S. Archer

发表

Nitrocinnamoyl and chlorocinnamoyl derivatives of dihydrocodeinone: in vivo and in vitro characterization of mu-selective agonist and antagonist activity.

J. Bidlack, J. McLaughlin, K. Hill, 1999, The Journal of pharmacology and experimental therapeutics.

Metopon and two unique derivatives: affinity and selectivity for the multiple opioid receptors.

D. Nowak, J. Bidlack, J. McLaughlin, 1995, European journal of pharmacology.

Antischistosomal drugs: past, present ... and future?

D. Cioli, S. Archer, L. Pica-Mattoccia, 1995, Pharmacology & therapeutics.

Suppression of morphine and cocaine self-administration in rats by a mixed mu antagonist-kappa agonist (N-CBM-TAMO) and a long-acting selective D1 antagonist (AS-300)

S. D. Glick, J. Bidlack, M. Teitler, 1996 .

Binding of oxamniquine to the DNA of schistosomes.

D. Cioli, S. Archer, L. Pica-Mattoccia, 1989, Transactions of the Royal Society of Tropical Medicine and Hygiene.

The chemotherapy of schistosomiasis.

S. Archer, 1985, Annual review of pharmacology and toxicology.

Hycanthone, a new active metabolite of lucanthone.

D. Rosi, S. Archer, G. Peruzzotti, 1967, Journal of medicinal chemistry.

Evidence for the mode of antischistosomal action of hycanthone.

D. Cioli, S. Archer, L. Pica-Mattoccia, 1985, Life sciences.

Preparation and antischistosomal and antitumor activity of hycanthone and some of its congeners. Evidence for the mode of action of hycanthone.

D. Cioli, S. Archer, L. Pica-Mattoccia, 1988, Journal of medicinal chemistry.

A New, Active Metabolite of ‘Miracil D’

D. Rosi, S. Archer, G. Peruzzotti, 1965, Nature.

14 beta-(Bromoacetamido)morphine irreversibly labels mu opioid receptors in rat brain membranes.

S. Archer, A. Seyed-Mozaffari, J. Bidlack, 1989, Biochemistry.

Drug resistance in schistosomes.

D. Cioli, S. Archer, L. Pica-Mattoccia, 1993, Parasitology today.

The Synthesis of Tryptophan from Gramine

S. Archer, C. Suter, N. Albertson, 1945 .

Synthesis and characterization of 4,4-difluoro-4-bora-3a,4a-diaza-s-indacene (BODIPY)-labeled fluorescent ligands for the mu opioid receptor.

H. Akil, P. Emmerson, A. Mansour, 1997, Biochemical pharmacology.

Arylacetamide kappa-selective opioid ligands

J. Bidlack, M. Wentland, A. D. Pechulis, 1997 .

Fluorescent staining of κ opioid receptors using naltrexamine derivatives and phycoerythrin

J. Bidlack, D. M. Lawrence, S. Archer, 1997 .

14β-Chlorocinnamoylamino derivatives of metopon : long-term μ-opioid receptor antagonists

J. Bidlack, J. McLaughlin, A. Sebastian, 1997 .

Antinociceptive evaluation of 14 beta-(bromoacetamido)-7,8-dihydro- N(cyclopropylmethyl)-normorphinone in mice.

J. Bidlack, Q. Jiang, S. Archer, 1993, European journal of pharmacology.

kappa opioid receptors in human microglia downregulate human immunodeficiency virus 1 expression.

K. Shark, J. Bidlack, W. Sheng, 1996, Proceedings of the National Academy of Sciences of the United States of America.

Augmentation of pharmacological properties of catecholamines by O-methyl transferase inhibitors.

S. Archer, A. Arnold, D. Wylie, 1960, The Journal of pharmacology and experimental therapeutics.

Photoaffinity ligands for the mu opioid receptor.

E. J. Simon, J. Hiller, S. Archer, 1993, Life sciences.

The Preparation of Some Iodinated Aminophenylalkanoic Acids

S. Archer, T. R. Lewis, 1949 .

Characterization of a polyclonal antibody to the μ opioid receptor

R. Zukin, R. Maneckjee, S. Archer, 1988, Journal of Neuroimmunology.

The preparation and cholecystographic properties of some aminotriiodophenylalkanoic acids.

S. Archer, J. O. Hoppe, T. R. Lewis, 1951, Journal of the American Pharmaceutical Association. American Pharmaceutical Association.

The Preparation of Some Iodinated Phenyl- and Pvridylalkanoic Acids†

S. Archer, J. O. Hoppe, T. R. Lewis, 1951 .

Narcotic Antagonists as Analgesics

L. Harris, A. Keats, S. Archer, 1962, Science.

SOME 14β-SUBSTITUTED ANALOGS OF N-(CYCLOPROPYLMETHYL)NORMORPHINE

H. Kosterlitz, S. Archer, M. Gillan, 1981 .

Some 14 beta-substituted analogues of N-(cyclopropylmethyl)normorphine.

H. Kosterlitz, S. Archer, M. Gillan, 1981, Journal of medicinal chemistry.

Diazotization of a 2-amino-1,3-selenazole

S. Archer, R. McGarry, 1982 .

A New Indole Synthesis1

S. Archer, B. Tullar, C. Koelsch, 1965 .

The Preparation and Some Reactions of Ethyl α-Acetamidoacetoacetate

J. King, S. Archer, B. Tullar, 1948 .

3α-(2-Diethylaminoethyl)-aminotropane and Related Compounds1,2

S. Archer, T. R. Lewis, M. Unser, 1957 .

The Chapman Rearrangement

S. Archer, J. W. Schulenberg, 2011 .

Synthesis of 6-substituted 7H-pyrido[4,3-c]carbazoles

S. Modi, S. Archer, A. Zayed, 1989 .

A NEW SYNTHESIS OF TRYPTOPHAN

S. Archer, C. Suter, N. Albertson, 1944 .

Notes - Preparation of Alkyl Vinyl Ketones

S. Archer, M. Unser, W. Dickinson, 1957 .

The Preparation of 2-Methyl-1-phenylbenzimidazole 3-Oxide

S. Archer, J. W. Schulenberg, 1965 .

Some 5-(Oxoalkyl)-2-thiohydantoins and Their Derivatives

S. Archer, E. Froelich, M. Unser, 1956 .

5-HEPTYL-2-THIOHYDANTION, A NEW ANTITUBERCULAR AGENT

E. J. Alexander, S. Archer, F. K. Kirchner, 1954 .

THE RACEMIZATION OF L(+)-2α-TROPANOL

M. Bell, S. Archer, T. R. Lewis, 1961 .

The preparation of some 6-substituted-2-thiouracils.

S. Archer, M. Jackman, A. J. Bergman, 1948, Journal of the American Chemical Society.

1-Ethyl-4-(3-tropanyl)-tetrahydro-1H-1,4-benzodiazepine

S. Archer, J. O. Hoppe, T. R. Lewis, 1957 .

Conformation of 3α-Phenyl-3β-tropanyl Phenyl Ketone; a Novel Nitrogen-Carbonyl Interaction

M. Bell, S. Archer, 1960 .

Factors Determining the Course and Mechanisms of Grignard Reactions. VIII. The Effect of Metallic Halides on the Reaction of Grignard Reagents with Aromatic Acyl Halides

S. Archer, M. Kharasch, W. Nudenberg, 1943 .

Methyl 3(α)-Acetoxy-11-ketocholanate

S. Archer, T. R. Lewis, M. Jackman, 1954 .

Analogues of hycanthone and lucanthone as antitumor agents.

R. Rej, S. Archer, T. Rugino, 1983, Journal of medicinal chemistry.

Synthesis of hycanthone

D. Rosi, S. Archer, G. Laidlaw, 1973 .

Chemistry of Nonpeptide Opioids

S. Archer, 1993 .

Synthesis and schistosomicidal acitivity of 6-chloro-5-[2-(diethylamino)ethyl]amino-8-quinolinemethanol.

D. Rosi, D. M. Bailey, S. Archer, 1970, Journal of medicinal chemistry.

Comparison of schistosomicidal activity of xanthenones and 4-methyl-3-chloroanilines and their hydroxymethyl analogs in Swiss mice and Syrian hamsters infected with Schistosoma mansoni.

D. Rosi, S. Archer, E. Dennis, 1969, Journal of medicinal chemistry.

Preparation and schistosomicidal activity of some 4-hydroxymethyl-3-chloroanilines.

D. Rosi, S. Archer, D. A. Berberian, 1967, Journal of medicinal chemistry.

A comparison of oral and parenteral activity of hycanthone and lucanthone in experimental infections with Schistosoma mansoni.

D. Rosi, S. Archer, E. Dennis, 1967, The American journal of tropical medicine and hygiene.

Schistosomicidal activity of lucanthone hydrochloride, hycanthone and their metabolites in mice and hamsters.

D. Rosi, S. Archer, E. Dennis, 1967, The Journal of parasitology.

Binding of tritiated hycanthone and hycanthone N-methylcarbamate to macromolecules of drug-sensitive and drug-resistant schistosomes.

D. Cioli, S. Archer, L. Pica-Mattoccia, 1988, Molecular and biochemical parasitology.

A possible metabolic basis for the schistosomicidal activity of Mirasan and N-(3-chloro-4-methylphenyl)-piperazine.

D. Rosi, A. Merola, S. Archer, 1967, Life sciences.

The Preparation of Some 1-Alkylamino- and Dialkylaminoalkylaminothiaxanthones1

S. Archer, C. Suter, 1952 .

An Abnormal Chapman Rearrangement

S. Archer, J. W. Schulenberg, 1960 .

The Use of Ethyl Acetamidomalonate in the Synthesis of Amino Acids. The Preparation of dl-Histidine, dl-Phenylalanine and dl-Leucine

S. Archer, N. Albertson, 1945 .

DOSE: RESPONSE EFFECTS ON NOREPINEPHRINE-DEPLETION OF RESERPINE AND OF GUANETHIDINE IN BRETYLIUM-PRETREATED RATS.

S. Archer, A. Arnold, J. P. McAuliff, 1963, Biochemical pharmacology.

PENTAZOCINE. STRONG ANALGESICS AND ANALGESIC ANTAGONISTS IN THE BENZOMORPHAN SERIES.

L. Harris, S. Archer, N. Albertson, 1964, Journal of medicinal chemistry.

The Alkylation of Benzene in the Presence of Acid Catalysts

S. Archer, R. Burwell, 1942 .

Napthoquinone antimalarials. XXX. 2-hydroxy-3-[omega-(1-adamantyl)alkyl]-1,4-naphthoquinones.

L. Fieser, S. Archer, D. A. Berberian, 1967, Journal of medicinal chemistry.

Naphthoquinone antimalarials. XXIX. 2-hydroxy-3-(omega-cyclohexylalkyl)-1,4-naphthoquinones.

L. Fieser, S. Archer, R. Lorenz, 1967, Journal of medicinal chemistry.

Ring-hydroxylated analogues of lucanthone as antitumor agents.

L. Fricker, R. Rej, K. J. Miller, 1982, Journal of medicinal chemistry.

Parasympatholytic (anticholinergic) esters of the isomeric 2-tropanols. 1. Glycolates.

E. Atkinson, M. Aceto, L. Harris, 1977, Journal of medicinal chemistry.

The enzymic methylation of pyrogallol.

R. Kullnig, S. Archer, A. Arnold, 1960, Archives of biochemistry and biophysics.

Narcotic Antagonists as Analgesics: Laboratory Aspects

L. Harris, S. Archer, B. Tullar, 1964 .

1-Acetamido-17-carbomethoxydihydrothebainone

S. Archer, C. W. Klinowski, K. Okaniwa, 1981 .

The preparation of some amides of 4,6-diaminoquinaldine.

S. Archer, M. Pratt, 1948, Journal of the American Chemical Society.

ISOMERIC 2-ACETOXYTROPINE METHIODIDES.

S. Archer, A. M. Lands, T. R. Lewis, 1962, Journal of medicinal and pharmaceutical chemistry.

Δ-(3,4-Dicarboxy)-furanvaleric and -acetic Acids

S. Archer, M. Pratt, 1944 .

Torsional motion and elasticity of the deoxyribonucleic acid double helix and its nucleosomal complexes.

C. Scholes, L. Lerman, S. Archer, 1982, Biochemistry.

The Preparation of 3-Iodoalizarin

S. Archer, M. Pratt, 1949 .

Identification of kappa opioid receptors in the immune system by indirect immunofluorescence.

J. Bidlack, J. Leary, D. M. Lawrence, 1995, Proceedings of the National Academy of Sciences of the United States of America.

Hydrogen Fluoride as a Condensing Agent. X.1 Rearrangements

J. Simons, S. Archer, D. I. Randall, 1940 .

Hybromet: a ligand for purifying opioid receptors.

E. J. Simon, R. Zukin, T. Gioannini, 1985, Journal of medicinal chemistry.

Preventing morphine antinociceptive tolerance by irreversible mu opioid antagonists before the onset of their antagonism

Q. Jiang, A. Sebastian, S. Archer, 1994, Regulatory Peptides.

Affinity labeling of mu opioid receptors by sulfhydryl alkylating derivatives of morphine and morphinone.

S. Archer, A. Seyed-Mozaffari, J. Bidlack, 1990, Molecular pharmacology.

Purification and characterization of the mu opiate receptor from rat brain using affinity chromatography.

R. Zukin, R. Maneckjee, J. Michael, 1985, Proceedings of the National Academy of Sciences of the United States of America.

Purification of the opiate receptor from rat brain.

J. Bidlack, L. Abood, S. Archer, 1981, Proceedings of the National Academy of Sciences of the United States of America.

Identification of opioid receptors in the immune system using a novel combination of selective opioid ligands and indirect phycoerythrin immunofluorescence.

J. Bidlack, D. M. Lawrence, S. Archer, 1995, Advances in experimental medicine and biology.

Synthesis and characterization of 7-nitrobenzo-2-oxa-1,3-diazole (NBD)-labeled fluorescent opioids.

P. Emmerson, F. Medzihradsky, S. Archer, 1992, Biochemical pharmacology.

Opioid ligands related to tifluadom

E. J. Simon, T. Gioannini, S. Archer, 1989 .

X-Ray Contrast Media for Cardiovascular Angiography

S. Archer, J. O. Hoppe, 1960, Angiology.

Affinity labeling of the mu opioid receptor in bovine striatal membranes with [3H]-14 beta-(bromoacetamido)-7,8-dihydromorphine.

R. Subbramanian, S. Archer, A. Seyed-Mozaffari, 1993, Biochemistry.

Observations on a series of aryl triiodo alkanoic acid derivatives with particular reference to a new cholecystographic medium, telepaque.

S. Archer, J. O. Hoppe, 1953, The American journal of roentgenology, radium therapy, and nuclear medicine.

Mode of action of the schistosomicide hycanthone: site of DNA alkylation.

W. El-hamouly, D. Cioli, S. Archer, 1990, Molecular and biochemical parasitology (Print).

Preparation and antitumor activity of an N-methylcarbamate derivative of amsacrine

J. Ruckdeschel, W. El-hamouly, S. Archer, 1993 .

Hycanthone resistance in schistosomes correlates with the lack of an enzymatic activity which produces the covalent binding of hycanthone to parasite macromolecules.

D. Cioli, S. Archer, L. Pica-Mattoccia, 1992, Molecular and biochemical parasitology.

Cyclazocine revisited

S. D. Glick, J. Bidlack, S. Archer, 2006, Neurochemical Research.

L(+)-2-Tropinone1

M. Bell, S. Archer, 1960 .

L(+)2-TROPINONE

M. Bell, S. Archer, 1958 .

Historical perspective on the chemistry and development of naltrexone.

S. Archer, 1981, NIDA research monograph.

Metabolism of 2,2-dichloro-N-[b-hydroxy-alpha-(hydroxymethyl)-p-(methylsulfinyl)-phenethyl] acetamide.

D. Rosi, S. Archer, A. Braemer, 1967, Life Science.

U50,488, a κ opioid receptor agonist, attenuates cocaine-induced increases in extracellular dopamine in the nucleus accumbens of rats

S. D. Glick, I. M. Maisonneuve, S. Archer, 1994, Neuroscience Letters.

Reaction of 4-methylpyrano[3,4-b]indol-3-one with (dimethyltriazen-1-yl)pyridinecarboxylic acids, precursors of 3,4-pyridynes

S. Modi, S. Archer, 1989 .

An efficient synthesis of C-11 substituted 6H-pyrido[4,3-b]carbazoles

J. J. Carey, S. Modi, S. Archer, 1991 .

Reaction of 4-Methylpyrano(3,4-b)indol-3-one with (Dimethyltriazen-1-yl)pyridinecarboxylic Acids, Precursors of 3,4-Pyridynes.

S. Modi, S. Archer, 1990 .

Synthesis of 6h-pyrido[4,3-b]carbazoles

S. Modi, S. Archer, A. Zayed, 1990 .

Hydrogen Fluoride as a Condensing Agent. XI. The Reaction of Alcohols and Ethers with Benzene1

J. Simons, S. Archer, 1940 .

An Efficient Synthesis of C-11 Substituted 6H-Pyrido(4,3-b)carbazoles.

J. J. Carey, S. Modi, S. Archer, 1991 .

Synthesis and biological properties of some 6H-pyrido[4,3-b]carbazoles.

B. Ross, D. Cioli, S. Archer, 1987, Journal of medicinal chemistry.

Indole‐2‐Acetic Acid Methyl Esters: Methyl 5‐Methoxyindole‐2‐Acetate

S. Modi, S. Archer, R. C. Oglesby, 2003 .

Synthesis of 6H-Pyrido(4,3-b)carbazoles.

S. Modi, S. Archer, A. Zayed, 1991 .

4-[(Aminoalkyl)amino]-1,2-dimethoxynaphthalenes as antimalarial agents.

S. Archer, P. Osei-Gyimah, S. Silbering, 1980, Journal of Medicinal Chemistry.

4-((AMINOALKYL)AMINO)-1,2-DIMETHOXYNAPHTHALENES AS ANTIMALARIAL AGENTS

S. Archer, P. Osei-Gyimah, S. Silbering, 1980 .

Inner Complexes of Uranium Containing 1,3-Dicarbonyl Chelating Groups

H. Brown, H. Schlesinger, S. Archer, 1953 .

1-(Indolylalkyl)-4-Arylpiperazines: A New Class of Tranquilizers

L. Harris, M. Bell, R. Kullnig, 1962 .

N-cyclobutylmethyl analog of normorphinone, N-CBM-TAMO: a short-term opioid agonist and long-term Mu-selective irreversible opioid antagonist.

J. Bidlack, S. Archer, A. Seyed-Mozaffari, 1996, The Journal of pharmacology and experimental therapeutics.

Effects of the structurally novel opioid 14 alpha, 14' beta-[dithiobis [(2-oxo-2,1-ethanediyl)imino]]bis(7,8-dihydromorphinone) on schedule-controlled behavior and thermal nociception in rhesus monkeys.

N. Mello, S. Negus, J. Bidlack, 1996, The Journal of pharmacology and experimental therapeutics.

N-Methyl and N-cyclopropylmethyl-14α,14′β-[dithiobis[(2-oxo-2,1-ethanediyl)imino]]bis(7,8-dihydro-5β-methyl-morphinone) MET-TAMO and N-CPM-MET-TAMO: Synthesis and opioid binding properties

J. Bidlack, A. Sebastian, S. Archer, 1995 .

14 alpha,14' beta-[Dithiobis[(2-oxo-2,1-ethanediyl)imino]]bis (7,8-dihydromorphinone) and 14 alpha,14' beta-[dithiobis[(2-oxo-2,1- ethanediyl)imino]]bis[7,8-dihydro-N-(cyclopropylmethyl)normorphinone]: chemistry and opioid binding properties.

J. Bidlack, Q. Jiang, S. Archer, 1994, Journal of medicinal chemistry.

5 beta-Methyl-14 beta-(p-nitrocinnamoylamino)-7,8-dihydromorphinone and its corresponding N-cyclopropylmethyl analog, N-cyclopropylmethylnor-5 beta-methyl-14 beta-(p-nitrocinnamoylamino)- 7,8-dihydromorphinone: mu-selective irreversible opioid antagonists.

J. Bidlack, Q. Jiang, A. Sebastian, 1994, The Journal of pharmacology and experimental therapeutics.

14 beta-[(p-nitrocinnamoyl)amino]morphinones, 14 beta-[(p-nitrocinnamoyl)amino]-7,8-dihydromorphinones, and their codeinone analogues: synthesis and receptor activity.

S. D. Glick, J. Bidlack, D. Deecher, 1993, Journal of medicinal chemistry.

Pharmacological study of 14 beta-(thioglycolamido)-7,8-dihydro-N(cyclopropylmethyl)-normor phinone (N-CPM-TAMO).

J. Bidlack, Q. Jiang, S. Archer, 1993, The Journal of pharmacology and experimental therapeutics.

Antinociceptive properties of two alkylating derivatives of morphinone: 14 beta-(thioglycolamido)-7,8-dihydromorphinone (TAMO) and 14 beta-(bromoacetamido)-7,8-dihydromorphinone (H2BAMO).

J. Bidlack, Q. Jiang, S. Archer, 1992, The Journal of pharmacology and experimental therapeutics.

14 beta-(2-bromoacetamido)morphine and 14 beta-(2-bromoacetamido)morphinone.

J. Bidlack, L. Abood, S. Archer, 1983, Journal of medicinal chemistry.

The resolution of ethyl 1,1-diphenyl-3-dimethyl-aminobutyl sulfone.

S. Archer, B. Tullar, W. Wetterau, 1948, Journal of the American Chemical Society.

Resistance of schistosomes to hycanthone and oxamniquine.

D. Cioli, S. Archer, L. Pica-Mattoccia, 1989, Memorias do Instituto Oswaldo Cruz.

Studies on some derivatives of oxamniquine.

W. El-hamouly, H. Schwartz, D. Cioli, 1988, Journal of medicinal chemistry.

The Cleavage of 3-Tropanyl Chloride with Potassium Cyanide1

S. Archer, T. R. Lewis, B. L. Zenitz, 1957 .

Synthesis, rodent biodistribution, dosimetry, metabolism, and monkey images of carbon-11-labeled (+)-2 alpha-tropanyl benzilate: a central muscarinic receptor imaging agent.

R. Koeppe, N. Petry, D. Jewett, 1992, Journal of nuclear medicine : official publication, Society of Nuclear Medicine.

Emetic activity of N-substituted norapomorphines.

E. Atkinson, S. Archer, F. J. Bullock, 1975, Journal of medicinal chemistry.

Synthesis and analgesic activity of some 14 beta-substituted analogues of morphine.

S. Archer, P. Osei-Gyimah, 1980, Journal of medicinal chemistry.

Synthesis of 5-methyl-6h-pyrido[4,3-b]carbazole-11-methanol

J. J. Carey, S. Modi, S. Archer, 1990 .

Synthesis of 5‐Methyl‐6H‐pyrido(4,3‐b)carbazole‐11‐methanol.

J. J. Carey, S. Modi, S. Archer, 1991 .

REACTION OF THEBAINE WITH DINITROGEN TETROXIDE

S. Archer, P. Osei-Gyimah, 1979 .

THE SYNTHESIS AND AGONIST ACTIVITY OF SOME 14β-SUBSTITUTED MORPHINE AND CODEINE DERIVATIVES

S. Archer, P. Osei-Gyimah, 1980 .

SYNTHESIS AND ANALGESIC ACTIVITY OF SOME 14β-SUBSTITUTED ANALOGS OF MORPHINE

S. Archer, P. Osei-Gyimah, 1980 .

Synthesis and analgesic activity of some 14 beta-substituted analogues of morphine.

S. Archer, P. Osei-Gyimah, 1980, Journal of Medicinal Chemistry.

The Preparation of Dimethyl-γ-cyclopentylidene-γ-phenylpropylamine and Related Compounds

S. Archer, B. Tullar, F. C. Nachod, 1949 .

The Cleavage of 3-Dimethylamino-1,1-diphenylbutyl Ethyl Sulfone

S. Archer, M. Auerbach, 1951 .

The preparation and properties of some benzohydryl sulfones.

S. Archer, C. Suter, M. Klenk, 1948, Journal of the American Chemical Society.

STRUCTURE-ACTIVITY RELATIONSHIPS OF 1-((3-INDOLYL)ALKYL)-4- ARYLPIPERAZINES. A NEW SERIES OF TRANQUILIZERS.

S. Archer, D. Wylie, 1962, Journal of medicinal and pharmaceutical chemistry.

A Synthesis of dl-Ornithine Hydrochloride

S. Archer, N. Albertson, 1945 .

CHEMICAL ASPECTS OF RADIOPAQUE AGENTS

S. Archer, 1959, Annals of the New York Academy of Sciences.