Jordi Castro

发表

Structure-activity relationships (SAR) and structure-kinetic relationships (SKR) of bicyclic heteroaromatic acetic acids as potent CRTh2 antagonists I.

M. Calbet, M. Zanuy, P. Eichhorn, 2014, Bioorganic & medicinal chemistry letters.

Structure-activity relationships (SAR) and structure-kinetic relationships (SKR) of bicyclic heteroaromatic acetic acids as potent CRTh2 antagonists III: the role of a hydrogen-bond acceptor in long receptor residence times.

M. Calbet, E. Gómez, R. S. Roberts, 2014, Bioorganic & medicinal chemistry letters.

Discovery of novel quaternary ammonium derivatives of (3R)-quinuclidinyl amides as potent and long acting muscarinic antagonists.

S. Espinosa, A. Gavaldá, V. Segarra, 2011, Bioorganic & medicinal chemistry letters.

Discovery of novel quaternary ammonium derivatives of (3R)-quinuclidinol esters as potent and long-acting muscarinic antagonists with potential for minimal systemic exposure after inhaled administration: identification of (3R)-3-{[hydroxy(di-2-thienyl)acetyl]oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[

S. Sentellas, S. Espinosa, V. Segarra, 2009, Journal of medicinal chemistry.

2-(1H-Pyrazol-1-yl)acetic acids as chemoattractant receptor-homologous molecule expressed on Th2 lymphocytes (CRTh2) antagonists.

M. Lehner, M. Calbet, P. Eichhorn, 2014, European journal of medicinal chemistry.

2-(1H-Pyrazol-4-yl)acetic acids as CRTh2 antagonists.

M. Lehner, M. Calbet, P. Eichhorn, 2013, Bioorganic & medicinal chemistry letters.

Structure-activity relationships (SAR) and structure-kinetic relationships (SKR) of sulphone-based CRTh2 antagonists.

M. Calbet, R. S. Roberts, P. Forns, 2016, European journal of medicinal chemistry.

Discovery of novel quaternary ammonium derivatives of (3R)-quinuclidinyl carbamates as potent and long acting muscarinic antagonists.

S. Espinosa, V. Segarra, J. Beleta, 2011, Bioorganic & medicinal chemistry letters.

Biphenyl Pyridazinone Derivatives as Inhaled PDE4 Inhibitors: Structural Biology and Structure-Activity Relationships.

M. Lehner, V. Segarra, P. Eichhorn, 2016, Journal of medicinal chemistry.

Structure-activity relationships (SAR) and structure-kinetic relationships (SKR) of pyrrolopiperidinone acetic acids as CRTh2 antagonists.

M. Calbet, P. Eichhorn, R. S. Roberts, 2014, Bioorganic & medicinal chemistry letters.