R. Escale

发表

Metalation and halogen‐metal exchange in the imidazo[1,2‐a]quinoxaline series

G. Subra, P. Bonnet, C. Deleuze-Masquéfa, 2001 .

Synthesis and antimalarial activity of new 1,12-bis(N,N'-acetamidinyl)dodecane derivatives.

H. Vial, S. Wein, M. Ouattara, 2007, Bioorganic & medicinal chemistry letters.

Potent antimalarial activity of 2-aminopyridinium salts, amidines, and guanidines.

H. Vial, M. Ancelin, Y. Bordat, 2007, Journal of medicinal chemistry.

Symmetrical choline-derived dications display strong anti-kinetoplastid activity.

Terry K. Smith, N. Quashie, H. D. de Koning, 2011, The Journal of antimicrobial chemotherapy.

Synthesis and Evaluation of Hybrid Bis‐cationic Salts as Antimalarial Drugs

H. Vial, T. Durand, S. Denoyelle, 2010, ChemMedChem.

Synthesis and contractile activity of new pseudopeptido and thioaromatic analogues of leukotriene D4.

T. Durand, J. Girard, C. Bonne, 1992, Prostaglandins.

Synthesis of a new pseudopeptidoleukotriene : The first LTD4 analogue with potent agonist activity

J. Girard, J. Rossi, R. Escale, 1991 .

Substituted cyclohexane as conformationally-restricted analogues of the peptido-leukotrienes

J. Girard, J. Rossi, R. Escale, 1989 .

Evaluation of amidoxime derivatives as prodrug candidates of potent bis-cationic antimalarials.

H. Vial, F. Bressolle, T. Durand, 2019, Bioorganic & medicinal chemistry letters.

Aza-indolizine with bridgehead nitrogen. Metalation, halogen-metal exchange and directed ortho-lithiation in the imidazo[1,2-a]pyrazine series

G. Subra, P. Bonnet, O. Vitse, 1998 .

Nucleophilic aromatic substitution reaction of some 3-nitroimidazo[1,2-a]pyridines with thioglycolate anion in DMF

G. Grassy, J. Teulade, R. Escale, 1981 .

New aspects of the nitration of some imidazo[1,2-a]pyridines. CNDO/2 calculations from X-ray structures

G. Grassy, J. Teulade, M. Payard,, 1982 .

Synthesis of tert‐Butoxycarbonyl‐Protected α‐Hydrazino Phosphonic Diesters by Electrophilic Amination with Di‐tert‐butyl Azodicarboxylate.

P. Dumy, J. Girard, J. Vidal, 1994 .

Lituarines A, B, and C: a new class of macrocyclic lactones from the New Caledonian sea pen Lituaria australasiae

J. Girard, A. Aumelas, J. Rossi, 1992 .

Synthetic phosphonamidate pseudopeptide

P. Dumy, J. Girard, J. Parello, 1991 .

A rational approach to the synthesis of phosphonamidate peptides

P. Dumy, J. Girard, R. Escale, 1994, Letters in Peptide Science.

A convenient synthetic approach to new α-(9-fluorenylmethoxycarbonylamino)alkylphosphonic acid derivatives

P. Dumy, J. Girard, J. Parello, 1992 .

Solid phase synthesis of phosphonopeptides from Fmoc phosphonodipeptides

P. Dumy, J. Girard, R. Escale, 1994 .

Development of the First Oral Bioprecursors of Bis‐alkylguanidine Antimalarial Drugs

H. Vial, T. Durand, M. Maynadier, 2014, ChemMedChem.

Strained cyclobutane compounds: 1H NMR analysis of a new 1‐substituted benzobicyclo[3.1.1]heptene system

J. Rossi, R. Escale, J. Chapat, 1981 .

Caulerpin, Caulerpicin, Caulerpa scalpelliformis: Comparative Acute Toxicity Study

J. Girard, D. Laurent, J. Rossi, 1984 .

Cyclisation reactions of some 3-nitrosoimidazo[1,2-a]-pyridines and-pyrimidines. Ring-opening/ring-closure reactions with triethyl phosphite: reassignment by X-ray crystal structure and nuclear magnetic resonance

J. Leger, G. Grassy, J. Teulade, 1983 .

Solution Parallel Synthesis of Cyclic Guanidines

P. Bonnet, J. Bompart, R. Escale, 2000 .

Imidazo[1,2-a]quinoxalines: synthesis and cyclic nucleotide phosphodiesterase inhibitory activity.

J. Vidal, P. Bonnet, A. Michel, 2001, European journal of medicinal chemistry.

Evaluation of Bis‐Alkylamidoxime O‐Alkylsulfonates as Orally Available Antimalarials

H. Vial, T. Durand, S. Wein, 2012, ChemMedChem.

Solution Parallel Synthesis of Cyclic Guanidines.

P. Bonnet, J. Bompart, R. Escale, 2000 .

A convenient Fmoc synthesis of phosphonamidate peptide

P. Dumy, J. Girard, J. Parello, 1993 .

Pharmacokinetic properties and metabolism of a new potent antimalarial N-alkylamidine compound, M64, and its corresponding bioprecursors.

H. Vial, F. Bressolle, Florence Gattacceca, 2011, European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences.

Evidence for the existence of high affinity binding sites for indomethacin on human blood platelets.

J. Girard, J. Bali, R. Magous, 1986, Molecular Pharmacology.

Ibogaine and Noribogaine: Structural Analysis and Stability Studies. Use of LC‐MS to Determine Alkaloid Contents of the Root Bark of Tabernanthe Iboga

L. Balas, R. Escale, J. Blayac, 2007 .

N-substituted bis-C-alkyloxadiazolones as dual effectors: efficient intermediates to amidoximes or amidines and prodrug candidates of potent antimalarials.

T. Durand, S. Wein, M. Degardin, 2009, Bioorganic & medicinal chemistry letters.

Mass spectra of new 3,5‐methano‐2,3,4,5‐tetrahydro‐1H‐1 and ‐2 benzazepines and oxo drivatives

J. Rossi, R. Escale, J. Vidal, 1986 .