J. Mérour

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Recent advances in the synthesis and properties of 4-, 5-, 6- or 7-azaindoles

S. Routier, F. Suzenet, B. Joseph, 2013 .

Reactions of 3‐oxo‐2,3‐dihydrobenzofuran with alkyl 2‐cyano‐3‐alkoxypropenoate and alkyl 2‐alkoxycarbonyl‐3‐alkoxypropenoate. Synthesis of pyran derivatives

F. Cossais, J. Mérour, 1991 .

Reactions 1‐acetyl‐3‐oxo‐2,3‐dihydroindole with alkyl 2‐cyano‐3‐alkoxypropenoate and alkyl 2‐alkoxycarbonyl‐3‐alkoxy‐propenoate. Synthesis of 9‐acetoxypyrrolo[1,2‐a]indol‐3‐one derivatives

J. Mérour, S. Piroelle, 1991 .

The Chemistry of Sulfur-Containing [5,5]-Fused Ring Systems With a Bridgehead Nitrogen

S. Routier, F. Buron, Marie-Aude Hiebel, 2018 .

Synthesis of Substituted Azepino[3,4-b]indole-1,5-diones

B. Joseph, J. Mérour, Julien Perron, 2004 .

Novel 5-azaindolocarbazoles as cytotoxic agents and Chk1 inhibitors.

B. Pfeiffer, J. Hickman, R. Golsteyn, 2008, Bioorganic & medicinal chemistry.

Synthesis of 4-substituted azepino[3,4-b]indole-1,5-diones

B. Joseph, J. Mérour, Julien Perron, 2003 .

Synthesis of Pyrido[2,3-b]indole Derivatives via Diels–Alder Reactions of 2- and 3-Vinylpyrrolo[2,3-b]pyridines

B. Joseph, S. Léonce, J. Mérour, 2000 .

DNA interaction and cytotoxicity of a new series of indolo[2,3-b]quinoxaline and pyridopyrazino[2,3-b]indole derivatives.

C. Bailly, P. Colson, C. Houssier, 2001, Chemico-biological interactions.

Mild and selective deprotection of carbamates with Bu4NF

S. Routier, Ulrich Jacquemard, J. Mérour, 2004 .

Convenient access to C-2 or C-5 substituted 4-azaindole derivatives

F. Saab, F. Schoentgen, S. Routier, 2010 .

Ring closure metathesis of indole 2-carboxylic acid allylamide derivatives

B. Joseph, J. Mérour, V. Bénéteau, 2002 .

Synthesis of benzo analogs of oxoarcyriaflavins and caulersine

S. Routier, J. Mérour, Aurélie Bourderioux, 2007 .

Intramolecular heck reaction: synthesis of potential antiinflammatory agents

B. Joseph, J. Mérour, O. Cornec, 1995 .

Synthesis and biological evaluation of novel phenylcarbazoles as potential anticancer agents.

L. Meijer, C. Bailly, O. Lozach, 2006, Journal of medicinal chemistry.

Synthesis of diphenylcarbazoles as cytotoxic DNA binding agents.

C. Bailly, J. Kluza, S. Routier, 2004, Organic & biomolecular chemistry.

Recent advances in the chemistry and biology of pyridopyrimidines.

M. Akssira, S. Routier, G. Guillaumet, 2015, European journal of medicinal chemistry.

Access to ring-fused azepino[3,4-b]indole-1,5-dione derivatives by ring-closing olefin metathesis

B. Joseph, J. Mérour, Julien Perron, 2004 .

Tetrahedron report number 808 Synthesis and reactivity of 4-, 5- and 6-azaindoles

F. Popowycz, B. Joseph, J. Mérour, 2007 .

Synthesis and Reactivity of 7-Azaindole (1H-Pyrrolo[2,3-b]pyridine)

F. Popowycz, S. Routier, B. Joseph, 2001 .

The Azaindole Framework in the Design of Kinase Inhibitors

P. Bonnet, S. Routier, F. Buron, 2014, Molecules.

Synthesis and Reactivity of 4-, 5- and 6-Azaindoles.

F. Popowycz, B. Joseph, J. Mérour, 2007 .

A New Synthesis of 2,3,4-Substituted Quinolines

J. Mérour, F. Tatibouët, 1978 .

Reactions of substituted 2,3-dihydro-1 H -indol-3-ones and pyrrolo[2,3- b ]pyridin-3-ones with Wittig and Horner–Emmons reagents: synthesis of 7-azatryptamine

J. Mérour, P. Gadonneix, E. Desarbre, 2001 .

Synthesis of 2-Substituted-1H-pyrrolo[2,3-b]pyridines: Preparation of 7-azaolivacine analogue and 7-azaindolopyridopyrimidine derivatives

J. Mérour, E. Desarbre, Sandrine Coudret, 1997 .

Convenient Synthesis of 8-Substituted 9H-Dipyrido[3,2-b:3‘,2‘-d]pyrrole (6-Aza-δ-carbolines)

J. Mérour, E. Desarbre, 1997 .

Palladium heteroannulation process for synthesis of substituted pyrrolo[2,3-b]pyridin-3-ones

J. Mérour, E. Desarbre, 1996 .

Synthesis and Reactivity of 7-Azaindoles: 1H-Pyrrolo[2,3- B]pyridines

B. Joseph, J. Mérour, 2001 .

Synthesis and biological evaluation of 7-azaindolocarbazoles

C. Bailly, P. Renard, B. Pfeiffer, 2002 .

First synthesis of symmetrical and non-symmetrical aza indolocarbazoles derivatives

S. Routier, D. Caignard, J. Mérour, 2002 .

Synthesis of Indolo[3,2-c]quinoline and Pyrido[3′,2′ : 4,5] [3,2-c]quinoline Derivatives

A. Mouaddib, B. Joseph, J. Mérour, 2000 .

A mild and selective method for N-Boc deprotection

S. Routier, J. Mérour, G. Coudert, 2002 .

Design and synthesis of a series of indole glycoprotein IIb/IIIa inhibitors.

G. Guillaumet, A. Frydman, B. Lesur, 2002, European journal of medicinal chemistry.

Synthesis and biological evaluation of new 2-(4,5-dihydro-1H-imidazol-2-yl)-3,4-dihydro-2H-1,4-benzoxazine derivatives.

P. Renard, M. Rettori, B. Pfeiffer, 2003, Journal of medicinal chemistry.

Attempted synthesis of ethyl 3,4‐dihydro‐2H‐1,4‐benzoxazine‐3‐carboxylate and 3‐acetate derivatives

G. Guillaumet, Stanislas Mayer, J. Mérour, 2001 .

New substituted 1,4-benzoxazine derivatives with potential intracellular calcium activity.

A. Monteil, G. Guillaumet, M. D. Pujol, 1998, Journal of medicinal chemistry.

Synthesis and Reactions of 1-Acetyl-2-benzylidene-3-oxo-2,3-dihydroindoles

J. Mérour, A. Buzas, 1989 .

A Straightforward Synthesis of Pyridopyrazino[2,3-b]indoles and Indolo[2,3-b]quinoxaline

A. P. Nikalje, S. Routier, J. Mérour, 2001 .

Synthesis and biological evaluation of novel naphthocarbazoles as potential anticancer agents.

P. Peixoto, C. Bailly, D. Caignard, 2005, Journal of medicinal chemistry.

Intramolecular Heck Coupling of Alkenyl 3-Iodoindole-2-carboxamide Derivatives

B. Joseph, J. Mérour, L. Chacun-Lefevre, 2001 .

Synthesis of naphthopyrrolo[3,4-c]carbazoles

S. Routier, J. Mérour, G. Coudert, 2001 .

Insertion d'allenes

J. Beňa, J. Mérour, C. Charrier, 1979 .

Insertion d'allenes: I. Reactions de cyclisation de complexes du fer η1-alkyl-γ-alleniques en η3-allylcyclopentenones. Discussion de l'etape d'insertion

J. Benaim, J. Mérour, C. Charrier, 1979 .

Synthesis and biological evaluation of new 3-(6-hydroxyindol-2-yl)-5-(Phenyl) pyridine or pyrazine V-Shaped molecules as kinase inhibitors and cytotoxic agents.

L. Meijer, O. Lozach, C. Guillouzo, 2011, European journal of medicinal chemistry.

Synthesis of 2,6-diphenylpyrazine derivatives and their DNA binding and cytotoxic properties.

C. Bailly, J. Goossens, N. Dias, 2005, European journal of medicinal chemistry.

Synthesis of indolo[1,2-b]isoquinolinediones; reduction of 2-[(substituted phenyl)methylidene]-3-oxo-2,3-dihydroindole

F. Cossais, J. Mérour, S. Piroelle, 1993 .

Synthesis of new fused and substituted benzo and pyrido carbazoles via C-2 (het)arylindoles

S. Routier, J. Mérour, Aurélie Bourderioux, 2008 .

A Straightforward Synthesis of 1,2-Dihydronaphtho[2,1-b]furans from 2-Naphthols

G. Guillaumet, J. Mérour, Axelle Arrault, 1999 .

Synthesis of 3,5-bis(2-indolyl)pyridine and 3-[(2-indolyl)-5-phenyl]pyridine derivatives as CDK inhibitors and cytotoxic agents.

L. Meijer, C. Bailly, O. Lozach, 2008, Bioorganic & medicinal chemistry.

Oxidation of indoles and 1,2-dihydro-3H-indol-3-ones

J. Mérour, E. Desarbre, L. Savelon, 1996 .

Synthesis and in vitro cytotoxic evaluation of N-substituted benzo[5,6]cycloheptal[b]indoles.

D. Alagille, B. Joseph, S. Léonce, 2000, Chemical & pharmaceutical bulletin.

Synthesis and Antitumoral Evaluation of 12-Substituted 6,7-Dihydrobenzo[4,5]-cyclohept[1,2-b]indole Derivatives

B. Joseph, S. Léonce, J. Mérour, 1998 .

Synthesis, cytotoxicity, DNA interaction and topoisomerase II inhibition properties of tetrahydropyrrolo[3,4-a]carbazole-1,3-dione and tetrahydropyrido-[3,2-b]pyrrolo[3,4-g]indole-1,3-dione derivatives.

C. Bailly, P. Colson, C. Houssier, 2001, Bioorganic & medicinal chemistry.

Synthesis and biological evaluation of novel oxophenylarcyriaflavins as potential anticancer agents.

C. Bailly, C. Guillouzo, R. le Guével, 2008, Organic & biomolecular chemistry.

Preparation and reactivity of 5-substituted azepino[3,4-b]indoles

B. Joseph, N. Laurent, J. Mérour, 2005 .

Synthesis and Reactivity of Azepino[3,4-b]indol-5-yl Trifluoromethanesulfonate

B. Joseph, J. Mérour, L. Chacun-Lefevre, 2000 .

Synthesis and biological activities of new furo[3,4-b]carbazoles: potential topoisomerase II inhibitors.

C. Bailly, S. Routier, E. Vedrenne, 2010, European journal of medicinal chemistry.

A Convenient Synthesis of Tryptamines

J. Mérour, A. Buzas, 1988 .

Synthesis of chromeno[3,4-b]indoles as Lamellarin D analogues: a novel DYRK1A inhibitor class.

L. Meijer, O. Lozach, S. Routier, 2012, European journal of medicinal chemistry.

First synthesis of pyrrolo[1,2:1′,2′]azepino[5,6-b]indole derivatives

B. Joseph, J. Mérour, Julien Perron, 2003 .

Synthesis of functionalised pyrido[4,3-b][1,4]oxazine and imidazo[1,2-a]pyridine derivatives

J. Leger, C. Jarry, G. Guillaumet, 2002 .

Attempted Synthesis of Ethyl 3,4‐Dihydro‐2H‐1,4‐benzoxazine‐3‐carboxylate and 3‐Acetate Derivatives.

G. Guillaumet, Stanislas Mayer, J. Mérour, 2001 .

A Straightforward Route to 4H‐1,4‐Benzoxazine‐2‐carbaldehydes by Swern Oxidation.

G. Guillaumet, J. Mérour, A. Bourlot, 1996 .

3D-QSAR CoMFA study on imidazolinergic I(2) ligands: a significant model through a combined exploration of structural diversity and methodology.

L Morin-Allory, P. Renard, C. Marot, 2000, Journal of medicinal chemistry.

A straightforward route to 4H‐1,4‐Benzoxazine‐2‐carbaldehydes by swern oxidation

G. Guillaumet, J. Mérour, A. Bourlot, 1996 .

Stereoselective addition reactions to chiral N-benzylidene-p-toluenesulfinamides. Application to the synthesis of optically active 1,2-diphenylethylamines

P. Moreau, J. Mérour, D. Bouzard, 1997 .

Intramolecular Heck reaction: Synthesis of benzo[4,5]cyclohepta[b]indole derivatives

B. Joseph, J. Mérour, O. Cornec, 1998 .

PALLADIUM-CATALYZED REACTIONS OF INDOLIC TRIFLATE WITH ALLYLIC ALCOHOLS

J. Mérour, Béatrice Malapel-Andrieu, 1998 .

Synthesis of 6-Substituted 5,6,7,12-Tetrahydrobenzo[4,5]cyclohept[b]indol-12-one Derivatives

A. Mouaddib, B. Joseph, S. Léonce, 1999 .

Synthesis and reactivity of substituted 3-([(Trifluoromethyl)sulfonyl]oxy)-1H-indole-2-carboxylate in palladium-catalyzed reactions

J. Mérour, Béatrice Malapel-Andrieu, 1998 .

Syntheses of 2-spiroindoles and pyrrolof[1,2-a]indoles

J. Mérour, B. M. and, 1998 .

Synthesis and reactivity of 1-substituted-3H-pyrrolo[2,3-b] pyridin-3-one

J. Mérour, E. Desarbre, 1994 .

Synthesis and Reactions of 1-Acetyl-2-benzylidene-3-oxo-2,3-dihydroindoles.

J. Mérour, A. Buzas, 1989 .

Synthesis of Substituted 1,4-Benzoxazepin-3-one Derivatives

J. Leger, C. Jarry, G. Guillaumet, 2004 .

Synthesis and Reactivity of (3-Oxo-2,3-dihydro-1H-ylidene)acetic Acid Alkyl Esters in Diels-Alder Reactions

J. Mérour, P. Gadonneix, E. Desarbre, 1996 .

A Straightforward Synthesis of Pyridopyrazino[2,3-b]indoles and Indolo[2,3-b]quinoxaline.

S. Routier, J. Mérour, G. Coudert, 2001 .

Regioselective Formylation of Ethyl 3,4-Dihydro-2H-1,4- benzoxazine-2-carboxylate or 2-Acetate Derivatives

G. Guillaumet, Stanislas Mayer, J. Mérour, 2001 .

Synthesis of 2,5- and 3,5-diphenylpyridine derivatives for DNA recognition and cytotoxicity.

C. Bailly, J. Goossens, N. Dias, 2005, European journal of medicinal chemistry.

Targeting DNA with novel diphenylcarbazoles.

Christian Bailly, C. Bailly, P. Colson, 2004, Biochemistry.

A convenient synthesis of 1,2-dihydro-3H-indol-3-ones and 1,2-dihydro-2H-indol-2-ones by Baeyer-Villiger oxidation

J. Mérour, E. Desarbre, A. Bourlot, 1994 .

New synthesis of (±)-2-piperazinecarboxylic acid.

J. Mérour, J. Y. Coadou, 1991 .

1-(Phenylsulfonyl)indol-2-yl Triflate: A Versatile Reagent for the Synthesis of 2-Substituted Indoles

B. Joseph, J. Mérour, Béatrice Malpel, 1996 .

Synthesis and reactivity of iron nitrosyl hydrides substituted with triphenyl phosphine

N. D. Venayak, J. Mérour, J. Roustan, 1983 .

Reactions of 3-([(trifluoromethyl)sulfonyl]oxy)-1H-indole derivatives with diamines and carbon nucleophiles. Synthesis of 6H-indolo[2,3-b]quinoxaline derivatives

J. Mérour, Béatrice Malapel-Andrieu, 1998 .

Reactions of 3‐([(Trifluoromethyl)sulfonyl]oxy)‐1H‐indole Derivatives with Diamines and Carbon Nucleophiles. Synthesis of 6H‐Indolo[2,3‐b]quinoxaline Derivatives.

J. Mérour, Béatrice Malapel-Andrieu, 1998 .

Synthesis and Reactivity of 1,4‐Oxazinoindole Derivatives

G. Guillaumet, B. Joseph, Stanislas Mayer, 2002 .

Arylation of 3-Oxo-2,3-Dihydroindoles with aryllead Triacetates

J. Mérour, J. Finet, L. Chichereau, 1992 .

Unusual schmidt rearrangement of 7,7a,8,9,10,12‐hexahydro benzo[h]pyrrolo[1,2‐b]‐isoquinoline‐7,10‐dione

R. Faure, J. Mérour, S. Piroelle, 1994 .

Synthesis of 6,7-dihydrobenzo[4,5]cyclohept-[1,2-b]indol-12(5H)-one and related compounds

X. Solans, B. Joseph, M. Font‐Bardia, 1997 .

Synthesis of Pyrano[3,2-b]indole Derivatives Based on Intramolecular Hetero-DielsAlder of 2-Benzylidene-2,3-dihydro-1H-indol-3-ones

J. Leger, C. Jarry, B. Joseph, 2003 .

Synthesis of benzo[5,6]cyclohepta[b]indol-6-one derivatives

D. Alagille, B. Joseph, C. Rousseau, 1999 .

ALKYLATION OF METHYL 3-HYDROXYINDOLE-2-CARBOXYLATE USE IN PYRIMIDINE SYNTHESIS

J. Mérour, A. Bourlot, 1995 .

First efficient synthesis of novel oxophenyl-arcyriaflavin analogs

S. Routier, J. Mérour, Aurélie Bourderioux, 2005 .

Comparison of the efficiencies of two TR-FRET methods to detect in vitro natural and synthesized inhibitors of the Raf/MEK/ERK signaling pathway

F. Saab, F. Schoentgen, S. Routier, 2010 .

Claisen Rearrangement of 2-Allyloxyindolic Ketoester via a Decarboxylative Process

J. Mérour, S. Piroelle, Béatrice Malapel-Andrieu, 1998 .

Claisen Rearrangement of 2‐Allyloxyindolic Ketoester via a Decarboxylative Process.

J. Mérour, S. Piroelle, Béatrice Malapel-Andrieu, 1999 .

Heck Annulation on 2-Position of Indoles or 1H-Pyrrolo[2,3-b]pyridine

J. Mérour, E. Desarbre, 1995 .

Heck Annulation on 2-Position of Indoles or 1H-Pyrrolo(2,3-b)pyridine.

J. Mérour, E. Desarbre, 1995 .

Schmidt rearrangement of 1,2,3,5,10,10a-hexahydropyrrolo[1,2-b]-isoquinoline-3,10-diones

F. Cossais, J. Mérour, S. Piroelle, 1994 .