L. Bischoff

发表

Kinetic modeling of carbon dioxide valorization with epoxides

A. Ledoux, L. Estel, V. Levacher, 2016 .

New family of peptidomimetics based on the imidazole motif.

Corinne Fruit, S. Petit, L. Bischoff, 2010, Organic letters.

Inhibition of vasopressinergic neurons by central injection of a specific aminopeptidase A inhibitor

P. Corvol, C. Llorens-Cortes, M. Fournié-Zaluski, 1998, Neuroreport.

One-pot synthesis of 2,3-dihydro-pyrrolopyridinones using in situ generated formimines.

Corinne Fruit, F. Marsais, L. Bischoff, 2006, Organic letters.

Binding properties of a highly potent and selective iodinated aminopeptidase N inhibitor appropriate for radioautography

M. Fournié-Zaluski, B. Roques, N. Luciani, 2000, FEBS Letters.

Design of silicon-based misonidazole analogues and (18)F-radiolabelling.

Corinne Fruit, P. Vera, F. Marsais, 2009, Nuclear medicine and biology.

Enantioselective hydrogenation reactions with a full set of preformed and prepared in situ chiral diphosphine-ruthenium (II) catalysts.

C. Pinel, V. Ratovelomanana-Vidal, J. Genêt, 1994 .

A Meldrum's Acid Based Multicomponent Synthesis of N‐Fmoc‐isoxazolidin‐5‐ones: Entry to N‐Fmoc‐β‐amino Acids

V. Levacher, L. Bischoff, Emmanuel Deau, 2017 .

Straightforward and Diastereoselective Synthesis of Tetrafunctionalized Thiol Synthons for the Design of Metallopeptidase Inhibitors

B. Roques, M. Fournié-Zaluski, C. David, 2000 .

Deprotonation of benzoxazole and oxazole using lithium magnesates.

F. Mongin, C. Hoarau, F. Marsais, 2005, The Journal of organic chemistry.

A very short route to enantiomerically pure coumarin-bearing fluorescent amino acids.

C. Garbay, L. Bischoff, Marie-Priscille Brun, 2004, Angewandte Chemie.

Preparation and Reactivity of Allyl N-[(Arylsulfonyl)oxy]carbamates, New Reagents for Electrophilic Transfer of an NHAlloc Group

C. Greck, J. Genêt, F. Ferreira, 1995 .

Towards a biomimetic synthesis of barrenazine A

F. Buron, F. Marsais, A. Turck, 2007 .

Ortho-Directed Palladium-Catalyzed Direct C–H Functionalization of 3-Picolinyl- and 3-(2-Cyanoethyl)pyrimidin-4(3H)-ones with Aryl Halides

C. Hoarau, V. Levacher, L. Bischoff, 2020, Synlett.

Ligand-free Pd-catalyzed and copper-assisted C-H arylation of quinazolin-4-ones with aryl iodides under microwave heating.

Corinne Fruit, Sylvain Laclef, T. Besson, 2015, Organic letters.

Aminomethylation of lithiated nicotinamide: access to new pyridolactams

Corinne Fruit, F. Marsais, Rabah Azzouz, 2008 .

Anionic, in situ generation of formaldehyde: a very useful and versatile tool in synthesis.

Corinne Fruit, F. Marsais, L. Bischoff, 2007, Organic letters.

Bicyclic 5-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Two Extra Heteroatoms 2:0

L. Bischoff, 2008 .

Orthopalladation of GFP-Like Fluorophores Through C-H Bond Activation: Scope and Photophysical Properties

C. Cativiela, A. Jiménez, E. Urriolabeitia, 2018, European Journal of Organic Chemistry.

Organometallic Fluorophores of d8 Metals (Pd, Pt, Au)

E. Urriolabeitia, C. Hoarau, L. Bischoff, 2018 .

Organocatalytic enantioselective synthesis of β-amino sulfonic acid derivatives.

V. Levacher, L. Bischoff, Emmanuel Deau, 2021, Chemical communications.

Synthesis of (3S, 4S)-4-hydroxy-2, 3, 4, 5-tetrahydropyridazine-3-carboxylic acid, component of luzopeptin A.

C. Greck, J. Genêt, L. Bischoff, 1995 .

A convenient synthesis of N-boc protected primary amines via the reaction of organoboranes with Li or K t-butyl-N-tosyloxycarbamate

J. Hájíček, C. Greck, J. Genêt, 1992 .

An efficient approach to new dihydroxyquinolizidines

Corinne Fruit, T. Tite, F. Marsais, 2010 .

Electrophilic Amination of Carbanions with Metalated t-Butyl N- Tosyloxycarbamate.

J. Hájíček, C. Greck, J. Genêt, 1994 .

Enantioselective Hydrogenation Reactions with a Full Set of Preformed and Prepared in situ Chiral Diphosphine‐Ruthenium(II) Catalysts.

C. Pinel, V. Ratovelomanana-Vidal, J. Genêt, 1994 .

A concise synthesis of lentiginosine derivatives using a pyridinium formation via the Mitsunobu reaction.

Corinne Fruit, F. Marsais, Rabah Azzouz, 2008, The Journal of organic chemistry.

Preparation and Reactivity of Allyl N-((Arylsulfonyl)oxy)carbamates, New Reagents for Electrophilic Transfer of an NHAlloc Group.

C. Greck, J. Genêt, F. Ferreira, 1996 .

Asymmetric synthesis of anti N-Boc-α-hydrazino-β-hydroxyesters from β-ketoesters by sequential catalytic hydrogenation and electrophilic amination

C. Pinel, C. Greck, J. Genêt, 1993 .

On the deprotonation of 3,5-dichloropyridine using lithium bases: in situ infrared spectroscopic studies

F. Mongin, F. Marsais, G. Quéguiner, 2005 .

SIDE-CHAIN-MODIFIED SULFONIC ANALOGUES OF ASPARTIC AND GLUTAMIC ACIDS : SYNTHESIS, PROTECTION, AND INCORPORATION INTO PEPTIDES

B. Roques, M. Fournié-Zaluski, C. David, 1999 .

2,4-Dinitrophenyl 4-Methoxybenzyl Disulfide: A New Efficient Reagent for the Electrophilic Sulfenylation of β-Amino Ester Enolates

B. Roques, H. Meudal, M. Fournié-Zaluski, 1997 .

Aminoacid-derived mercaptoimidazoles.

Corinne Fruit, F. Marsais, S. Petit, 2009, Organic & biomolecular chemistry.

First discrete autoradiographic distribution of aminopeptidase N in various structures of rat brain and spinal cord using the selective iodinated inhibitor [125I]RB 129

M. Fournié-Zaluski, B. Roques, S. Parsadaniantz, 2001, Neuroscience.

An approach to the manzamine alkaloids modelled on a biogenetic theory

D. Spring, T. Claridge, J. Baldwin, 1997 .

Pd(0)-Catalyzed Direct Inter- and Intramolecular C–H Functionalization of 4-Carboxyimidazoles

L. Meerpoel, P. Angibaud, C. Hoarau, 2020, Synlett.

Mild addition of carbon nucleophiles to pyridine and quinoline N-oxides under different activation conditions

Rabah Azzouz, L. Bischoff, Bertrand Lecointre, 2014 .

Synthesis and biological evaluation of a novel (99m)Tc labeled 2-nitroimidazole derivative as a potential agent for imaging tumor hypoxia.

P. Vera, C. Papamicaël, V. Le Joncour, 2013, Bioorganic & medicinal chemistry letters.

Mild Addition of Carbon Nucleophiles to Pyridine and Quinoline N-Oxides under Different Activation Conditions.

Rabah Azzouz, L. Bischoff, Bertrand Lecointre, 2014 .

An alternative route to the proline derivative (2S,5R)-5-ethoxycarbonylmethyl-pyrrolidine-2-carboxylic acid from protected glutamic acid

C. Garbay, L. Bischoff, Marie-Priscille Brun, 2003 .

Investigation of subsite preferences in aminopeptidase A (EC 3.4.11.7) led to the design of the first highly potent and selective inhibitors of this enzyme.

B. Roques, C. Llorens-Cortes, H. Meudal, 1999, Journal of medicinal chemistry.

Insights in the Synthesis of Imidazolones from Aldehydes, Isocyanides, or Oxazolines.

C. Hoarau, L. Bischoff, Christine Baudequin, 2022, The Journal of organic chemistry.

Pd-Catalyzed direct C-H functionalization of imidazolones with aryl- and alkenyl halides.

C. Hoarau, L. Bischoff, Christine Baudequin, 2015, Chemical Communications.

Formation of Imidazolones by Ring Closure of α-Isocyanoamides: Exploring New Reactivities

C. Hoarau, L. Bischoff, Christine Baudequin, 2020, Synlett.

Pd(0)-Catalyzed Direct C-H Functionalization of 2-H-4-Benzylidene Imidazolones: Friendly and Large-Scale Access to GFP and Kaede Protein Fluorophores.

C. Hoarau, C. Perrio, L. Bischoff, 2016, Chemistry.

Pd-Catalyzed Direct C—H Functionalization of Imidazolones with Aryl- and Alkenyl Halides.

C. Hoarau, L. Bischoff, Christine Baudequin, 2015 .

Isoform-selective HDAC1/6/8 inhibitors with an imidazo-ketopiperazine cap containing stereochemical diversity

A. Ganesan, W. Sippl, C. Romier, 2018, Philosophical Transactions of the Royal Society B: Biological Sciences.

Efficient Conversion of Epoxides into Carbonates with CO2 and a Single Organocatalyst: Laboratory and Kilogram-Scale Experiments

A. Ledoux, L. Estel, F. Marsais, 2019, Synlett.

Regioselective opening of N-Cbz glutamic and aspartic anhydrides with carbon nucleophiles

Corinne Fruit, Corinne Fruit, F. Marsais, 2006 .

Synthesis of new 18F-radiolabeled silicon-based nitroimidazole compounds.

V. Grégoire, P. Vera, A. Bol, 2013, Bioorganic & medicinal chemistry.

Mild, Efficient, One-Pot Synthesis of Imidazolones Promoted by N,O-Bistrimethylsilylacetamide (BSA)

L. Colombeau, C. Hoarau, L. Bischoff, 2016, Synlett.

On the racemisation of aspartic anhydride during its preparation

Corinne Fruit, F. Buron, F. Marsais, 2007 .

Synthesis of [3(R)‐amino‐2(S)‐sulfhydryl‐5‐sulfonate]‐pentanoyl‐(S)‐3‐[125I]‐iodotyrosyl‐(S)‐aspartic acid: a radiolabelled inhibitor of aminopeptidase A

B. Roques, L. Bischoff, Christelle David-Basei, 2001 .

An efficient protocol for the preparation of pyridinium and imidazolium salts based on the Mitsunobu reaction

Corinne Fruit, F. Marsais, S. Petit, 2008 .