Christelle Marminon

发表

Phenolic indeno[1,2-b]indoles as ABCG2-selective potent and non-toxic inhibitors stimulating basal ATPase activity

Mathieu Marchivie, Joachim Jose, Jean Guillon, 2015, Drug design, development and therapy.

Uncompetitive nanomolar dimeric indenoindole inhibitors of the human breast cancer resistance pump ABCG2.

A. di Pietro, B. Sarkadi, P. Falson, 2020, European journal of medicinal chemistry.

QSAR Model of Indeno[1,2-b]indole Derivatives and Identification of N-isopentyl-2-methyl-4,9-dioxo-4,9-Dihydronaphtho[2,3-b]furan-3-carboxamide as a Potent CK2 Inhibitor

S. Haidar, J. Jose, M. Le Borgne, 2019, Molecules.

Self-Assembled Supramolecular Nanoparticles Improve the Cytotoxic Efficacy of CK2 Inhibitor THN7

F. Perret, J. Jose, M. Le Borgne, 2018, Pharmaceuticals.

Development of Pharmacophore Model for Indeno[1,2-b]indoles as Human Protein Kinase CK2 Inhibitors and Database Mining

A. Poso, T. Laitinen, S. Haidar, 2017, Pharmaceuticals.

Inhibition of Shiga toxin-converting bacteriophage development by novel antioxidant compounds

Karolina Pierzynowska, G. Węgrzyn, L. Saso, 2018, Journal of enzyme inhibition and medicinal chemistry.

Microwave-accelerated multicomponent synthesis and X-ray characterization of novel benzothiadiazinone dioxide derivatives, analogues of Monastrol

S. Bouacida, M. Le Borgne, Z. Bouaziz, 2021, Research on Chemical Intermediates.

Semi-synthesis, topoisomerase I and kinases inhibitory properties, and antiproliferative activities of new rebeccamycin derivatives.

C. Bailly, P. Renard, B. Pfeiffer, 2003, Bioorganic & medicinal chemistry.

Syntheses and antiproliferative activities of rebeccamycin analogues bearing two 7-azaindole moieties.

P. Renard, B. Pfeiffer, M. Prudhomme, 2003, Bioorganic & medicinal chemistry.

Broad-Spectrum Anticancer Activity and Pharmacokinetic Properties of a Prenyloxy-Substituted Indeno[1,2-b]indole Derivative, Discovered as CK2 Inhibitor

J. Jose, M. Le Borgne, Ehab El-Awaad, 2021, Pharmaceuticals.

Synthesis, Spectroscopic Characterization, and In Vitro Antibacterial Evaluation of Novel Functionalized Sulfamidocarbonyloxyphosphonates

M. Le Borgne, Z. Bouaziz, J. Lebreton, 2018, Molecules.

Rebeccamycin Derivatives as Dual DNA-Damaging Agents and Potent Checkpoint Kinase 1 Inhibitors

L. Meijer, P. Peixoto, B. Pfeiffer, 2008, Molecular Pharmacology.

Novel α-sulfamidophosphonate analogues of fotemustine: efficient synthesis using ultrasound under solvent-free conditions

T. Ben Hadda, M. Berredjem, Christelle Marminon, 2020, Monatshefte für Chemie - Chemical Monthly.

Diels-Alder reactions between acrolein N,N-dimethylhydrazone and N-benzylated benzotriazole-, indazole- or indole-4,7-diones

R. Terreux, B. Fenet, Christelle Marminon, 2009 .

DNA targeting of two new antitumour rebeccamycin derivatives.

C. Bailly, P. Colson, C. Houssier, 2002, European journal of medicinal chemistry.

Candidate Molecule Selection Based on In Silico Predicted ADMET Properties of 12 Indenoindole Derivatives

R. Terreux, A. Pietro, M. Gustin, 2016 .

Synthesis of N-benzylated indole-, indazole- and benzotriazole-4,7-diones

R. Barret, Christelle Marminon, P. Nebois, 2007 .

Ninhydrins inhibit carbonic anhydrases directly binding to the metal ion.

C. Supuran, J. Jose, Silvia Bua, 2020, European journal of medicinal chemistry.

Microwave-assisted oxidation of indan-1-ones into ninhydrins

J. Jose, Z. Bouaziz, Christelle Marminon, 2015 .

Syntheses and antiproliferative activities of 7-azarebeccamycin analogues bearing one 7-azaindole moiety.

C. Bailly, P. Renard, B. Pfeiffer, 2003, Journal of medicinal chemistry.

Novel N-acylsulfamoyl-oxazolidin-2ones: Synthesis, antitumor activity, X-ray crystallographic study, molecular docking and POM analyses

T. Hadda, S. Bouacida, M. Berredjem, 2022, Journal of Molecular Structure.

Synthesis, in silico study (DFT, ADMET) and crystal structure of novel sulfamoyloxy-oxazolidinones: Interaction with SARS-CoV-2

K. Bacharı, S. Bouacida, Z. Bouaziz, 2022, Journal of Molecular Structure.

Converting potent indeno[1,2-b]indole inhibitors of protein kinase CK2 into selective inhibitors of the breast cancer resistance protein ABCG2.

Joachim Jose, Jean Guillon, A. di Pietro, 2015, Journal of medicinal chemistry.

Synthesis and modulation properties of imidazo[4,5-b]pyridin-7-one and indazole-4,7-dione derivatives towards the Cryptosporidium parvum CpABC3 transporter.

S. Radix, N. Walchshofer, P. Lawton, 2010, European journal of medicinal chemistry.

Unexpected Binding Mode of a Potent Indeno[1,2-b]indole-Type Inhibitor of Protein Kinase CK2 Revealed by Complex Structures with the Catalytic Subunit CK2α and Its Paralog CK2α′

J. Jose, K. Niefind, D. Lindenblatt, 2017, Pharmaceuticals.

Preparation and characterization of CK2 inhibitor-loaded cyclodextrin nanoparticles for drug delivery.

F. Perret, J. Jose, H. Parrot-Lopez, 2013, International journal of pharmaceutics.

Diacritic Binding of an Indenoindole Inhibitor by CK2α Paralogs Explored by a Reliable Path to Atomic Resolution CK2α′ Structures

J. Jose, K. Niefind, D. Lindenblatt, 2019, ACS omega.

Inhibitors of ABCG2-mediated multidrug resistance: Lead generation through computer-aided drug design.

L. Goracci, V. Chaptal, P. Falson, 2023, European journal of medicinal chemistry.

Mechanistic basis of breast cancer resistance protein inhibition by new indeno[1,2-b]indoles

S. Ambudkar, J. Jose, F. Rego, 2021, Scientific Reports.

Dimers from dechlorinated rebeccamycin: synthesis, interaction with DNA, and antiproliferative activities.

C. Bailly, P. Renard, B. Pfeiffer, 2002, European journal of medicinal chemistry.

Syntheses and antiproliferative activities of new rebeccamycin derivatives with the sugar unit linked to both indole nitrogens.

P. Renard, B. Pfeiffer, M. Prudhomme, 2002, Journal of medicinal chemistry.

Unexpected Binding Mode of a Potent Indeno[1,2-b]indole-Type Inhibitor of Protein Kinase CK2 Revealed by Complex Structures with the Catalytic Subunit CK2α and Its Paralog CK2α′

J. Jose, K. Niefind, D. Lindenblatt, 2017, Pharmaceuticals.