K. Solomon

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Identification and Characterization of INCB 9471 , an Allosteric Noncompetitive Small-Molecule Antagonist of C-C Chemokine Receptor 5 with Potent Inhibitory Activity against Monocyte Migration and HIV-1 Infection

P. Scherle, N. Zhou, F. Baribaud, 2011 .

Identification and Characterization of INCB9471, an Allosteric Noncompetitive Small-Molecule Antagonist of C-C Chemokine Receptor 5 with Potent Inhibitory Activity against Monocyte Migration and HIV-1 Infection

P. Scherle, N. Zhou, F. Baribaud, 2011, Journal of Pharmacology and Experimental Therapeutics.

(Z)-2-(4-Nitrobenzylidene)-1-benzofuran-3(2H)-one

G. Krishna, J. Prasad, N. Ravikumar, 2011, Acta crystallographica. Section E, Structure reports online.

Discovery of CC chemokine receptor-3 (CCR3) antagonists with picomolar potency.

G. Trainor, M. Covington, C. Decicco, 2005, Journal of medicinal chemistry.

Cutting edge: a dominant negative form of TNF-alpha converting enzyme inhibits proTNF and TNFRII secretion.

G. Wu, R. Newton, K. Solomon, 1999, Journal of immunology.

CC chemokine receptor-3 (CCR3) antagonists: improving the selectivity of DPC168 by reducing central ring lipophilicity.

I. Kariv, K. Vaddi, M. Covington, 2007, Bioorganic & medicinal chemistry letters.

Synthesis and evaluation of cis-3,4-disubstituted piperidines as potent CC chemokine receptor 2 (CCR2) antagonists.

D. J. Nelson, P. Scherle, Gengjie Yang, 2008, Bioorganic & medicinal chemistry letters.

Discovery of disubstituted cyclohexanes as a new class of CC chemokine receptor 2 antagonists.

D. J. Nelson, S. Mandlekar, P. Scherle, 2008, Journal of medicinal chemistry.

Selective Inhibition of Eosinophil Influx into the Lung by Small Molecule CC Chemokine Receptor 3 Antagonists in Mouse Models of Allergic Inflammation

K. McIntyre, S. Mandlekar, J. Trzăskos, 2006, Journal of Pharmacology and Experimental Therapeutics.

CCR3 antagonists: a potential new therapy for the treatment of asthma. Discovery and structure-activity relationships.

G. Trainor, M. Covington, C. Decicco, 2002, Bioorganic & medicinal chemistry letters.

Use of lacZ fusions to measure in vivo expression of the first three genes of the Escherichia coli unc operon

D. K. Hsu, K. Solomon, W. Brusilow, 1989, Journal of bacteriology.

Discovery and Pharmacological Characterization of a Novel Rodent-Active CCR2 Antagonist, INCB3344

P. Scherle, F. Baribaud, L. Leffet, 2005, The Journal of Immunology.

Selective Inhibition of Eosinophil Influx into the Lung by Small Molecule CCR3 Antagonists in Mouse Models of Allergic Inflammation

K. McIntyre, S. Mandlekar, J. Trzăskos, 2006 .

Discovery of INCB9471, a Potent, Selective, and Orally Bioavailable CCR5 Antagonist with Potent Anti-HIV-1 Activity.

P. Scherle, K. Vaddi, Joseph Glenn, 2010, ACS medicinal chemistry letters.

2,4-Disubstituted piperidines as selective CC chemokine receptor 3 (CCR3) antagonists: synthesis and selectivity.

G. Trainor, M. Covington, C. Decicco, 2006, Bioorganic & medicinal chemistry letters.

QSAR studies on diclofenac analogues as potent cyclooxygenase inhibitors using CoMFA and CoMSIA

S. S. Rajan, K. Solomon, K. Arvind, 2014, Medicinal Chemistry Research.

Semi-synthetic modification of nimbolide to 6-homodesacetylnimbin and 6-desacetylnimbin and their cytotoxic studies

S. S. Rajan, G. Anitha, S. Narasimhan, 2007, Journal of Asian natural products research.

Efficient catalyst-free Domino approach for the synthesis of novel 2-benzazepine derivatives in water

G. Krishna, K. Kumar, D. Rambabu, 2010 .

An efficient ultrasound promoted catalyst-free protocol for the synthesis of chromeno[4,3-b]quinolin-6-ones

J. Prasad, K. Solomon, G. Gopikrishna, 2011 .

Photochemically enhanced binding of small molecules to the tumor necrosis factor receptor-1 inhibits the binding of TNF-α

D. Underwood, P. Domaille, K. Ramnarayan, 2001, Proceedings of the National Academy of Sciences of the United States of America.

An Efficient Ultrasound Promoted Catalyst‐Free Protocol for the Synthesis of Chromeno[4,3‐b]quinolin‐6‐ones (III).

J. Prasad, K. Solomon, G. Gopikrishna, 2012 .

Capped diaminopropionamide-glycine dipeptides are inhibitors of CC chemokine receptor 2 (CCR2).

P. Scherle, A. Tebben, Gengjie Yang, 2007, Bioorganic & medicinal chemistry letters.

Enhanced solubility, permeability, and tabletability of nicorandil by salt and cocrystal formation

N. Shastri, A. Nangia, Anurag Lodagekar, 2021 .

Molecular salts of 2,6-dihydroxybenzoic acid (2,6-DHB) with N-heterocycles: Crystal structures, spectral properties and Hirshfeld surface analysis

O. Blacque, K. Solomon, Ramanathan Venkatnarayan, 2017 .

Vibrational and electronic absorption spectra of (Z)-2-(4-nitrobenzylidene)-1-benzofuran-3(2H)-one

V. Veeraiah, G. Krishna, K. Chaitanya, 2012 .

Fluoroquinolone salts with carboxylic acids.

K. A. Kumar, A. Nangia, R. Dandela, 2011, Journal of pharmaceutical sciences.

Synthesis, crystal structure, spectral characterization and fluorescence studies of salts of α-mangostin with APIs

S. S. Rajan, N. Ravikumar, K. Solomon, 2013 .

From rigid cyclic templates to conformationally stabilized acyclic scaffolds. Part I: the discovery of CCR3 antagonist development candidate BMS-639623 with picomolar inhibition potency against eosinophil chemotaxis.

I. Kariv, S. Mandlekar, A. Tebben, 2008, Bioorganic & medicinal chemistry letters.

Discovery and structure-activity relationship of N-(ureidoalkyl)-benzyl-piperidines as potent small molecule CC chemokine receptor-3 (CCR3) antagonists.

G. Trainor, M. Covington, C. Decicco, 2002, Journal of medicinal chemistry.

Discovery and Pharmacological Characterization of a Novel Rodent-Active CCR2 Antagonist, INCB3344

P. Scherle, F. Baribaud, T. Burn, 2005, The Journal of Immunology.

INCB16562, a JAK1/2 selective inhibitor, is efficacious against multiple myeloma cells and reverses the protective effects of cytokine and stromal cell support.

J. Fridman, Jun Li, X. Wen, 2010, Neoplasia.

Mutations in the C-terminal hydrophobic domain of pseudorabies virus gIII affect both membrane anchoring and protein export

L. Enquist, A. Robbins, K. Solomon, 1991, Journal of virology.

Naftopidil Molecular Salts with Improved Dissolution and Permeation

A. Nangia, Srinu Tothadi, R. Dandela, 2020 .

Biology of TACE inhibition

K. Vaddi, M. Covington, P. Haley, 2001, Annals of the rheumatic diseases.

Detailed molecular structure (XRD), conformational search, spectroscopic characterization (IR, Raman, UV, fluorescence), quantum mechanical properties and bioactivity prediction of a pyrrole analogue

Renjith Thomas, K. Srikanth, T. Pooventhiran, 2020, Heliyon.

UseoflacZFusions ToMeasureInVivoExpression oftheFirst ThreeGenesoftheEscherichia coli uncOperon

K. Solomon, W. Brusilow, W. Hsu, 1989 .

IN-SILICO INTERACTION STUDIES ON INHIBITORY ACTION OF TETRANORTRITERPENOIDS ON ACTIN

S. S. Rajan, K. Solomon, K. Arvind, 2012 .

Effect of an uncE ribosome-binding site mutation on the synthesis and assembly of the Escherichia coli proton-translocating ATPase.

K. Solomon, W. Brusilow, K A Solomon, 1988, The Journal of biological chemistry.

The fate of pro-TNF-alpha following inhibition of metalloprotease-dependent processing to soluble TNF-alpha in human monocytes.

M. Covington, C. Decicco, R. Newton, 1997, Journal of immunology.

3,3′-[(4-Nitrophenyl)methylene]bis(4-hydroxy-2H-chromen-2-one)

N. Ravikumar, K. Solomon, G. Gopikrishna, 2012, Acta crystallographica. Section E, Structure reports online.

Purification and cloning of aggrecanase-1: a member of the ADAMTS family of proteins.

R. Wynn, R. Copeland, R. Wynn, 1999, Science.

Structural, spectroscopic (FT-IR, FT-Raman) and theoretical studies of the 1:1 cocrystal of isoniazid with p-coumaric acid

N. Ravikumar, K. Solomon, Gopikrishna Gaddamanugu, 2013 .

Characterization of a Novel Rodent-Active Discovery and Pharmacological

P. Scherle, F. Baribaud, L. Leffet, 2013 .

Isoxazolines as Potent Antagonists of the Integrin αvβ3

P. Jadhav, J. Wityak, S. Mousa, 2000 .

Quantitation of cellular receptors by a new immunocytochemical flow cytometry technique.

R. Zagursky, A. Schwartz, K. Solomon, 1995, BioTechniques.