M. Kahn

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A merger of rational drug design and combinatorial chemistry: development and application of peptide secondary structure mimetics.

M Kahn, H. Kim, H O Kim, 2000, Combinatorial chemistry & high throughput screening.

A Merger of Rational Drug Design and Combinatorial Chemistry: Development and Application of Peptide Secondary Structure Mimetics

H. Kim, M. Kahn, 2001 .

Δ9-Tetrahydrocannabinolic acid A, the precursor to Δ9-tetrahydrocannabinol (THC).

B. Foxman, M. Kahn, J. Skell, 2021, Acta crystallographica. Section C, Structural chemistry.

The design and synthesis of a nonpeptide mimic of erabutoxin

M. Kahn, P. Zieske, B. Chen, 1987 .

The design and synthesis of a nonpeptide mimic of an immunosuppressing peptide

B. Devens, M. Kahn, 1986 .

Design, synthesis and conformational analysis of γ-turn peptide mimetics of bradykinin

Michael E. Johnson, H. Nakanishi, M. Kahn, 1992 .

Design and synthesis of nonpeptide mimetics of jaspamide.

H. Nakanishi, M. Johnson, J. Lee, 2009, International journal of peptide and protein research.

The incorporation of β-turn prosthetic units into merrifield solid phase peptide synthesis

S. Bertenshaw, M. Kahn, 1989 .

Methodology for the synthesis of mimetics of peptide β-turns

M. Kahn, Barbara B. Chen, 1987 .

An anomalous mannich reaction of a trimethylsilyl enol ether

S. Danishefsky, M. Kahn, M. Silvestri, 1982 .

Nonpeptide mimetics of jaspamide

M. Kahn, 1988 .

29 – DESIGN OF PEPTIDOMIMETICS

Michael Kahn, Hiroshi Nakanishi, H. Nakanishi, 2003 .

Concepts and progress in the development of peptide mimetics.

M Kahn, M. Hatada, M. Bös, 1993, Journal of medicinal chemistry.

Control of ring junction stereochemistry via radical cyclization

G. Stork, M. Kahn, 1985 .

High-throughput synthesis and optimization of thrombin inhibitors via urazole alpha-addition and Michael addition.

J. Urban, M. Nguyen, P. D. Boatman, 2003, Bioorganic & Medicinal Chemistry Letters.

Stereospecific total syntheses of dl-coriolin and dl-coriolin B

R. Zamboni, S. Danishefsky, M. Kahn, 1981 .

Control of ring junction stereochemistry via radical cyclization

G. Stork, M. Kahn, 1985 .

Design and synthesis of a protein. beta. -turn mimetic

V. Madison, M. Voss, C. Cook, 1990 .

A convenient preparation of 1-phenylsulfonyl-3-iodomethylindole

M. Kahn, Michito Sato, 1990 .

Phosphine mediated synthesis of 2-methylidene-3-amino esters and ketones

S. Bertenshaw, M. Kahn, 1989 .

Secondary structure peptide mimetics: design, synthesis, and evaluation of beta-strand mimetic thrombin inhibitors.

J. P. Shea, M. Eguchi, H. Nakanishi, 1999, Journal of medicinal chemistry.

β-SHEET MIMETICS AND USE THEREOF AS INHIBITORS OF BIOLOGICALLY ACTIVE PEPTIDES OR PROTEINS

M. Eguchi, P. D. Boatman, H. Kim, 1997 .

Enantiospecific routes to 3,4 disubstituted azetidinones

M. Kahn, K. Fujita, 1991 .

A highly stereoselective osmium tetroxide-catalyzed hydroxylation of γ-hydroxy α,β-usaturated esters

G. Stork, M. Kahn, 1983 .

Anionic oxy-cope reaction of a divinyl cyclobutanol, pleuromutilin model study

M. Kahn, 1980 .

Total synthesis of dl-coriolin

R. Zamboni, S. Danishefsky, M. Kahn, 1980 .

Nonpeptide mimetics of .beta.-turns: a facile oxidative intramolecular cycloaddition of an azodicarbonyl system

M. Kahn, Barbara B. Chen, K. Fujita, 1988 .

Design and synthesis of hypertrehalosemic hormoe mimetics

Michael E. Johnson, T. Hayes, M. Kahn, 1993 .

Regiospecific Michael reactions to an enedione

S. Danishefsky, M. Kahn, 1981 .

Regiospecificity in the Diels-Alder reactions of an enedione

S. Danishefsky, M. Kahn, 1981 .

Loops and Secondary Structure Mimetics: Development and Applications in Basic Science and Rational Drug Design

Michael Kahn, H. Uri Saragovi, Mark I. Greene, 1992, Bio/Technology.

Enlistment of combinatorial techniques in drug development.

M S Lee, H Nakanishi, M Kahn, 1999, Current opinion in drug discovery & development.

Peptidomimetics of the immunoglobulin supergene family--a review.

H. Nakanishi, S. Ramurthy, M. Kahn, 1993, Gene.

Design, synthesis, and application of peptide secondary structure mimetics.

M. Eguchi, M. Kahn, 2002, Mini reviews in medicinal chemistry.

A HIGHLY STEREOSELECTIVE OSMIUM TETROXIDE-CATALYZED HYDROXYLATION OF Γ-HYDROXY α,β-UNSATURATED ESTERS

G. Stork, M. Kahn, 1984 .

The three‐dimensional solution structure of a constrained peptidomimetic in water and in chloroform observation of solvent induced hydrophobic cluster

H. Nakanishi, Min S. Lee, M. Kahn, 1995, FEBS letters.

Design and synthesis of a mimetic from an antibody complementarity-determining region.

M Kahn, H. Nakanishi, M. Greene, 1991, Science.

Sculpted immunogens; B-cell epitope optimization using constrained secondary structure libraries.

J. Urban, M. Klein, C. Sia, 1996, Bioorganic & medicinal chemistry.

Peptide mimetics of the thrombin-bound structure of fibrinopeptide A.

M Kahn, A. Tulinsky, S. Bertenshaw, 1992, Proceedings of the National Academy of Sciences of the United States of America.

Peptidomimetic antagonists designed to inhibit the binding of CD4 to HIV GP120.

M S Lee, M Kahn, H. Nakanishi, 1994, Bioorganic & medicinal chemistry.

The design and synthesis of mimetics of peptide β‐turns

Michael E. Johnson, M. Kahn, Barbara B. Chen, 1988 .

Pharmaceutical applications of peptidomimetics

J. Urban, M. Klein, C. Sia, 1996, Letters in Peptide Science.

Nonpeptide β-turn mimetics of enkephalin

Michael E. Johnson, H. Nakanishi, S. M. Tuladhar, 1993 .

Highly efficient and versatile synthesis of libraries of constrained beta-strand mimetics.

J. Urban, M. Nguyen, C. Lum, 1998, Bioorganic & medicinal chemistry letters.