & medicinal chemistry letters.

Monobactams--structure-activity relationships leading to SQ 26,776.

C. Cimarusti, W. Koster, W. Slusarchyk, 1981, The Journal of antimicrobial chemotherapy.

Deacylation of amides: removal of the acyl side-chain from cephamycin derivatives

H. Applegate, C. Cimarusti, W. Slusarchyk, 1980 .

(±)-(1α,2β,3α)-9-[2,3-bis(hydroxymethyl)cyclobutyl]guanine [(±)-BHCG or SQ 33 054]: A potent and selective inhibitor of herpesviruses

M. Young, J. Clark, K. Mazina, 1990 .

Synthesis of potent and highly selective inhibitors of human tryptase.

G. Bisacchi, W. Meng, R. Zahler, 2002, Bioorganic & medicinal chemistry letters.

The configuration and conformation of cularine

S. Roy, J. Craig, R. Manske, 1966 .

Synthesis and antiviral activity of novel isonucleoside analogs.

S. Spergel, J. Clark, J. Tino, 1993, Journal of medicinal chemistry.

Broad-spectrum antiviral activity of the acyclic guanosine phosphonate (R,S)-HPMPG.

M. Young, K. Mazina, M. Haffey, 1988, Antiviral research.

Discovery of (R)-7-cyano-2,3,4, 5-tetrahydro-1-(1H-imidazol-4-ylmethyl)-3- (phenylmethyl)-4-(2-thienylsulfonyl)-1H-1,4-benzodiazepine (BMS-214662), a farnesyltransferase inhibitor with potent preclinical antitumor activity.

S. Chong, J. Hunt, Soong-Hoon Kim, 2000, Journal of medicinal chemistry.

Synthesis and antiviral activity of 1-cyclobutyl-5-(2-bromovinyl)uracil nucleoside analogues and related compounds.

M. Young, G. Bisacchi, J. Tino, 1992, Journal of medicinal chemistry.

An MTP inhibitor that normalizes atherogenic lipoprotein levels in WHHL rabbits.

H. Jamil, C. Chu, R. Gregg, 1998, Science.

Monocyclic beta-lactam antibiotics produced by bacteria.

J. S. Wells, D. Floyd, K. Bush, 1981, Nature.

Synthesis of potent and selective 2-azepanone inhibitors of human tryptase.

G. Bisacchi, C. Kwon, S. Bolton, 2004, Bioorganic & medicinal chemistry letters.

Synthesis of mercury mercaptide azetidinones via 2- and 4-methylthio-substituted cephalosporins

J. E. Dolfini, H. Applegate, M. Puar, 1978 .

7-[2-hydroxyethyl] cephalosporanic acid derivatives

H. Applegate, C. Cimarusti, W. Slusarchyk, 1979 .

The structure of the lipid portion of the antibiotic prasinomycin.

W. Slusarchyk, F. Weisenborn, 1969, Tetrahedron letters.

The Aporphine Alkaloids

M. Shamma, W. Slusarchyk, 1964 .

Diastereomeric 7-ureidoacetyl cephalosporins. II. 7beta [[[(Aminocarbonyl) amino]-2-thienylacetyl] amino]-7-methoxy-3-[[(1-methyl-1H-tetrazol-5-yl) thio] methyl]-8-oxo-5-thia-1-azabicyclo [4.2.0] oct-2-ene-2-carboxylic acid.

M. Young, M. Ondetti, J. E. Dolfini, 1978, Journal of antibiotics (Tokyo. 1968).

Discovery and structure-activity relationships of imidazole-containing tetrahydrobenzodiazepine inhibitors of farnesyltransferase.

J. Hunt, V. Manne, C. Ricca, 1999, Journal of medicinal chemistry.

The problem of the 1,2,9,10-tetraoxygenated aporphines and the structure of the quaternary aporphine from Fagara tinguassoiba.

M. Shamma, W. Slusarchyk, 1967, Tetrahedron.

The problem of the 1,2,9,10-tetraoxygenated aporphines and the synthesis of (±)-1-hydroxy-2,9,10-trimethoxyaporphine

M. Shamma, W. Slusarchyk, 1965 .

The synthesis of glaucine, O-methylcorydine, and pseudocorydine via phenolic oxidative coupling

M. Shamma, W. Slusarchyk, 1965 .

Broad-spectrum antiviral activity of the acyclic guanosine phosphonate (R,S)-HPMPG.

M. Young, K. Mazina, M. Haffey, 1988, Antiviral research.