J. Ezquerra

发表

Conformationally constrained serotonin analogues: Stereoselective synthesis of trans-3-(2-aminocycloalkyl)indoles by aziridine ring opening

C. Lamas, C. Pedregal, J. J. Vaquero, 1996 .

Stereoselective reactions of lithium enolates derived from N-BOC protected pyroglutamic esters

C. Pedregal, F. Sánchez-Ferrando, J. Ezquerra, 1993 .

Stereoselective double alkylation of ethyl N-boc-pyroglutamate

J. Vaquero, C. Pedregal, J. Deeter, 1994 .

A new approach to the synthesis of 2-aminoimidazo[1,2-a]pyridine derivatives through microwave-assisted N-alkylation of 2-halopyridines

C. Hamdouchi, J. Alvarez-Builla, J. A. Vega, 1999 .

4-Substituted D-glutamic acid analogues: the first potent inhibitors of glutamate racemase (MurI) enzyme with antibacterial activity.

Jose-Alfredo Martin, J. Mcgee, Ana Sánchez, 2002, Journal of medicinal chemistry.

General method for the synthesis of 5-arylpyrrole-2-carboxylic acids

C. Pedregal, J. Alvarez-Builla, J. J. Vaquero, 1993 .

Synthesis of α-substituted and α,α-disubstituted α-amino acids by controlled mono- and dialkylation of ethyl N-diphenylmethyleneglycinate

C. Pedregal, R. Pleixats, M. Moreno-Mañas, 1993 .

Organic sonochemistry. Synthesis and use of Reissert compounds under PTC-ultrasound

J. Alvarez-Builla, J. Ezquerra, 1988 .

Phase transfer catalysis under ultrasound. Alkylation of isoquinoline Reissert compound

J. Alvarez-Builla, J. Ezquerra, 1984 .

A microwave synthesis of the cis and trans isomers of 3-hydroxy-2-(4-methoxyphenyl)-2,3-dihydro-1,5-benzothiazepin-4(5H)-one: The influence of solvent and power output on the diastereoselectivity

J. Alvarez-Builla, J. A. Vega, J. J. Vaquero, 1996 .

Short synthesis and anti-rhinoviral activity of imidazo[1,2-a]pyridines: the effect of acyl groups at 3-position.

C. Hamdouchi, B. Heinz, J. Alvarez-Builla, 1999, Bioorganic & medicinal chemistry letters.

Efficient Reagents for the Synthesis of 5-, 7-, and 5,7-Substituted Indoles Starting from Aromatic Amines: Scope and Limitations

C. Lamas, C. Pedregal, M. Garcia-Martin, 1996 .

Highly chemoselective reduction of N-Boc protected lactams

C. Pedregal, M. C. Carreño, J. G. Ruano, 1994 .

Stereoselective Michael Addition of Glycine Anions to Chiral Fischer Alkenylcarbene Complexes. Asymmetric Synthesis of beta-Substituted Glutamic Acids.

S. García‐Granda, C. Pedregal, J. Flórez, 1999, The Journal of organic chemistry.

Improved Preparation of Diethyl Bromomethylphosphonate and Diiodomethane-Catalyzed Triethylphosphite Michaelis-Arbuzov Isomerization

A. Roglans, J. Ezquerra, B. Yruretagoyena, 1995 .

New enantioselective approach to α-allokainoids by Michael addition to chiral 4-substituted 2,3-didehydroprolinate

A. Escribano, J. Ezquerra, A. Rubio, 1995 .

4-benzyl-2,3-didehydroprolinate as a homochiral template for michael additions. Synthesis of enantiopure α-allokainoids, β-kainoids, 2,3-methanoprolines and other 3,4-disubstituted prolines

J. J. Vaquero, J. Ezquerra, A. Rubio, 1996 .

Suzuki-type cross-coupling reaction of 1-benzyl-2-iodo-1H-benzimidazoles with aryl boronic acids: A regioselective route to N-alkylated 6-alkoxy-2-aryl-1H-benzimidazoles

C. Lamas, J. J. Vaquero, J. Ezquerra, 1997 .

Stereoselective synthesis of 1,3,4-substituted tetrahydro-β-carbolines from indoles based on selective transformations

C. Lamas, C. Pedregal, J. J. Vaquero, 1997 .

Stereocontrolled Synthesis of 5α- and 5β-Substituted Kainic Acids

C. Pedregal, A. Mateo, J. Ezquerra, 1999 .

STEREOSELECTIVE ADDITION OF GRIGNARD-DERIVED ORGANOCOPPER REAGENTS TO N-ACYLIMINIUM IONS : SYNTHESIS OF ENANTIOPURE 5- AND 4,5-SUBSTITUTED PROLINATES

C. Pedregal, J. Ezquerra, I. Collado, 1995 .

Ethyl N-(diphenylmethylene)glycinate as anionic glycine equivalent. Monoalkylation, dialkylation and Michael additions under solid-liquid phase-transfer catalysis

C. Pedregal, R. Pleixats, M. Moreno-Mañas, 1996 .

Diastereoselective functionalization of 5-hydroxy prolinates by tandem Horner-Emmons-Michael reaction

C. Pedregal, J. J. Vaquero, J. Ezquerra, 1994 .

Stereoselective functionalisation of N-Boc pyroaminoadipic acid: Synthesis of 5-substituted aminoadipic and pipecolic acids

C. Pedregal, M. C. Carreño, J. G. Ruano, 1995 .

Mild and Efficient Palladium-Mediated C-N Cross-Coupling Reaction between DNA-Conjugated Aryl Bromides and Aromatic Amines.

A. Torrado, J. Ezquerra, Eduardo de Pedro Beato, 2019, ACS combinatorial science.

Stereoselective Michael Addition of Glycine Anions to Chiral Fischer Alkenylcarbene Complexes. Asymmetric Synthesis of β‐Substituted Glutamic Acids.

S. García‐Granda, C. Pedregal, J. Flórez, 2000 .

Regioselective nucleophilic attack on N-BOC-pyroglutamate ethyl ester

C. Pedregal, J. D. Mendoza, J. Ezquerra, 1992 .

Stereoselective formal [3 + 2] cycloaddition of N-alkylidene glycine ester anions to chiral Fischer alkenylcarbene complexes. Asymmetric synthesis of 3,4,5-trisubstituted prolines.

C. Pedregal, J. Flórez, J. Barluenga, 2002, The Journal of organic chemistry.

Enantiospecific synthesis of (1S,2S,5R,6S)-2-aminobicyclo[3.1.0]hexane-2,6-dicarboxylic acid by a modified Corey-Link reaction

C. Domínguez, J. Ezquerra, S. Baker, 1998 .

Synthesis of Enantiomerically Pure 4-Substituted Glutamic Acids and Prolines: General Aldol Reaction of Pyroglutamate Lactam Lithium Enolate Mediated by Et2O.cntdot.BF3

C. Pedregal, M. C. Carreño, A. Escribano, 1995 .

A novel application of the Ullmann coupling reaction for the alkylsulfenylation of 2-amino-imidazo[1,2-a]pyridine

C. Hamdouchi, J. Ezquerra, J. Blas, 1999 .

Synthesis of γ,δ-unsaturated 6-hydroxy substituted α-amino acids by palladium-catalyzed alkylation of monoepoxydienes

C. Pedregal, C. Nájera, A. Mazon, 1997 .

Solid phase synthesis of glutamic acid derivatives via nucleophilic ring opening of N-Boc pyroglutamate with heteronucleophiles

E. Dominguez, J. Ezquerra, J. Blas, 2000 .

New enantioselective approach to the total synthesis of (−)-α-Kainic Acid

J. J. Vaquero, J. Ezquerra, A. Rubio, 1998 .

Enantiospecific synthesis of the the tricyclxc nucleus of acetoxycrenulide by claisen ring exfansion

L. Paquette, Wei He, J. Ezquerra, 1990 .

Suitability of the Claisen ring expansion protocol for crenulide diterpene construction

L. Paquette, Wei He, J. Ezquerra, 1995 .

Stereoselective Cyclopropanation of Enones with Ethyl Dimethylsulfonium Acetate Bromide in the Presence of DBU.

C. Pedregal, C. Domínguez, J. Monn, 1997 .

Regioselective ring opening of chiral N-boc protected pyroglutamate and pyroaminoadipate ethyl esters with heteronucleophiles

C. Pedregal, A. Escribano, M. Molina, 1993 .

Chemoselective nucleophilic attack on N-acyl derivatives of (S)-ethyl 4,4-dimethyl pyroglutamate (DMPG).

J. Alvarez-Builla, J. J. Vaquero, J. Espinosa, 2003, Organic letters.

Conformationally constrained ACPD analogues. Synthesis and resolution of 3-aminobicyclo[3,3,0]octane-1,3-dicarboxylic acids

C. Avendaño, J. Ezquerra, W. Prowse, 1995 .

Synthesis of 3- and 4-substituted cyclic α-amino acids structurally related to ACPD

Ismael Gracia, M. Yus, J. Sansano, 1995 .

STEREOSELECTIVE SYNTHESIS OF 2,3-DISUBSTITUTED GLUTAMIC ACID DERIVATIVES BY CONJUGATE ADDITION TO 3,4-DIDEHYDROPYROGLUTAMATES

C. Pedregal, G. Guillena, C. Nájera, 1998 .

2-Methylpyridinium salts as 1,4-dinucleophiles. Quinolizinium salts from the westphal condensation

J. Alvarez-Builla, J. Ezquerra, G. G. Trigo, 1985 .

2,3'-disubstituted-2-(2'-carboxycyclopropyl)glycines as potent and selective antagonists of metabotropic glutamate receptors.

D. Schoepp, C. Pedregal, A. Mazon, 1998, Bioorganic & medicinal chemistry letters.

New uses of the westphal condensation. Synthesis of pi-donor-pi-acceptor heterocycles.

J. Vaquero, J. Alvarez-Builla, F. Sánchez-Ferrando, 1991 .

Stereoselective cyclopropanation of enones with ethyl dimethylsulfonium acetate bromide in the presence of DBU

C. Pedregal, C. Domínguez, J. Monn, 1997 .

Quinolizinium salts as fluorescent probes for N-nucleophiles

M. A. Martín, J. Alvarez-Builla, B. Castillo, 1985 .

Short and efficient enantioselective synthesis of cis and trans pyrrolidine-2,5 dicarboxylic acids

C. Pedregal, J. G. Ruano, J. Ezquerra, 1993 .

First Trapping Reaction of N-Boc Ethyl 3,4-Dehydropyroglutamate with Cyclopentadiene

C. Pedregal, J. Ezquerra, A. Rubio, 1995 .

4-Alkyl- and 4-cinnamylglutamic acid analogues are potent GluR5 kainate receptor agonists.

B. Ballyk, C. Dominguez, D. Bleakman, 2000, Journal of medicinal chemistry.

(2S,4S)-amino-4-(2,2-diphenylethyl)pentanedioic acid selective group 2 metabotropic glutamate receptor antagonist.

D. Schoepp, C. Pedregal, B. Johnson, 1998, Bioorganic & medicinal chemistry letters.

2‐Methylpyridinium salts as 1,4‐dinucleophiles. II. Westphal condensation with substituted pyridinium substrates

J. Alvarez-Builla, J. Ezquerra, 1986 .

4-Alkylidenyl glutamic acids, potent and selective GluR5 agonists.

B. Ballyk, C. Dominguez, D. Bleakman, 2000, Bioorganic & medicinal chemistry letters.

Synthesis of bis(α-amino acids) by palladium-catalyzed allylic double substitution

C. Pedregal, C. Nájera, A. Mazon, 1995 .

Chemoselective Arylsulfenylation of 2-Aminoimidazol[1,2-a]pyridines by Phenyliodine(III) Bis(trifluoroacetate) (PIFA)

C. Hamdouchi, J. Ezquerra, C. Sanchez, 1998 .

Chemoselective Arylsulfenylation of 2-Aminoimidazol[1,2-a]pyridines by Phenyliodine(III) Bis(trifluoroacetate) (PIFA)

C. Hamdouchi, J. Ezquerra, C. Sanchez, 1998 .

New uses of westphal condensation : synthesis of flavocorylene and related indolo[2,3-a]quinolizinium salts

J. Vaquero, J. Alvarez-Builla, J. Ezquerra, 1991 .

Asymmetric synthesis of (+)-2-aminobicyclo[3.1.0]hexane-2,6-dicarboxylic acid (LY354740)

C. Domínguez, J. Ezquerra, M. Espada, 1997 .

Asymmetric Michael addition reactions using ethyl (S)-4,4-dimethylpyroglutamate as a chiral auxiliary

C. Avendaño, J. Ezquerra, Lourdes Prieto, 1999 .

Ethyl 4,4-dimethyl pyroglutamate (DMPG): a chiral auxiliary in cyclopropanation and carbonyl group activator

J. Ezquerra, Pablo García Losada, S. Mantecón, 2010 .