A. Wegert

发表

Quantitative Assessment of Drug Delivery to Tissues and Association with Phospholipidosis: A Case Study with Two Structurally Related Diamines in Development.

A. Kless, E. Hoppe, F. Held, 2017, Molecular pharmaceutics.

Preclinical Lead Optimization of a 1,2,4-Triazole Based Tankyrase Inhibitor

S. Krauss, Albert Galera‐Prat, M. Nazaré, 2020, Journal of medicinal chemistry.

Chlorodifluoromethyl-substituted monosaccharide derivatives--radical activation of the carbon-chlorine-bond.

M. Hein, R. Miethchen, N. Hoffmann, 2006, Carbohydrate research.

Development of a 1,2,4-Triazole-Based Lead Tankyrase Inhibitor: Part II

Albert Galera‐Prat, M. Nazaré, L. Lehtiö, 2021, Journal of medicinal chemistry.

Novel SAR for quinazoline inhibitors of EHMT1 and EHMT2.

M. Kubbutat, G. Müller, C. Schächtele, 2019, Bioorganic & medicinal chemistry letters.

Design and Synthesis of Enantiomerically Pure Decahydroquinoxalines as Potent and Selective κ-Opioid Receptor Agonists with Anti-Inflammatory Activity in Vivo.

R. Autar, S. Ständer, D. Metze, 2017, Journal of medicinal chemistry.

The Tankyrase Inhibitor OM-153 Demonstrates Antitumor Efficacy and a Therapeutic Window in Mouse Models

S. Krauss, I. Meerts, Albert Galera‐Prat, 2022, Cancer research communications.

Structure–Activity Relationship Studies on (R)‐PFI‐2 Analogues as Inhibitors of Histone Lysine Methyltransferase SETD7

F. Rutjes, J. Mecinović, Danny C. Lenstra, 2018, ChemMedChem.

Synthesis of 2,3- or 1,2-unsaturated derivatives of 2-deoxy-2-trifluoromethylhexopyranoses.

R. Miethchen, H. Reinke, A. Wegert, 2004, Carbohydrate Research.

Examining sterically demanding lysine analogs for histone lysine methyltransferase catalysis

Yali Wang, J. Mecinović, Hong Guo, 2020, Scientific Reports.

Methylation of geometrically constrained lysine analogues by histone lysine methyltransferases.

F. Rutjes, J. Mecinović, Paul B. White, 2020, Chemical communications.