V. Whiterock

发表

Frequency of CYP1A2 polymorphism in beagle dogs.

T. Delmonte, Lester Hui, M. Sinz, 2007, Drug metabolism letters.

40 Hz Auditory Steady-State Response Is a Pharmacodynamic Biomarker for Cortical NMDA Receptors

M. Ahlijanian, Yulia Benitex, Yili Yang, 2016, Neuropsychopharmacology.

Development of 1H-Pyrazolo[3,4-b]pyridines as Metabotropic Glutamate Receptor 5 Positive Allosteric Modulators.

M. D. Hill, J. Macor, T. Molski, 2016, ACS medicinal chemistry letters.

Discovery of (R)-N-(3-(7-methyl-1H-indazol-5-yl)-1-(4-(1-methylpiperidin-4-yl)-1-oxopropan-2-yl)-4-(2-oxo-1,2-dihydroquinolin-3-yl)piperidine-1-carboxamide (BMS-742413): a potent human CGRP antagonist with superior safety profile for the treatment of migraine through intranasal delivery.

J. Macor, R. Schartman, G. Thalody, 2013, Bioorganic & medicinal chemistry letters.

Triazolopyridine ethers as potent, orally active mGlu2 positive allosteric modulators for treating schizophrenia.

M. Seager, J. Macor, A. Hendricson, 2017, Bioorganic & medicinal chemistry.

Synthesis, oral bioavailability determination, and in vitro evaluation of prodrugs of the antiviral agent 9-[2-(phosphonomethoxy)ethyl]adenine (PMEA).

J. C. Martin, J. Starrett, D. Tortolani, 1994, Journal of medicinal chemistry.

Discovery and Preclinical Evaluation of BMS-955829, a Potent Positive Allosteric Modulator of mGluR5.

J. Macor, Amy Easton, Anand Balakrishnan, 2016, ACS medicinal chemistry letters.

Disposition in animals of a new anti-HIV agent: 2',3'-didehydro-3'-deoxythymidine.

L. Klunk, J. Russell, V. Whiterock, 1990, Drug metabolism and disposition: the biological fate of chemicals.

Prodrugs of 2',3'-didehydro-3'-deoxythymidine (D4T): synthesis, antiviral activity, and rapid pharmacokinetic evaluation.

J. C. Martin, J. Starrett, D. Tortolani, 1994, Journal of pharmaceutical sciences.

Pharmacokinetics of A New Anti-HIV Ageht: 2′,3′-Dideoxy-2′,3′-Didehydrothymidine (d4T)

L. Klunk, J. Russell, V. Whiterock, 1989 .

Pharmacokinetics and antiviral activity of a novel isonucleoside, BMS-181165, against simian varicella virus infection in African green monkeys.

J. Clark, K. Soike, J. Russell, 1994, Antiviral research.

Oxazolidinone-based allosteric modulators of mGluR5: Defining molecular switches to create a pharmacological tool box.

J. Macor, Amy Easton, Anand Balakrishnan, 2016, Bioorganic & medicinal chemistry letters.

Synthesis, Oral Bioavailability Determination, and in vitro Evaluation of Prodrugs of the Antiviral Agent 9‐(2‐(Phosphonomethoxy)ethyl) adenine (PMEA).

J. Starrett, D. Tortolani, J. Russell, 1994 .

Determination of 9-[(2-phosphonylmethoxy)ethyl]adenine in rat urine by high-performance liquid chromatography with fluorescence detection.

L. Klunk, J. Russell, V. Whiterock, 1991, Journal of chromatography.

Structure activity relationship studies of 3-arylsulfonyl-pyrido[1,2-a]pyrimidin-4-imines as potent 5-HT₆ antagonists.

D. Langley, R. Westphal, P. Sivaprakasam, 2014, Bioorganic & medicinal chemistry.

Azepino-indazoles as calcitonin gene-related peptide (CGRP) receptor antagonists.

Kimberly A. Widmann, Ping Chen, J. Macor, 2020, Bioorganic & medicinal chemistry letters.

Design and Characterization of a Novel Fluorinated Magnetic Resonance Imaging Agent for Functional Analysis of Bile Acid Transporter Activity

J. Polli, J. Raufman, Su Xu, 2013, Pharmaceutical Research.

Phenacetin Pharmacokinetics in CYP1A2-Deficient Beagle Dogs

M. Sinz, Daniel G Morgan, K. Lentz, 2012, Drug Metabolism and Disposition.

Difluorocyclobutylacetylenes as positive allosteric modulators of mGluR5 with reduced bioactivation potential.

J. Macor, Amy Easton, Anand Balakrishnan, 2016, Bioorganic & medicinal chemistry letters.

Calcitonin Gene-Related Peptide (CGRP) Receptor Antagonists: Heterocyclic Modification of a Novel Azepinone Lead.

Kimberly A. Widmann, Ping Chen, J. Macor, 2021, Bioorganic & medicinal chemistry letters.