B. Maggio

发表

Novel 4-(3-phenylpropionamido), 4-(2-phenoxyacetamido) and 4-(cinnamamido) substituted benzamides bearing the pyrazole or indazole nucleus: synthesis, biological evaluation and mechanism of action.

A. D’Anneo, M. Lauricella, D. Raffa, 2019, Bioorganic chemistry.

N‐(Indazolyl)benzamido Derivatives as CDK1 Inhibitors: Design, Synthesis, Biological Activity, and Molecular Docking Studies

C. Colomba, M. Tolomeo, L. Titone, 2009, Archiv der Pharmazie.

Synthesis and antiproliferative activity of 3-(2-cloroethyl)-5- methyl-6-phenyl-8-(trifluoromethyl)-5,6-dihydropyrazolo[3,4- f][1,2,3,5]tetrazepin-4-(3H)-one

M. Tolomeo, M. V. Raimondi, S. Grimaudo, 2022 .

4-Diazopyrazole Derivatives as Potential New Antibiofilm Agents

M. V. Raimondi, D. Schillaci, D. Raffa, 2008, Chemotherapy.

(E)-2-{[1-(3,11-Dimethyl-4-methylene-10-oxo-1-phenyl-4,5,10,11-tetrahydro-1H-benzo[b]pyrazolo[3,4-f][1,5]diazocin-5-yl)ethylidene]amino}-N-methyl-N-(3-methyl-1-phenyl-1H-pyrazol-5-yl)benzamide

F. Meneghetti, B. Maggio, 2013, Acta crystallographica. Section E, Structure reports online.

Synthesis and Pharmacological Activities of Novel 3‐(Isoxazol‐3‐yl)‐quinazolin‐4(3H)‐one Derivatives

A. Caruso, V. Cutuli, N. Mangano, 1999, Archiv der Pharmazie.

Sortase A Inhibitors: Recent Advances and Future Perspectives.

M. V. Raimondi, D. Schillaci, D. Raffa, 2015, Journal of medicinal chemistry.

A new class of phenylhydrazinylidene derivatives as inhibitors of Staphylococcus aureus biofilm formation

A. Leonchiks, B. Manachini, M. V. Raimondi, 2016, Medicinal Chemistry Research.

Discovery of a New Class of Sortase A Transpeptidase Inhibitors to Tackle Gram-Positive Pathogens: 2-(2-Phenylhydrazinylidene)alkanoic Acids and Related Derivatives

D. Zhulenkovs, A. Leonchiks, L. Basile, 2016, Molecules.

4-(3H)-quinazolinones N-3 substituted with a five membered heterocycle: A promising scaffold towards bioactive molecules.

D. Raffa, F. Plescia, G. Daidone, 2020, European journal of medicinal chemistry.

Nonclassical Pschorr and Sandmeyer Reactions in Pyrazole Series

F. Meneghetti, G. Bombieri, D. Raffa, 2005 .

Consecutive Pschorr–Sandmeyer reactions in a pyrazole series. Part 2.1 Access to the [2]benzopyrano[4,3-c]pyrazole system of pharmaceutical interest

G. Bombieri, F. Benetollo, D. Raffa, 1998 .

Synthesis and anti-staphylococcal activity of new 4-diazopyrazole derivatives.

M. Vitale, M. V. Raimondi, D. Schillaci, 2012, European journal of medicinal chemistry.

Pyrazolobenzotriazinone Derivatives as COX Inhibitors: Synthesis, Biological Activity, and Molecular‐Modeling Studies

F. Plescia, C. Cannizzaro, G. Tringali, 2010, Archiv der Pharmazie.

Pyrazolo[3,4‐d]pyrimidine Derivatives as COX‐2 Selective Inhibitors: Synthesis and Molecular Modelling Studies

M. V. Raimondi, D. Raffa, F. Plescia, 2009, Archiv der Pharmazie.

Synthesis and pharmacological study of ethyl 1-methyl-5-(substituted 3,4-dihydro-4-oxoquinazolin-3-yl)-1H-pyrazole-4-acetates.

A. Caruso, A. Caruso, V. Cutuli, 2001, European journal of medicinal chemistry.

Synthesis and pharmacological study of ethyl 1-methyl-5-[2-substituted-4-oxo-3(4H)-quinazolinyl]-1H-pyrazole-4-acetates

A. Caruso, M. Amico-Roxas, D. Raffa, 1994 .

Antimicrobial and antineoplastic activities of new 4-diazopyrazole derivatives

G. Perra, M. Marongiu, C. Musiu, 1998 .

Synthesis, cytotoxicity, and inhibitory effects on tubulin polymerization of a new 3-heterocyclo substituted 2-styrylquinazolinones.

E. Hamel, D. Schillaci, R. Bai, 2004, European journal of medicinal chemistry.

Synthesis and antileukemic activity of new 3-(5-methylisoxazol-3-yl) and 3-(pyrimidin-2-yl)-2-styrylquinazolin-4(3H)-ones.

D. Schillaci, D. Raffa, F. Plescia, 2004, Farmaco.

Synthesis and antileukemic activity of new 3-(1-phenyl-3-methylpyrazol-5-yl)-2-styrylquinazolin-4(3H)-ones.

D. Schillaci, D. Raffa, F. Plescia, 2004, Farmaco.

Synthesis, Cytotoxicity, and Inhibitory Effects on Tubulin Polymerization of a New 3‐Heterocyclo Substituted 2‐Styrylquinazolinones.

E. Hamel, D. Schillaci, R. Bai, 2004 .

Synthesis and in vitro antileukemic activity of new 4-triazenopyrazole derivatives.

D. Schillaci, D. Raffa, G. Daidone, 2004, Farmaco.

Synthesis and antifungal activity of new N-isoxazolyl-2-iodobenzamides.

D. Schillaci, L. Torta, D. Raffa, 1999, Farmaco.

Synthesis and Antiproliferative Activity of Novel 3‐(Indazol‐3‐yl)‐quinazolin‐4(3H)‐one and 3‐(Indazol‐3‐yl)‐benzotriazin‐4(3H)‐one Derivatives

D. Schillaci, D. Raffa, F. Plescia, 1999, Archiv der Pharmazie.

Recent advanced in bioactive systems containing pyrazole fused with a five membered heterocycle.

M. V. Raimondi, D. Raffa, F. Plescia, 2015, European journal of medicinal chemistry.

Synthesis, antiproliferative activity, and mechanism of action of a series of 2-{[(2E)-3-phenylprop-2-enoyl]amino}benzamides.

E. Hamel, M. Tolomeo, M. V. Raimondi, 2011, European journal of medicinal chemistry.

Synthesis of substituted 3-amino-N-phenyl-1H-indazole-1-carboxamides endowed with antiproliferative activity.

M. Tolomeo, M. V. Raimondi, R. Pipitone, 2011, European journal of medicinal chemistry.

Synthesis and pharmacological evaluation of 1-methyl-5-[substituted-4 (3H)-oxo-1,2,3-benzotriazin-3-yl]-1H-pyrazole-4-acetic acid derivatives.

D. Schillaci, A. Caruso, V. Cutuli, 1998, Farmaco.

Synthesis, crystallographic studies and biological evaluation of some 2-substituted 3-indazolyl-4(3H)-quinazolinones and 3-indazolyl-4(3H)-benzotriazinones

G. Bombieri, D. Schillaci, F. Benetollo, 1996 .

3 alpha-hydroxysteroid dehydrogenase inhibitory activity of some N(3)-(1-R-4-carboxypyrazol-5-yl)-1,2,3-benzotriazin-4(3H)-one and quinazolin-4(3H)-one acids.

D. Schillaci, D. Raffa, G. Daidone, 1994, Farmaco.

Synthesis and antileukemic activity of new 3-(5-methylisoxazol-3-yl) and 3-(pyrimidin-2-yl)-2-styrylquinazolin-4(3H)-ones.

D. Schillaci, D. Raffa, F. Plescia, 2004, Farmaco.

Phenylamides of 1‐Phenyl (or Methyl)‐5‐benzamidopyrazole‐4‐carboxylic Acid as Vratizolin Analogs with Analgesic and Antiinflammatory Activities

A. Caruso, N. Mangano, D. Raffa, 2001, Archiv der Pharmazie.

Synthesis and antiproliferative activity of 3-amino-N-phenyl-1H-indazole-1-carboxamides.

F. Meneghetti, G. Gallo, M. Tolomeo, 2009, European journal of medicinal chemistry.

Synthesis and biological evaluation of new indazole derivatives

F. Meneghetti, G. Bombieri, M. V. Raimondi, 2010 .

Synthesis, benzodiazepine receptor binding and molecular modelling of isochromeno[4,3-c]pyrazol-5(1H)-one derivatives.

M. Trincavelli, C. Martini, F. Meneghetti, 2012, European journal of medicinal chemistry.

Oxidative halogenation of substituted pyrroles with Cu(II). Part IV. Bromination of 2‐(2′‐hydroxybenzoyl)pyrrole. A new synthesis of bioactive analogs of monodeoxypyoluteorin

D. Schillaci, B. Maggio, M. Ciofalo, 1994 .

Synthesis, antiproliferative activity and possible mechanism of action of novel 2-acetamidobenzamides bearing the 2-phenoxy functionality.

A. D’Anneo, M. Lauricella, E. Hamel, 2015, Bioorganic & medicinal chemistry.

Pharmaceutical Potential of Synthetic and Natural Pyrrolomycins

M. V. Raimondi, D. Schillaci, D. Raffa, 2015, Molecules.

RADICAL CYCLIZATION AND 1,5-HYDROGEN TRANSFER IN SELECTED AROMATIC DIAZONIUM SALTS

F. Ferrante, D. Raffa, G. Daidone, 2014 .

Recent discoveries of anticancer flavonoids.

M. V. Raimondi, D. Raffa, F. Plescia, 2017, European journal of medicinal chemistry.

Synthesis and antifungal activity of new N-(1-phenyl-4-carbetoxypyrazol-5-yl)-, N-(indazol-3-yl)- and N-(indazol-5-yl)-2-iodobenzamides.

D. Schillaci, L. Torta, D. Raffa, 2002, Il Farmaco.

Synthesis and antiproliferative activity of 3-(2-chloroethyl)-5-methyl-6-phenyl-8-(trifluoromethyl)-5,6-dihydropyrazolo[3,4-f][1,2,3,5]tetrazepin-4-(3H)-one.

M. Tolomeo, M. V. Raimondi, S. Grimaudo, 2015, European journal of medicinal chemistry.

Synthesis and induction of G0-G1 phase arrest with apoptosis of 3,5-dimethyl-6-phenyl-8-(trifluoromethyl)-5,6-dihydropyrazolo[3,4-f][1,2,3,5]tetrazepin-4(3H)-one.

M. Tolomeo, E. Barbusca, G. Cannizzo, 2008, European journal of medicinal chemistry.

Synthesis and in vitro antileukemic activity of new 4-triazenopyrazole derivatives.

D. Schillaci, D. Raffa, G. Daidone, 2004, Farmaco.

Synthesis and antiproliferative activity of triazenoindazoles and triazenopyrazoles: a comparative study.

D. Schillaci, D. Raffa, F. Plescia, 2004, European journal of medicinal chemistry.

Salicylanilide and its heterocyclic analogues. A comparative study of their antimicrobial activity.

D. Schillaci, G. Daidone, B. Maggio, 1990, Die Pharmazie.

Pyrazolo[3,4‐d]pyrimidine Derivatives as COX‐2 Selective Inhibitors: Synthesis and Molecular Modelling Studies

M. V. Raimondi, D. Raffa, F. Plescia, 2009, Archiv der Pharmazie.

Recent Advanced in Bioactive Systems Containing Pyrazole Fused with a Five Membered Heterocycle

M. V. Raimondi, D. Raffa, F. Plescia, 2015 .

Anthranilamide-based 2-phenylcyclopropane-1-carboxamides, 1,1'-biphenyl-4-carboxamides and 1,1'-biphenyl-2-carboxamides: Synthesis biological evaluation and mechanism of action.

A. D’Anneo, M. Lauricella, M. V. Raimondi, 2017, European journal of medicinal chemistry.

Comparative structural studies of 4-diazopyrazole derivatives by X-ray diffraction and theoretical investigation

R. Artali, G. Bombieri, M. V. Raimondi, 2005 .

The role of (E)-6-chloro-3-(3-methyl-1-phenyl-1H-pyrazol-5-yl)-2-styrylquinazolin-4(3H)-one in the modulation of cannabinoidergic system. A pilot study

F. Plescia, M. V. Raimondi, C. Cannizzaro, 2018, Pharmacological reports : PR.

Synthesis and biofilm formation reduction of pyrazole-4-carboxamide derivatives in some Staphylococcus aureus strains.

B. Manachini, M. V. Raimondi, D. Schillaci, 2016, European journal of medicinal chemistry.

A new class of phenylhydrazinylidene derivatives as inhibitors of Staphylococcus aureus biofilm formation

A. Leonchiks, B. Manachini, M. V. Raimondi, 2016, Medicinal Chemistry Research.

Synthesis and bio fi lm formation reduction of pyrazole-4-carboxamide derivatives in some Staphylococcus aureus strains

B. Manachini, M. V. Raimondi, D. Schillaci, 2016 .

Synthesis and antiproliferative activity of new derivatives containing the polycyclic system 5,7:7,13-dimethanopyrazolo[3,4-b]pyrazolo[3',4':2,3]azepino[4,5-f]azocine.

D. Carlisi, M. Lauricella, M. V. Raimondi, 2014, European journal of medicinal chemistry.

Synthesis of new 3-(3-phenyl-isoxazol-5-yl) or 3-[(3-phenyl-isoxazol-5-yl)-amino] substituted 4(3H)-quinazolinone derivatives with antineoplastic activity.

D. Schillaci, D. Raffa, F. Plescia, 1999, Die Pharmazie.

Sortase A Inhibitors: Recent Advances and Future Perspectives.

M. V. Raimondi, D. Schillaci, D. Raffa, 2015, Journal of medicinal chemistry.

Pyrazolobenzotriazinone Derivatives as COX Inhibitors: Synthesis, Biological Activity, and Molecular‐Modeling Studies

F. Plescia, C. Cannizzaro, G. Tringali, 2010, Archiv der Pharmazie.

Synthesis and induction of G0-G1 phase arrest with apoptosis of 3,5-dimethyl-6-phenyl-8-(trifluoromethyl)-5,6-dihydropyrazolo[3,4-f][1,2,3,5]tetrazepin-4(3H)-one.

M. Tolomeo, E. Barbusca, G. Cannizzo, 2008, European journal of medicinal chemistry.

Synthesis and antiproliferative activity of a natural like glycoconjugate polycyclic compound.

A. D’Anneo, M. Lauricella, M. V. Raimondi, 2016, European journal of medicinal chemistry.