G. Lucente

发表

4-Amino-1,2-dithiolane-4-carboxylic acid (Adt) as cysteine conformationally restricted analogue. Synthetic protocol for Adt containing peptides.

E. Morera, M. Nalli, F. Pinnen, 2000, Bioorganic & medicinal chemistry letters.

Novel chemotactic For-Met-Leu-Phe-OMe (fMLF-OMe) analogues based on met residue replacement by 4-amino-proline scaffold: synthesis and bioactivity.

A. Mollica, D. Torino, S. Spisani, 2009, Bioorganic & medicinal chemistry.

Synthesis, conformation and biological activity of centrally modified pseudopeptidic analogues of For-Met-Leu-Phe-OMe

A. Masi, A. Sansone, S. Spisani, 2007, Amino Acids.

Hybrid α/β-peptides: For-Met-Leu-Phe-OMe analogues containing geminally disubstituted β2,2- and β3,3-amino acids at the central position

A. Mollica, D. Torino, S. Spisani, 2006, Amino Acids.

Modified chemotactic peptides: Synthesis and activity of an azaTic-containing fMLP-OMe analogue

S. Spisani, G. Lucente, G. Pagani Zecchini, 2005, Amino Acids.

β-Peptido sulfonamides: for-Met-Leu-Phe-OMe analogues containing taurine and chiral β-amino-ethanesulfonic acid residues

M. Nalli, A. Sansone, S. Spisani, 2004 .

Synthesis and activity of HCO-Met-Leu-Phe-OMe analogues containing beta-alanine or taurine at the central position.

K. Varani, M. Nalli, S. Spisani, 2003, Farmaco.

Exploring the interest of 1,2-dithiolane ring system in peptide chemistry. Synthesis of a chemotactic tripeptide and x-ray crystal structure of a 4-amino-1,2-dithiolane-4-carboxylic acid derivative.

G. Ortar, E. Morera, M. Nalli, 2002, Bioorganic & medicinal chemistry.

Synthesis and activity on human neutrophil functions of fMLF-OMe analogs containing alkyl spacers at the central position.

E. Morera, M. Nalli, S. Spisani, 2001, Farmaco.

Bioactive fMLF-OMe analogs containing a N-terminal oximic or formylhydrazonic moiety.

S. Spisani, G. Lucente, M. Paglialunga Paradisi, 2000, The journal of peptide research : official journal of the American Peptide Society.

Biscarbamate analogues of the chemotactic tripeptide fMLF-OMe.

M. Nalli, S. Spisani, G. Lucente, 2000, Farmaco.

Chemotactic Peptide Analogues Centrally Constrained Chemotactic N‐Formyltripeptides: Synthesis, Conformation, and Activity of Two New Analogues

M. Paci, S. Spisani, G. Lucente, 1996 .

Modified chemotactic peptides: Synthesis, conformation, and biological activity of for‐Thp‐Leu‐ΔzPhe‐OMe

G. Cerichelli, G. Pochetti, S. Traniello, 1994 .

Modified chemotactic peptides: synthesis, crystal conformation, and activity of For‐Hse(Me)‐Leu‐Phe‐OMe

G. Pochetti, S. Traniello, S. Spisani, 1994, Biopolymers.

Cyclic Analogs of Chemotactic Formylpeptides, I.: Synthesis and Biological Activity of For‐Cys‐Leu‐Phe‐Cys‐OMe

S. Traniello, S. Spisani, G. Lucente, 1993, Archiv der Pharmazie.

Synthesis and Chemotactic Activity of the fMLP Analog HCO‐Hmb‐Leu‐Phe‐OMe

S. Traniello, S. Spisani, G. Lucente, 1993, Archiv der Pharmazie.

Synthesis and biological evaluation of new active For‐Met‐Leu‐Phe‐OMe analogues containing para‐substituted Phe residues

A. Mollica, A. Stefanucci, S. Spisani, 2012, Journal of peptide science : an official publication of the European Peptide Society.

Peptide backbone folding induced by the C(alpha)-tetrasubstituted cyclic alpha-amino acids 4-amino-1,2-dithiolane-4-carboxylic acid (Adt) and 1-aminocyclopentane-1-carboxylic acid (Ac5c). A joint computational and experimental study.

A. Mollica, E. Morera, M. Aschi, 2003, Organic & biomolecular chemistry.

New potent biphalin analogues containing p-fluoro-l-phenylalanine at the 4,4′ positions and non-hydrazine linkers

V. Hruby, A. Mollica, A. Stefanucci, 2011, Amino Acids.

Prevention of peroxynitrite-dependent damage by carnosine and related sulphonamido pseudodipeptides

M. Fontana, L. Pecci, F. Pinnen, 2002, Cellular and Molecular Life Sciences CMLS.

Peptides containing 4‐amino‐1,2‐dithiolane‐4‐carboxylic acid (Adt): conformation of Boc‐Adt‐Adt‐NHMe and NH ⃛S interactions

A. Mollica, E. Morera, M. Aschi, 2005, Journal of peptide science : an official publication of the European Peptide Society.

Synthesis of 1,2-dithiolane analogues of leucine for potential use in peptide chemistry.

E. Morera, F. Pinnen, G. Lucente, 2002, Organic letters.

Biochemical properties of new synthetic carnosine analogues containing the residue of 2,3-diaminopropionic acid: the effect of N-acetylation

M. Fontana, L. Pecci, I. Cacciatore, 2005, Amino Acids.

Topographically constrained aromatic α-aza-amino acids. Part 2. New azaTic-containing peptides: Synthesis, conformation, and intramolecular NH…N interaction

F. Mazza, G. Lucente, G. Mastropietro, 1999 .

Synthesis and activity of fibrillogenesis peptide inhibitors related to the 17-21 beta-amyloid sequence.

R. Chiaraluce, V. Consalvi, A. Masi, 2009, European journal of medicinal chemistry.

α-Peptide/β-sulfonamidopeptide hybrids: Analogs of the chemotactic agent for-Met-Leu-Phe-OMe

A. Masi, A. Sansone, S. Spisani, 2006 .

Chemotactic peptides: fMLF-OMe analogues incorporating proline-methionine chimeras as N-terminal residue.

A. Mollica, K. Varani, S. Spisani, 2006, Bioorganic & medicinal chemistry.

Peptides containing the sulfonamide junction. 2. Structure and conformation of Z-Tau-Pro-D-Phe-NHiPr.

E. Morera, F. Mazza, A. Calcagni, 2000, Biopolymers.

Synthesis and evaluation of new endomorphin analogues modified at the Pro(2) residue.

V. Hruby, A. Mollica, D. Torino, 2009, Bioorganic & medicinal chemistry letters.

α-Hydroxymethylation of Schiff Bases Derived from α-Amino Acid Esters

A. Calcagni, D. Rossi, G. Lucente, 1981 .

Bicyclic peptides: Solution conformation and Ca2+ binding of the heterodetic bicyclic decapeptide cyclo(Glu1‐Leu2‐Pro3‐Gly4‐Ser5‐Ile6‐Pro7‐Ala8)‐cyclo(1γ → 5β) Phe9‐Gly10

L. Paolillo, F. Pinnen, G. Lucente, 1989 .

Conformationally Constrained Histidines in the Design of Peptidomimetics: Strategies for the χ-Space Control

A. Mollica, A. Stefanucci, I. Cacciatore, 2011, International journal of molecular sciences.

On the trapping of sulphenic acids from penicillin sulphoxides

P. G. Sammes, D. Barton, G. Lucente, 1970 .

A convenient route to pyrrolidine-2-phosphonic acid dipeptides

G. Lucente, M. P. Paradisi, I. Torrini, 2009 .

Male fertility: core chemical structure in pharmacological research.

B. Silvestrini, M. Bonanomi, G. Lucente, 2002, Contraception.

Synthesis of peptides containing 1,2,3,4-tetrahydroquinoline-2-carboxylic acid. Part 2. Crystal and molecular structure of a 1H,3H,5H-oxazolo[3,4-a]quinolin-3-one derivative obtained from a linear tripeptide

W. Fedeli, F. Mazza, G. Lucente, 1979 .

Synthesis of 2-alkoxy-2-phenylacetamido-carboxylic acids

F. Pantanella, G. Lucente, A. Romeo, 1967 .

Proline-glutamate chimeras in isopeptides. Synthesis and biological evaluation of conformationally restricted glutathione analogues.

A. Mollica, A. Caccuri, A. Di Stefano, 2003, Bioorganic & medicinal chemistry.

Design and synthesis of glutathione analogues.

G. Luisi, F. Pinnen, G. Lucente, 1998, Farmaco.

cis-4-amino-L-proline residue as a scaffold for the synthesis of cyclic and linear endomorphin-2 analogues: part 2.

V. Hruby, A. Mollica, L. Mannina, 2012, Journal of medicinal chemistry.

Synthesis, stereochemistry and conformational properties of diastereomeric cyclic dipeptides containing tetrahydro-1,4-thiazine-3,5-dicarboxylic acid

G. Lucente, M. P. Paradisi, I. Torrini, 1990 .

Synthesis and properties of chemotactic peptide analogs. I. Crystal structure and molecular conformation of HCO-Met-leu-Ain-OMe.

G. Pochetti, F. Mazza, G. Lucente, 2009, International journal of peptide and protein research.

Synthesis and activity of endomorphin-2 and morphiceptin analogues with proline surrogates in position 2.

V. Hruby, A. Mollica, A. Masi, 2010, European journal of medicinal chemistry.

Retrosulfonamido peptide analogues. Synthesis and crystal conformation of Boc-Pro-Leu-Ψ(NH-SO2)-Gly-NH2

G. Pochetti, F. Mazza, G. Lucente, 1991 .

Structure and conformation of peptides containing the sulphonamide junction. III. Synthesis, crystal and molecular structure of a taurine containing peptidic oxa-cyclol.

G. Pochetti, F. Mazza, F. Pinnen, 2009, International journal of peptide and protein research.

Structure and conformation of peptides containing the sulphonamide junction. I. N-acetyl-tauryl-L-phenylalanine methyl ester.

G. Pochetti, F. Mazza, A. Calcagni, 2009, International journal of peptide and protein research.

Structure and conformation of peptides containing the sulfonamide junction. II. Synthesis and conformation of cyclo[-MeTau-Phe-DPro-].

G. Pochetti, F. Mazza, F. Pinnen, 2009, International journal of peptide and protein research.

Synthesis and activity of the glutathione analogue γ‐(L‐γ‐azaglutamyl)‐L‐cysteinyl‐glycine

G. Luisi, S. Dupré, F. Pinnen, 2009 .

Synthesis and Activity of the Glutathione Analogue γ‐(L‐γ‐Oxaglutamyl)‐L‐cysteinyl‐glycine

G. Luisi, S. Dupré, F. Pinnen, 1996 .

Conformational properties of β-residue-containing oligopeptides in apolar solvent

A. Mollica, M. Aschi, F. Mazza, 2006 .

Chemotactic tripeptides incorporating at position 2 α-aminoacid residues with unsaturated side chains

D. Torino, A. Sansone, S. Spisani, 2008, Amino Acids.

Isopeptide bonds in chemotactic tripeptides. Synthesis and activity of lysine-containing fMLF analogs.

A. Mollica, M. Nalli, S. Spisani, 2002, The journal of peptide research : official journal of the American Peptide Society.

Peptides containing the sulfonamide junction: Synthesis, structure, and conformation of Z-Tau-Pro-Phe-NHiPr

M. Paci, G. Luisi, G. Pochetti, 1997 .

Cyclization of activated tosyl-peptides

G. Lucente, P. Frattesi, 1972 .

Synthesis of cyclols from some small peptides via amide–amide reaction

G. Lucente, A. Romeo, 1971 .

Cyclols-formation from tripeptide systems and structure assignment by carbon-13 nuclear magnetic resonance.

F. Conti, G. Lucente, G. Zanotti, 2009, International journal of peptide and protein research.

Evidence for a base catalyzed interconversion of azacyclols derived from N-(acylalanyl)-phenylalanyl-prolin-lactams

G. Lucente, G. Zanotti, A. Romeo, 2005, Experientia.

Approaches to pseudopeptidic ergopeptines. Part 3.1 Consequences of the incorporation of an α-azaphenylalanine residue into the ergotamine oxa-cyclolic system

G. Luisi, F. Pinnen, A. Calcagni, 1997 .

Synthesis and x-ray crystal structure of a tripeptidic cyclol

W. Fedeli, F. Pinnen, G. Lucente, 1981 .

Cyclization of activated N-benzyloxycarbonyl-tripeptides

F. Pinnen, G. Lucente, G. Zanotti, 1978 .

Approaches to pseudopeptidic ergopeptines. Synthesis and molecular structure of an α-aza-phenylalanine-containing oxa-cyclol

G. Luisi, F. Pinnen, G. Lucente, 1993 .

Cyclols, cyclodepsipeptides, and N-acyl-diketopiperazines from linear precursors. Synthesis and crystal structure of 10-membered cyclodepsipeptides.

F. Mazza, F. Pinnen, G. Lucente, 2009, International journal of peptide & protein research.

Approach to the use of benzylpenicillinacylase for configurational correlations of amino compounds

D. Rossi, G. Lucente, A. Romeo, 1978 .

Azacyclols from n-(2-denzyloxycarbonylamino-acyl)-lactams

G. Lucente, G. Zanotti, P. Frattesi, 1973 .

Ten-membered cyclotripeptides: II. Synthesis and crystal structure of cyclo(-β-alanyl-L-phenylalanyl-L-prolyl-)

F. Pinnen, G. Lucente, E. Gavuzzo, 2009 .

Cyclization under mild conditions of anthraniloyl- and N-methyl-anthraniloyl dipeptides.

A. Di Muro, F. Pinnen, G. Lucente, 2009, International journal of peptide and protein research.

Cyclization under mild conditions of cysteine containing peptides

F. Pinnen, G. Lucente, G. Zanotti, 1985 .

Ten-membered cyclotripeptides: Influence of the ring-flexibility on intramolecular reactions

F. Pinnen, G. Lucente, G. Zanotti, 1985 .

APPROACHES TO PSEUDOPEPTIDIC ERGOPEPTINES. PART 3. CONSEQUENCES OF THE INCORPORATION OF AN ALPHA -AZAPHENYLALANINE RESIDUE INTO THE ERGOTAMINE OXA-CYC LOLIC SYSTEM

G. Luisi, F. Pinnen, A. Calcagni, 1997 .

Cyclization under mild conditions of salicyloyl-dipeptides.

G. Luisi, F. Pinnen, A. Calcagni, 2009, International journal of peptide and protein research.

N-Acyl-diketopiperazines. II: Crystal structure and conformation of N-(pyruvoyl)-cyclo-(L-phenylalanyl-D-prolyl)

G. Pochetti, F. Mazza, A. Calcagni, 2009 .

Approaches to pseudopeptidic ergopeptines. Part 2. Consequences of the incorporation of an α-azaproline residue into the oxacyclolic system

G. Luisi, F. Pinnen, A. Calcagni, 1994 .

Endoannular interactions in cysteine-containing cyclotripeptides: one-step synthesis and crystal structure of a tetracyclic aza-cyclol

F. Pinnen, G. Lucente, E. Gavuzzo, 1988 .

Peptidic thiacyclols. Synthesis and structural studies

W. Fedeli, F. Mazza, F. Pinnen, 1984 .

Peptide cyclols. Crystal structure and molecular conformation of the oxacyclol derived from L-2-hydroxyisovaleryl-L-phenylalanyl-L-proline

A. Segre, W. Fedeli, F. Mazza, 1982 .

Cyclol formation from tripeptides containing β-alanine

F. Pinnen, G. Lucente, G. Zanotti, 1982 .

Peptidic cyclols. Synthesis, and crystal and molecular structure of a tricyclic thia-cyclol

W. Fedeli, F. Mazza, F. Pinnen, 1980 .

Ten-membered cyclotripeptides: Crystal structure and conformation of cyclo(-N-methylanthraniloyl-L-phenylalanyl-L-prolyl-)

F. Pinnen, G. Lucente, E. Gavuzzo, 2009 .

Ten-membered cyclotripeptides. III. Synthesis and conformation of cyclo(-Me beta Ala-Phe-Pro-) and cyclo(-Me beta Ala-Phe-DPro-).

G. Luisi, F. Pinnen, G. Lucente, 2009, International journal of peptide and protein research.

Structure-activity relationships of biphalin analogs and their biological evaluation on opioid receptors.

A. Mollica, A. Stefanucci, I. Cacciatore, 2012, Mini reviews in medicinal chemistry.

Pseudopeptides containing the 2-hydrazonoacyl fragment: analogs of the chemotactic agent HCO-Met-Leu-Phe-OMe.

M. Nalli, S. Spisani, I Torrini, 2001, The journal of peptide research : official journal of the American Peptide Society.

Synthesis and properties of chemotactic peptide analogs

G. Pochetti, A. Giuliani, F. Mazza, 2009 .

The use of benzylpenicillinacylase fromEscherichia coli in the resolution of some racemicβ-,γ-,δ- andɛ-amino-acids

D. Rossi, G. Lucente, A. Romeo, 1977, Experientia.

Use ofEscherichia coli A.T.C.C. 9637 for the asymmetric hydrolysis of amino acid derivatives

D. Rossi, G. Lucente, A. Romeo, 1965, Experientia.

Hydrolysis of N-phenylacetyl derivatives of amino compounds by benzylpenicillin-acylase. Steric course of the reaction

D. Rossi, G. Lucente, G. Zanotti, 1971 .

Antinociceptive profile of potent opioid peptide AM94, a fluorinated analogue of biphalin with non‐hydrazine linker

A. Mollica, A. Stefanucci, S. Pieretti, 2013, Journal of peptide science : an official publication of the European Peptide Society.

The cis-4-amino-L-proline residue as a scaffold for the synthesis of cyclic and linear endomorphin-2 analogues.

V. Hruby, A. Mollica, Cristina Campestre, 2012, Journal of medicinal chemistry.

N-acyl-diketopiperazines: crystal structure and conformation of N-(N-phenylacetyl-L-alanyl)-cyclo-(L-phenylalanyl-D-prolyl)

W. Fedeli, F. Mazza, F. Pinnen, 2009 .

Synthesis and structural studies of N‐p‐toluensulfonyl cyclodipeptides

G. Pochetti, F. Mazza, A. Calcagni, 1989, Biopolymers.

Potential energy calculations on phenylalanine rotamers in different boat forms of proline-containing cyclic dipeptides.

G. Pochetti, F. Mazza, G. Lucente, 2009, International journal of peptide & protein research.

Peptide azacyclols from linear precursors

F. Pinnen, G. Lucente, G. Zanotti, 1983 .

Nine-membered cyclodepsitripeptides containing the retroisomeric sequence of ergot peptides.

G. Luisi, F. Pinnen, A. Calcagni, 2009, International journal of peptide and protein research.

Investigation of amino acid containing [FeFe] hydrogenase models concerning pendant base effects.

H. Görls, B. Keppler, W. Weigand, 2009, Journal of inorganic biochemistry.

γ-Turn conformation induced by α,α-disubstituted amino acids with a cyclic six-membered side chain

G. Pochetti, F. Mazza, G. Lucente, 1995 .

Use of Escherichia coli A.T.C.C. 9637 for the asymmetric hydrolysis of amino acid derivatives.

D. Rossi, G. Lucente, A. Romeo, 1965, Experientia.

Synthesis, conformation, and biological activity of two fMLP‐OMe analogues containing the new 2‐[2′‐(methylthio) ethyl] methionine residue

G. Pochetti, S. Traniello, S. Spisani, 1997, Biopolymers.

Rearrangements of penicillin sulphoxides

P. G. Sammes, D. Barton, G. Lucente, 1970 .

Synthesis and evaluation of new endomorphin-2 analogues containing (Z)-alpha,beta-didehydrophenylalanine (Delta(Z)Phe) residues.

V. Hruby, A. Mollica, D. Torino, 2010, Journal of medicinal chemistry.

Cyclic dipeptides containing proline. Structure and conformation of cyclo(-L-Phe-L-Pro-), C14H16N2O2

F. Mazza, F. Pinnen, G. Lucente, 1984 .

Modified chemotactic peptides: synthesis, conformation, and activity of HCO-Thp-Ac6c-Phe-OMe.

G. Pochetti, S. Traniello, S. Spisani, 1998, Biopolymers.

For‐Met‐Lys‐Phe‐ For‐Met‐Lys‐Phe‐: A new cyclic analogue of the chemotactic formylpeptides

G. Pochetti, S. Traniello, S. Spisani, 1995, Biopolymers.

X-ray crystal structure and conformation of N-(tert-butyloxycarbonyl)-L-methionyl-(1-aminocyclopent-3-ene-1-carbonyl)-L-phenylalanine methyl ester (Boc0-Met1-Cpg2-Phe3-OMe)

A. Mollica, D. Torino, M. Camalli, 2009 .

Synthesis, conformation, and activity of HCO‐Met‐ΔZ Leu‐Phe‐Ome, an active analogue of chemotactic N‐formyltripeptides

G. Veglia, M. Paci, G. Pochetti, 1993, Biopolymers.