Anamika Singh

发表

Structure-activity relationships of peptides incorporating a bioactive reverse-turn heterocycle at the melanocortin receptors: identification of a 5800-fold mouse melanocortin-3 receptor (mMC3R) selective antagonist/partial agonist versus the mouse melanocortin-4 receptor (mMC4R).

A. Edison, J. Rocca, C. Haskell-Luevano, 2013, Journal of medicinal chemistry.

Incorporation of a bioactive reverse-turn heterocycle into a peptide template using solid-phase synthesis to probe melanocortin receptor selectivity and ligand conformations by 2D 1H NMR.

A. Edison, C. Haskell-Luevano, M. Dirain, 2011, Journal of medicinal chemistry.

Structure-activity relationships (SAR) of melanocortin and agouti-related (AGRP) peptides.

C. Haskell-Luevano, Erica M. Haslach, Anamika Singh, 2010, Advances in experimental medicine and biology.

Synthesis and Structure-Activity Relationships of Substituted Urea Derivatives on Mouse Melanocortin Receptors.

C. Haskell-Luevano, Huisuo Huang, M. Dirain, 2016, ACS chemical neuroscience.

1,2,3-Triazole Rings as a Disulfide Bond Mimetic in Chimeric AGRP-Melanocortin Peptides: Design, Synthesis, and Functional Characterization.

J. Rocca, Cody J Lensing, K. Freeman, 2017, ACS chemical neuroscience.

1,4-Disubstituted-[1,2,3]triazolyl-Containing Analogues of MT-II: Design, Synthesis, Conformational Analysis, and Biological Activity

Manuela Grimaldi, Paolo Rovero, Chiara Testa, 2014, Journal of medicinal chemistry.

Synthesis and Pharmacology of α/β(3)-Peptides Based on the Melanocortin Agonist Ac-His-dPhe-Arg-Trp-NH2 Sequence.

K. Freeman, C. Haskell-Luevano, S. R. Tala, 2015, ACS medicinal chemistry letters.

Human β-Defensin 1 and β-Defensin 3 (Mouse Ortholog mBD14) Function as Full Endogenous Agonists at Select Melanocortin Receptors.

Mark D. Ericson, R. Speth, B. Smeester, 2018, Journal of medicinal chemistry.

1,4-Disubstituted-[1,2,3]triazolyl-Containing Analogues of MT-II: Design, Synthesis, Conformational Analysis, and Biological Activity

M. Scrima, M. Grimaldi, A. D'Ursi, 2014, Journal of Medicinal Chemistry.

Microwave-assisted preparations of amidrazones and amidoximes.

A. Katritzky, N. Khashab, N. Kirichenko, 2006, The Journal of organic chemistry.

A new and facile route for the synthesis of chiral 1,2-diamines and 2,3-diamino acids

Anamika Singh, U. K. Nadir, R. Krishna, 2005 .

Microwave-induced clay-catalyzed ring opening of N-tosylaziridines: a green approach to achiral and chiral diamines

Anamika Singh, U. K. Nadir, 2005 .

Biguanidines, gunaylureas and guanylthioureas

A. Katritzky, S. R. Tala, Anamika Singh, 2010 .

Synthesis of Functionalized N‐Arylsulfonyl Aziridines from α,β‐Unsaturated Esters, Amides, Ketones, and Nitriles Using N,N‐Dichloroarylsulfonamides as Nitrogen Source

Anamika Singh, U. K. Nadir, 2004 .

Biguanidines, Guanylureas and Guanylthioureas

A. Katritzky, S. R. Tala, Anamika Singh, 2010 .

Synthesis and antimicrobial activity of Schiff's and Mannich bases of 1H-indole-2,3-dione derivatives.

Ey, P. Manoj, P. Surendran, 2010 .

Synthesis, Biophysical, and Pharmacological Evaluation of the Melanocortin Agonist AST3-88: Modifications of Peptide Backbone at Trp 7 Position Lead to a Potent, Selective, and Stable Ligand of the Melanocortin 4 Receptor (MC4R)

A. Levine, A. Edison, B. Gosnell, 2014, ACS chemical neuroscience.

Design, Synthesis, Conformational Analysis, and Biological Activity

M. Scrima, M. Grimaldi, A. Papini, 2014 .