G. Papeo

发表

A Submarine Journey: The Pyrrole-Imidazole Alkaloids †

C. Piutti, B. Malgesini, B. Forte, 2009, Marine drugs.

Italian Chemists’ Contributions to Named Reactions in Organic Synthesis: An Historical Perspective †

M. Pulici, G. Papeo, 2013, Molecules.

A new glycociamidine ring precursor: syntheses of (Z)-hymenialdisine, (Z)-2-debromohymenialdisine, and (+/-)-endo-2-debromohymenialdisine.

D. Borghi, M. Varasi, G. Papeo, 2005, Organic letters.

Poly(ADP-ribose) polymerase inhibition in cancer therapy: are we close to maturity?

A. Montagnoli, P. Orsini, B. Forte, 2009, Expert opinion on therapeutic patents.

Asymmetric Synthesis of 4(R)Tert-Butyl-8a(S)Hydroxycarbonyl-4,6,7,8,8a,9-Hexahydro-1-Alkyl-Pyrrolo[3,2-f]Indolizines via Intramolecular Iminium Ion Cyclization

M. Resmini, M. Sisti, R. Annunziata, 1997 .

Use of acridinium-based photocatalyst in the Giese-type coupling of arylboronic acids with electron poor olefins

M. De Amici, M. Caldarelli, G. Papeo, 2022, Tetrahedron Letters.

MutT Homolog 1 (MTH1): The Silencing of a Target.

G. Papeo, 2016, Journal of medicinal chemistry.

PARP inhibitors in cancer therapy: an update

E. Casale, A. Montagnoli, A. Cirla, 2013, Expert opinion on therapeutic patents.

Design of β-amino alcohols as chiral auxiliaries in the electrophilic amination of 1,3,2-oxazaphospholanes

G. Sello, M. Sisti, L. Paleari, 1996 .

Stereoselective synthesis of (Z)-axino- and (Z)-debromoaxinohydantoin

D. Borghi, N. Mongelli, F. Quartieri, 2009 .

Oxindole alkaloids. A novel non-biomimetic entry to (−)-Horsfiline.

G. Palmisano, M. Sisti, R. Annunziata, 1996 .

Synthesis of functionally diverse and conformationally constrained polycyclic analogues of proline and prolinol.

S. Hanessian, M. Angiolini, M. Beretta, 2003, The Journal of organic chemistry.

A straightforward total synthesis of (-)-chaetominine.

D. Borghi, B. Malgesini, C. Gennari, 2009, Chemistry.

Total synthesis of (±)-cyclooroidin

D. Borghi, M. Varasi, G. Papeo, 2005 .

Synthesis of 7,5-fused bicyclic lactams by stereoselective radical cyclization

O. Carugo, L. Manzoni, C. Scolastico, 1994 .

Design of β-Amino Alcohols as Chiral Auxiliaries in the Electrophilic Amination of 1,3,2-Oxazaphospholanes.

G. Sello, M. Sisti, L. Paleari, 1997 .

Total Synthesis of (+)‐7,11‐Helianane and (+)‐5‐Chloro‐7,11‐helianane through Stereoselective Aromatic Claisen Rearrangement

D. Borghi, C. Gennari, F. Quartieri, 2011 .

Oxindole Alkaloids. A Novel Non-Biomimetic Entry to (-)-Horsfiline.

G. Palmisano, M. Sisti, R. Annunziata, 1996 .

Synthesis of 3 10-helix-inducing constrained analogues of L-proline.

Eric Therrien, S. Hanessian, G. Papeo, 2004, The Journal of organic chemistry.

Polyfluorinated amino acids for sensitive 19F NMR-based screening and kinetic measurements.

Nicola Mongelli, Anna Vulpetti, Marina Veronesi, 2007, Journal of the American Chemical Society.

Sensitivity improvement in 19F NMR-based screening experiments: theoretical considerations and experimental applications.

Nicola Mongelli, Detlef Moskau, Rainer Kümmerle, 2005, Journal of the American Chemical Society.

Rapid NMR‐based functional screening and IC50 measurements performed at unprecedentedly low enzyme concentration

Nicola Mongelli, Marina Veronesi, Claudio Dalvit, 2005 .

Synthesis of a preclavulones analogous : (±) 8,12-trans-(5Z, 14Z)-9-oxo-prosta-5,10,14-trienoic acid methyl ester via its 10-11 dihydroprecursor from allyl 2-oxo-cyclopentanecarboxylate

G. Papeo, D. Pirillo, M. D. Giacomo, 1993 .

Nicotinoyl azide (NCA)-mediated Mitsunobu reaction: An expedient one-pot transformation of alcohols into azides

M. Varasi, P. Vianello, G. Papeo, 2004 .

Discovery and optimization of pyrrolo[1,2-a]pyrazinones leads to novel and selective inhibitors of PIM kinases.

E. Casale, E. Felder, A. Galvani, 2013, Bioorganic & medicinal chemistry.

Discovery of 2-[1-(4,4-Difluorocyclohexyl)piperidin-4-yl]-6-fluoro-3-oxo-2,3-dihydro-1H-isoindole-4-carboxamide (NMS-P118): A Potent, Orally Available, and Highly Selective PARP-1 Inhibitor for Cancer Therapy.

Antonella Isacchi, Enrico Pesenti, Fabio Zuccotto, 2015, Journal of medicinal chemistry.

Identification of soyasaponins by liquid chromatography–thermospray mass spectrometry

N. Fuzzati, R. Pace, F. Peterlongo, 1997 .

Discovery of Stereospecific PARP-1 Inhibitor Isoindolinone NMS-P515.

A. Isacchi, E. Casale, E. Felder, 2019, ACS medicinal chemistry letters.

Stereoselective synthesis of 3,4-dihydropyrrolo[1,2-a]pyrazin-1(2H)-one derivatives as PIM kinase inhibitors inspired from marine alkaloids.

A. Isacchi, E. Casale, E. Felder, 2022, Chirality.

Improved synthesis of polyfluorinated l-lysine for 19F NMR-based screening

E. Felder, B. Malgesini, N. Mongelli, 2009, Molecular Diversity.

A Submarine Journey: The Pyrrole‐—Imidazole Alkaloids

B. Malgesini, B. Forte, F. Quartieri, 2010 .

Insights into PARP Inhibitors’ Selectivity Using Fluorescence Polarization and Surface Plasmon Resonance Binding Assays

A. Montagnoli, A. Leone, N. Avanzi, 2014, Journal of biomolecular screening.

Photocatalytic Radical Coupling of Organoborates with α-Halogenated Electron-Poor Olefins.

T. Pirali, G. Papeo, N. Colombo, 2023, The Journal of organic chemistry.