R. Chakrasali

发表

Allosteric Indole Amide Inhibitors of p97: Identification of a Novel Probe of the Ubiquitin Pathway.

Vsevolod A. Peshkov, F. Zhang, P. Wipf, 2016, ACS medicinal chemistry letters.

Gamendazole, an orally active indazole carboxylic acid male contraceptive agent, targets HSP90AB1 (HSP90BETA) and EEF1A1 (eEF1A), and stimulates Il1a transcription in rat Sertoli cells.

T. Kinzy, B. Blagg, G. Georg, 2008, Biology of reproduction.

A novel potent indazole carboxylic acid derivative blocks spermatogenesis and is contraceptive in rats after a single oral dose.

G. Georg, Sudhakar R. Jakkaraj, J. Tash, 2008, Biology of reproduction.

Characterization of novel competitive inhibitors of P. falciparum cGMP-dependent protein kinase

N. Goodey, P. Bhanot, J. Siekierka, 2021, bioRxiv.

Cyclocondensation of α-hydroxyimino-β-alkyl/arylimino-β-methylthioketones with hydrazine hydrate: synthesis of 3(5)-aryl-5(3)-alkyl/arylamino-4-nitroso (or amino) pyrazoles

H. Ila, R. Chakrasali, H. Junjappa, 1993 .

Reaction of polarized ketene S,N-acetals with bromoacetaldehyde diethyl acetal: synthesis of 1-substituted 3-acyl- and 3-nitro-2-methylthiopyrroles and 1,2-annulated 3-acylpyrroles

H. Ila, R. Chakrasali, H. Junjappa, 1989 .

Reaction of acylketene S,N-acetals with malonyl chloride: synthesis of novel 1,5-substituted 4-hydroxy-6-methylthio-2(1H)-pyridones and 6,8-substituted 4-hydroxy-7-methylthio-2,5-dioxo-5,6-dihydro-2H-pyrano[3,2-c]pyridines

H. Ila, R. Chakrasali, H. Junjappa, 1988 .

Cycloaddition of Sodium Azide to Polarized Ketene S,S- and S,N-Acetals: Synthesis of Novel Substituted Triazole and Tetrazole Derivatives

H. Ila, R. Chakrasali, H. Junjappa, 1988 .

Cycloaddition of Aroyl/Acylketene S,N-Acetals with Tosyl Azide: Synthesis of Novel 4-Aroyl/Acyl-5-amino-1H-1,2,3-triazoles and 3,4-Annulated 1,2,3-Triazoles

H. Ila, R. Chakrasali, H. Junjappa, 1988 .

Development of highly potent and selective diaminothiazole inhibitors of cyclin-dependent kinases.

A. Becker, C. Cubitt, Huijong Han, 2013, Journal of medicinal chemistry.

Regio- and chemoselective conjugate 1,4-reduction of α-oxoketene dithioacetals with sodium borohydride and sodium cyanoborohydride

H. Ila, R. Chakrasali, H. Junjappa, 1990 .

Development of highly potent and selective diaminothiazole inhibitors of cyclin-dependent kinases.

A. Becker, C. Cubitt, Huijong Han, 2013, Journal of Medicinal Chemistry.

A novel potent indazole carboxylic acid derivative blocks spermatogenesis and is contraceptive in rats after a single oral dose.

Sudhakar R. Jakkaraj, J. Tash, B. Attardi, 2008, Biology of reproduction.