K. Kraus

发表

Isoxazolyl, oxazolyl, and thiazolylpropionic acid derivatives as potent α4β1 integrin antagonists

A. Milici, A. Duplantier, L. Chupak, 2001 .

Biarylcarboxylic acids and -amides: inhibition of phosphodiesterase type IV versus [3H]rolipram binding activity and their relationship to emetic behavior in the ferret.

A. Marfat, J. Cheng, H. Masamune, 1996, Journal of medicinal chemistry.

Optimization of the physicochemical and pharmacokinetic attributes in a 6-azauracil series of P2X7 receptor antagonists leading to the discovery of the clinical candidate CE-224,535.

A. Kalgutkar, C. Gabel, R. Shepard, 2011, Bioorganic & medicinal chemistry letters.

Pulmonary Eosinophilia in a Murine Model of Allergic Inflammation Is Attenuated by Small Molecule α4β1 Antagonists

A. Milici, C. Andresen, A. Duplantier, 2002 .

Synthesis and in vitro profile of a novel series of catechol benzimidazoles. The discovery of potent, selective phosphodiesterase type IV inhibitors with greatly attenuated affinity for the [3H]rolipram binding site

James F. Eggler, A. Marfat, H. Masamune, 1995 .

SAR of a series of 5,6-dihydro-(9H)-pyrazolo[3,4-c]-1,2,4-triazolo[4,3-alpha]pyridines as potent inhibitors of human eosinophil phosphodiesterase.

John B. Cheng, A. Duplantier, T. H. Jenkinson, 2007, Journal of medicinal chemistry.

Pulmonary eosinophilia in a murine model of allergic inflammation is attenuated by small molecule alpha4beta1 antagonists.

A. Milici, C. Andresen, A. Duplantier, 2002, The Journal of pharmacology and experimental therapeutics.

1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-phenylpiperidines as mGluR2 positive allosteric modulators for the treatment of psychosis.

A. Ganong, F. Tingley, J. Siuciak, 2011, Journal of medicinal chemistry.

Rotationally restricted mimics of rigid molecules: nonspirocyclic hydantoin aldose reductase inhibitors.

P. Kelbaugh, K. Kraus, R. Schnur, 1989, Journal of medicinal chemistry.

3-Benzyl-1,3-oxazolidin-2-ones as mGluR2 positive allosteric modulators: Hit-to lead and lead optimization.

Lei Zhang, John Candler, Ivan Efremov, 2009, Bioorganic & medicinal chemistry letters.

7-Oxo-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridines as novel inhibitors of human eosinophil phosphodiesterase.

F. Dicapua, J. Cheng, A. Williams, 1998, Journal of medicinal chemistry.