Emanuela Berrino

发表

Amine- and Amino Acid-Based Compounds as Carbonic Anhydrase Activators

S. Carradori, C. Supuran, A. Angeli, 2021, Molecules.

New thiopyrimidine-benzenesulfonamide conjugates as selective carbonic anhydrase II inhibitors: synthesis, in vitro biological evaluation, and molecular docking studies.

C. Supuran, Ahmed S. Abdelsamie, Ahmed M. El Kerdawy, 2020, Bioorganic & medicinal chemistry.

Synthesis and Evaluation of Carbonic Anhydrase Inhibitors with Carbon Monoxide Releasing Properties for the Management of Rheumatoid Arthritis.

C. Supuran, D. Vullo, C. Ghelardini, 2019, Journal of medicinal chemistry.

Synthesis and carbonic anhydrase inhibitory properties of novel 4-(2-aminoethyl)benzenesulfonamide-dipeptide conjugates.

C. Supuran, C. Capasso, G. Bartolucci, 2019, Bioorganic chemistry.

Novel Insights on CAI-CORM Hybrids: Evaluation of the CO Releasing Properties and Pain-Relieving Activity of Differently Substituted Coumarins for the Treatment of Rheumatoid Arthritis.

S. Carradori, C. Supuran, C. Ghelardini, 2023, Journal of medicinal chemistry.

Advances in microwave-assisted synthesis and the impact of novel drug discovery

Claudiu T Supuran, Emanuela Berrino, C. Supuran, 2018, Expert opinion on drug discovery.

New 1H‐indole‐2,3‐dione 3‐thiosemicarbazones with 3‐sulfamoylphenyl moiety as selective carbonic anhydrase inhibitors

C. Supuran, N. Karalı, A. Akdemir, 2022, Archiv der Pharmazie.

Bioorganometallic derivatives of 4-hydrazino-benzenesulphonamide as carbonic anhydrase inhibitors: synthesis, characterisation and biological evaluation

C. Supuran, R. Arancibia, Emanuela Berrino, 2020, Journal of enzyme inhibition and medicinal chemistry.

A class of carbonic anhydrase IX/XII – selective carboxylate inhibitors

C. Supuran, A. El‐Faham, Z. Almarhoon, 2020, Journal of enzyme inhibition and medicinal chemistry.

New sulfonamides containing organometallic-acylhydrazones: synthesis, characterisation and biological evaluation as inhibitors of human carbonic anhydrases

C. Supuran, Néstor Novoa, R. Arancibia, 2019, Journal of enzyme inhibition and medicinal chemistry.

Azidothymidine “Clicked” into 1,2,3-Triazoles: First Report on Carbonic Anhydrase–Telomerase Dual-Hybrid Inhibitors

S. Carradori, C. Supuran, T. Peat, 2020, Journal of medicinal chemistry.

Carbonic anhydrase inhibitors for the treatment of epilepsy and obesity

F. Carta, Emanuela Berrino, 2019, Carbonic Anhydrases.

In Silico Identification and Biological Evaluation of Antioxidant Food Components Endowed with Human Carbonic Anhydrase IX and XII Inhibition

C. Supuran, A. Salatino, F. Trapasso, 2020, Antioxidants.

In Silico Identification and Biological Evaluation of Antioxidant Food Components Endowed with IX and XII hCA Inhibition

C. Supuran, A. Salatino, F. Trapasso, 2020 .

Novel Insights on Human Carbonic Anhydrase Inhibitors Based on Coumalic Acid: Design, Synthesis, Molecular Modeling Investigation, and Biological Studies

S. Carradori, C. Supuran, A. Ciogli, 2022, International journal of molecular sciences.

Modulating the Efficacy of Carbonic Anhydrase Inhibitors through Fluorine Substitution.

C. Supuran, F. Carta, A. Martin-Mingot, 2021, Angewandte Chemie.

Toxicity evaluation of sulfamides and coumarins that efficiently inhibit human carbonic anhydrases

C. Supuran, C. Capasso, S. Parkkila, 2020, Journal of enzyme inhibition and medicinal chemistry.

Novel approaches for designing drugs that interfere with pH regulation

C. Supuran, Emanuela Berrino, 2019, Expert opinion on drug discovery.

Carbonic Anhydrase Inhibitors of Different Structures Dilate Pre-Contracted Porcine Retinal Arteries

C. Supuran, F. Carta, S. Selleri, 2019, International Journal of Molecular Sciences.

Novel Sulfamide-Containing Compounds as Selective Carbonic Anhydrase I Inhibitors

C. Supuran, M. Botta, A. Mugelli, 2017, Molecules.

A Novel Class of Dual-Acting DCH-CORMs Counteracts Oxidative Stress-Induced Inflammation in Human Primary Tenocytes

S. Carradori, Cristina Campestre, M. Gallorini, 2021, Antioxidants.

SLC-0111 enaminone analogs, 3/4-(3-aryl-3-oxopropenyl) aminobenzenesulfonamides, as novel selective subnanomolar inhibitors of the tumor-associated carbonic anhydrase isoform IX.

C. Supuran, D. Vullo, Ghada S. Hassan, 2019, Bioorganic chemistry.

Inhibition of α-, β-, γ-, and δ-carbonic anhydrases from bacteria and diatoms with N′-aryl-N-hydroxy-ureas

C. Supuran, C. Capasso, Z. Alothman, 2018, Journal of enzyme inhibition and medicinal chemistry.

In Silico-Guided Identification of New Potent Inhibitors of Carbonic Anhydrases Expressed in Vibrio cholerae.

C. Supuran, C. Capasso, A. Angeli, 2020, ACS medicinal chemistry letters.

Synthesis of novel benzenesulfamide derivatives with inhibitory activity against human cytosolic carbonic anhydrase I and II and Vibrio cholerae α- and β-class enzymes

C. Supuran, A. Mugelli, C. Capasso, 2018, Journal of enzyme inhibition and medicinal chemistry.

Modulating the Efficacy of Carbonic Anhydrase Inhibitors through Fluorine Substitution

C. Supuran, F. Carta, A. Martin-Mingot, 2021, Angewandte Chemie.

Dual Carbonic Anhydrase IX/XII Inhibitors and Carbon Monoxide Releasing Molecules Modulate LPS-Mediated Inflammation in Mouse Macrophages

S. Carradori, C. Supuran, H. Schweikl, 2021, Antioxidants.

Mechanisms of the Antiproliferative and Antitumor Activity of Novel Telomerase-Carbonic Anhydrase Dual-Hybrid Inhibitors.

C. Supuran, M. Ferraroni, A. Veselovsky, 2021, Journal of medicinal chemistry.

1,2,4-Trisubstituted imidazolinones with dual carbonic anhydrase and p38 mitogen-activated protein kinase inhibitory activity.

C. Supuran, Hanan H. Georgey, Emanuela Berrino, 2019, Bioorganic chemistry.

N-aryl-N'-ureido-O-sulfamates as potent and selective inhibitors of hCA VB over hCA VA: Deciphering the binding mode of new potential agents in mitochondrial dysfunctions.

C. Supuran, T. Tuccinardi, A. Angeli, 2020, Bioorganic chemistry.

Zeta-carbonic anhydrases show CS2 hydrolase activity: A new metabolic carbon acquisition pathway in diatoms?

E. Langella, C. Supuran, M. Polentarutti, 2021, Computational and structural biotechnology journal.

Rho-kinase inhibitors in the management of glaucoma

C. Supuran, Emanuela Berrino, 2019, Expert opinion on therapeutic patents.

Uncovering Novel Capsaicin Inhibitory Activity towards Human Carbonic Anhydrase Isoforms IX and XII by Combining In Silico and In Vitro Studies

C. Supuran, A. Salatino, F. Trapasso, 2023, Antioxidants.

An innovative spectroscopic approach for qualitative and quantitative evaluation of Mb-CO from myoglobin carbonylation reaction through chemometrics methods

S. Carradori, C. Supuran, Alane Beatriz Vermelho, 2021, Spectrochimica Acta Part A: Molecular and Biomolecular Spectroscopy.

Escinosome thermosensitive gel optimizes efficacy of CAI-CORM in a rat model of rheumatoid arthritis.

C. Supuran, C. Ghelardini, L. Mannelli, 2023, Journal of controlled release : official journal of the Controlled Release Society.

Design and synthesis of 6-arylpyridine-tethered sulfonamides as novel selective inhibitors of carbonic anhydrase IX with promising antitumor features toward the human colorectal cancer.

Tamer M. Ibrahim, C. Supuran, F. Şahin, 2023, European journal of medicinal chemistry.