D. Su

发表

Biaryl ethers as novel non-nucleoside reverse transcriptase inhibitors with improved potency against key mutant viruses.

Kenneth D Anderson, M. Lai, J. Vacca, 2009, Journal of medicinal chemistry.

Biaryl ethers as potent allosteric inhibitors of reverse transcriptase and its key mutant viruses: aryl substituted pyrazole as a surrogate for the pyrazolopyridine motif.

Kenneth D Anderson, M. Lai, J. Vacca, 2010, Bioorganic & medicinal chemistry letters.

Structure-Based Design of a Novel SMYD3 Inhibitor that Bridges the SAM-and MEKK2-Binding Pockets.

Tony W Dean, R. Annan, A. P. Graves, 2016, Structure.

A High-Throughput Dose-Response Cellular Thermal Shift Assay for Rapid Screening of Drug Target Engagement in Living Cells, Exemplified Using SMYD3 and IDO1

R. Annan, A. P. Graves, D. Mcnulty, 2018, SLAS discovery : advancing life sciences R & D.

Discovery of Isoxazole Amides as Potent and Selective SMYD3 Inhibitors.

J. Luengo, A. P. Graves, M. Pappalardi, 2019, ACS medicinal chemistry letters.

Pharmacological characterization and radioligand binding properties of a high-affinity, nonpeptide, bradykinin B1 receptor antagonist.

M. Bock, R. Freidinger, R. Chang, 2004, European journal of pharmacology.

Discovery of a potent, non-peptide bradykinin B1 receptor antagonist.

M. Bock, R. M. Dipardo, R. Freidinger, 2003, Journal of the American Chemical Society.

Total Synthesis of Epothilone A.

A. Balog, E. J. Sorensen, S. Danishefsky, 1996 .

Binding modes of dihydroquinoxalinones in a homology model of bradykinin receptor 1.

M. Bock, R. Freidinger, R. Chang, 2005, Biochemical and biophysical research communications.

Models for the Synthesis of Pluramycin Antibiotics. Rearrangement of Mono‐Protected Aminoglycal‐Substituted Cyclohexadienediols

K. A. Parker, D. Su, 2005 .

Total Syntheses of Epothilones A and B

A. Balog, E. J. Sorensen, S. Danishefsky, 1997 .

Silver(I) Oxide

D. Wright, A. Demchenko, Phillip M. Pelphrey, 2015 .

Synthesis of C-Aryl Furanosides by the “Reverse Polarity” Strategy

K. A. Parker, D. Su, 1996 .

The “Reverse Polarity” Approach to Ravidomycin. Aryl C‐Aminoglycosides from a Lithiated Aminoglycal

K. A. Parker, D. Su, 2005 .

Silver(II) Oxide

K. A. Parker, D. Su, 2001 .

REMOTE EFFECTS IN MACROLIDE FORMATION THROUGH RING-FORMING OLEFIN METATHESIS : AN APPLICATION TO THE SYNTHESIS OF FULLY ACTIVE EPOTHILONE CONGENERS

T. Chou, A. Balog, E. J. Sorensen, 1997 .

Structure–Activity Relationship of the Epothilones and the First In Vivo Comparison with Paclitaxel†

Susan Band Horwitz, T. Chou, A. Balog, 1997 .

Discovery of Orally Bioavailable Ligand Efficient Quinazolindiones as Potent and Selective Tankyrases Inhibitors.

R. Keenan, M. Cheung, A. Oliff, 2021, ACS medicinal chemistry letters.

Total Synthesis of (–)‐Epothilone B: An Extension of the Suzuki Coupling Method and Insights into Structure–Activity Relationships of the Epothilones

Susan Band Horwitz, Erik J. Sorensen, T. Chou, 1997 .

2-Aminobenzophenones as a novel class of bradykinin B1 receptor antagonists.

M. Bock, R. Freidinger, R. Chang, 2008, Journal of medicinal chemistry.

Potent bradykinin B1 receptor antagonists: 4-substituted phenyl cyclohexanes.

M. Bock, R. Freidinger, R. Chang, 2007, Bioorganic & medicinal chemistry letters.

Development of an efficient and selective radioligand for bradykinin B1 receptor occupancy studies.

M. Bock, R. Freidinger, R. Chang, 2004, Bioorganic & Medicinal Chemistry Letters.

Generation and Characterization of a Human Bradykinin Receptor B1 Transgenic Rat as a Pharmacodynamic Model

M. Bock, R. M. Dipardo, R. Chang, 2004, Journal of Pharmacology and Experimental Therapeutics.

Long-Range Inhibitor-Induced Conformational Regulation of Human IRE1α Endoribonuclease Activity

Leanna E. Shuster, K. Evans, S. Sweitzer, 2015, Molecular Pharmacology.

Synthesis of 2,5-disubstituted-3-cyanoindoles

Leanna E. Shuster, A. Kaura, K. Evans, 2012 .

Stereoselective syntheses and evaluation of compounds in the 8-desmethylepothilone a series: Some surprising observations regarding their chemical and biological properties

Susan Band Horwitz, Erik J. Sorensen, T. Chou, 1997 .

Substituted tetrahydroquinolines as potent allosteric inhibitors of reverse transcriptase and its key mutants.

Kenneth D Anderson, Youwei Yan, M. Lai, 2009, Bioorganic & Medicinal Chemistry Letters.

Identification of the critical residues of bradykinin receptor B1 for interaction with the kinins guided by site-directed mutagenesis and molecular modeling.

M. Bock, R. Chang, J. Hess, 2006, Biochemistry.

Farnesyl transferase inhibitors cause enhanced mitotic sensitivity to taxol and epothilones.

N. Rosen, M. Moasser, N. Kohl, 1998, Proceedings of the National Academy of Sciences of the United States of America.

Long-Range Inhibitor-Induced Conformational Regulation of Human IRE1α Endoribonuclease Activity

Leanna E. Shuster, K. Evans, C. Buser, 2015, Molecular Pharmacology.

Total Syntheses of Epothilones A and B.

A. Balog, E. J. Sorensen, S. Danishefsky, 1998 .