Eric Stefan

发表

7-(4H-1,2,4-Triazol-3-yl)benzo[c][2,6]naphthyridines: a novel class of Pim kinase inhibitors with potent cell antiproliferative activity.

Adam Siddiqui-Jain, Diwata Macalino, Nicole Streiner, 2011, Bioorganic & medicinal chemistry letters.

Discovering the anticancer potential of non-oncology drugs by systematic viability profiling

Joshua A. Bittker, James M. McFarland, Vickie M. Wang, 2020, Nature Cancer.

Non-oncology drugs are a source of previously unappreciated anti-cancer activity

Joshua A. Bittker, James M. McFarland, Vickie M. Wang, 2019, bioRxiv.

Stereoselective synthesis of the C9-C19 fragment of lyngbyaloside B and C via ether transfer.

Richard E. Taylor, Eric Stefan, 2012, Organic letters.

Discovery of small-molecule positive allosteric modulators of Parkin E3 ligase

L. Silvian, A. Weihofen, W. Hirst, 2021, iScience.

Discovery and SAR of 5-(3-chlorophenylamino)benzo[c][2,6]naphthyridine-8-carboxylic acid (CX-4945), the first clinical stage inhibitor of protein kinase CK2 for the treatment of cancer.

Adam Siddiqui-Jain, J. Bliesath, M. Omori, 2011, Journal of medicinal chemistry.

Pre-clinical characterization of CX-4945, a potent and selective small molecule inhibitor of CK2 for the treatment of cancer

Adam Siddiqui-Jain, J. Bliesath, M. Omori, 2011, Molecular and Cellular Biochemistry.

Novel potent pyrimido[4,5-c]quinoline inhibitors of protein kinase CK2: SAR and preliminary assessment of their analgesic and anti-viral properties.

Adam Siddiqui-Jain, Nicole Streiner, Caroline B. Ho, 2011, Bioorganic & medicinal chemistry letters.

1,5-Hydride transfer protocol for the synthesis of β-branched polyketide structural units

Richard E. Taylor, Eric Stefan, 2015 .

Total Synthesis and Structural Reassignment of Lyngbyaloside C Highlighted by Intermolecular Ketene Esterification.

Richard E. Taylor, Chia‐Fu Chang, Eric Stefan, 2015, Chemistry.

Ether Transfer Methodology: Application to the Synthesis of Polyketide Natural Products

Richard E. Taylor, Eric Stefan, 2013 .

Concise enantioselective synthesis of diospongins A and B.

A. Nalin, Richard E. Taylor, Eric Stefan, 2013, Tetrahedron.

Stabilization of the Max Homodimer with a Small Molecule Attenuates Myc-Driven Transcription.

Vincent L. Butty, Charles Y. Lin, P. Clemons, 2019, Cell chemical biology.

Synthesis and SAR of inhibitors of protein kinase CK2: novel tricyclic quinoline analogs.

Adam Siddiqui-Jain, Diwata Macalino, S. O'Brien, 2012, Bioorganic & medicinal chemistry letters.