J. Magano

发表

Chromatography- and Lyophilization-Free Synthesis of a Peptide-Linker Conjugate

J. Teixeira, Jian Wang, J. Rizzo, 2014 .

Synthesis of a novel analytical reagent for the determination of active sites for conjugation on a catalytic aldolase monoclonal antibody

J. Teixeira, C. Bradshaw, A. Bhat, 2012 .

Palbociclib Commercial Manufacturing Process Development. Part II: Regioselective Heck Coupling with Polymorph Control for Processability

Brian P. Jones, K. Leeman, N. Ide, 2016 .

Synthetic approaches to the neuraminidase inhibitors zanamivir (Relenza) and oseltamivir phosphate (Tamiflu) for the treatment of influenza.

J. Magano, 2009, Chemical reviews.

Kilogram-Lab-Scale Oxindole Synthesis via Palladium-Catalyzed C–H Functionalization

J. Magano, E. Kiser, Russell James Shine, 2012 .

Development of an Air-Stable, Broadly Applicable Nickel Source for Nickel-Catalyzed Cross-Coupling

Sebastien Monfette, J. Magano, 2015 .

Large-Scale Amidations in Process Chemistry: Practical Considerations for Reagent Selection and Reaction Execution

J. Magano, 2022, Organic Process Research & Development.

Transition metal-catalyzed couplings in process chemistry : case studies from the pharmaceutical industry

J. R. Dunetz, J. Magano, 2013 .

The Evolution of High-Throughput Experimentation in Pharmaceutical Development and Perspectives on the Future

Ling Li, Emma McInturff, Ke Wang, 2019, Organic Process Research & Development.

Overcoming the Challenges of Making a Single Enantiomer N-1 Substituted Tetrazole Prodrug Using a Tin-Mediated Alkylation and Enzymatic Resolution

Shu Yu, R. Kumar, D. W. Piotrowski, 2019, Organic Process Research & Development.

2-(Diethylamino)ethanethiol, a new reagent for the odorless deprotection of aromatic methyl ethers.

T. Nussbaumer, Jerry D. Clark, J. Magano, 2006, The Journal of organic chemistry.

Large-Scale Applications of Amide Coupling Reagents for the Synthesis of Pharmaceuticals

Gerald A. Weisenburger, Javier Magano, Joshua R. Dunetz, 2016 .

Recent synthetic approaches to oseltamivir phosphate (Tamiflu™) for the treatment of influenza

J. Magano, 2011 .

Large-scale applications of transition metal-catalyzed couplings for the synthesis of pharmaceuticals.

Javier Magano, Joshua R Dunetz, J. R. Dunetz, 2011, Chemical reviews.

A CONVENIENT REDUCTION OF HIGHLY FUNCTIONALIZED AROMATIC CARBOXYLIC ACIDS TO ALCOHOLS WITH BORANE-THF AND BORON TRIFLUORIDE-ETHERATE

J. Magano, E. Iakovleva, K. Sexton, 2002 .

Large-Scale Carbonyl Reductions in the Pharmaceutical Industry

J. R. Dunetz, J. Magano, 2012 .

Development of a Scalable Synthesis for an Inhaled pan-JAK Inhibitor

J. Coe, Seungwon Chung, L. Samp, 2019, Organic Process Research & Development.

Diastereoselective, large scale synthesis of β-amino acids via asymmetric enamide hydrogenation as α2δ ligands for the treatment of generalized anxiety disorder and insomnia

J. Magano, D. Bowles, B. G. Conway, 2009 .

The Synthesis of (S)-5-Fluoro-1-(2-fluorophenyl)-3-(piperidin-3-ylmethoxy)-1H-indazole, a Norepinephrine/Serotonin Reuptake Inhibitor for the Treatment of Fibromyalgia

Derek Greene, E. Nord, Michael Waldo, 2008 .

Practical Synthesis of 1-(7-Fluoro-naphthalen-1-yl)piperazine Hydrochloride

J. Magano, A. Akin, Michael H. Chen, 2008 .

Large‐Scale Applications of Transition Metal Removal Techniques in the Manufacture of Pharmaceuticals

J. Magano, 2013 .

2‐(Diethylamino)ethanethiol, a New Reagent for the Odorless Deprotection of Aromatic Methyl Ethers.

T. Nussbaumer, Jerry D. Clark, J. Magano, 2007 .

Streamlined Synthesis of a Bicyclic Amine Moiety Using an Enzymatic Amidation and Identification of a Novel Solid Form

S. G. Ruggeri, S. Kulkarni, Amber M. Johnson, 2021 .

Recent Synthetic Approaches to Oseltamivir Phosphate (Tamiflu) for the Treatment of Influenza

J. Magano, 2012 .

Expeditious, large scale preparation of ethyl (R)-5-methyl-3-oxo octanoate via a cross Claisen reaction between N-acyl oxazolidinone derivatives and the magnesium enolate of potassium ethyl malonate

J. Magano, T. N. Nanninga, D. D. Winkle, 2008 .

An efficient stereoselective synthesis of [3S(1S,9S)]-3-[[[9-(benzoylamino) octahydro-6,10-dioxo-6H-pyridazino-(1,2-a)(1,2)-diazepin-1-yl]-carbonyl ]amino]-4-oxobutanoic acid, an interleukin converting enzyme (ICE) inhibitor.

J. Rubin, M. H. Chen, J. Magano, 1999, Bioorganic & medicinal chemistry letters.

Route Optimization of the Non-covalent Modulator of Hemoglobin PF-07059013 for the Treatment of Sickle Cell Disease, Part I: From Discovery Synthesis to First Kilogram-Scale Manufacture

C. Limberakis, Aaron F. Baldwin, Sebastien Monfette, 2023, Organic Process Research & Development.

AN EFFICIENT AND SCALABLE SYNTHESIS OF METHYL 3-HYDROXYMETHYLBENZOATE

J. G. Davidson, M. H. Chen, J. Magano, 2000 .

An Efficient and Scalable Synthesis of Methyl 3-Hydroxymethylbenzoate (III).

J. G. Davidson, M. H. Chen, J. Magano, 2000 .

Recent Large-Scale Applications of Transition Metal-Catalyzed Couplings for the Synthesis of Pharmaceuticals

J. R. Dunetz, J. Magano, 2011 .

Kinetic and Data-Driven Reaction Analysis for Pharmaceutical Process Development

Bryan M. Li, Jason Mustakis, J. Magano, 2020, Industrial & Engineering Chemistry Research.