Céline M'kadmi

发表

Cardioprotective Angiotensin-(1–7) Peptide Acts as a Natural-Biased Ligand at the Angiotensin II Type 1 Receptor

C. Boularan, A. Pathak, J. Senard, 2016, Hypertension.

The 1,2,4-triazole as a scaffold for the design of ghrelin receptor ligands: development of JMV 2959, a potent antagonist

A. Moulin, Jean Martinez, J. Fehrentz, 2012, Amino Acids.

Trisubstituted 1,2,4-triazoles as ligands for the ghrelin receptor: on the significance of the orientation and substitution at position 3.

A. Moulin, Jean Martinez, J. Fehrentz, 2008, Bioorganic & medicinal chemistry letters.

Agonism, Antagonism, and Inverse Agonism Bias at the Ghrelin Receptor Signaling*

Jean Martinez, J. Fehrentz, S. Denoyelle, 2015, The Journal of Biological Chemistry.

Design and Characterization of a Triazole-Based Growth Hormone Secretagogue Receptor Modulator Inhibiting the Glucoregulatory and Feeding Actions of Ghrelin.

S. Cantel, J. Fehrentz, S. Denoyelle, 2022, Biochemical pharmacology.

Gastrin releasing peptide receptor-directed radioligands based on a bombesin antagonist: synthesis, (111)in-labeling, and preclinical profile.

E. Krenning, M. de Jong, Jean Martinez, 2013, Journal of medicinal chemistry.

N-Terminal Liver-Expressed Antimicrobial Peptide 2 (LEAP2) Region Exhibits Inverse Agonist Activity toward the Ghrelin Receptor.

S. Cantel, J. Fehrentz, S. Denoyelle, 2018, Journal of medicinal chemistry.

New ligands of the ghrelin receptor based on the 1,2,4-triazole scaffold by introduction of a second chiral center.

A. Blayo, Jean Martinez, J. Fehrentz, 2016, Bioorganic & medicinal chemistry letters.

A new way to silicone-based peptide polymers.

C. Enjalbal, Jean Martínez, B. Nottelet, 2015, Angewandte Chemie.

GHSR-D2R heteromerization modulates dopamine signaling through an effect on G protein conformation

H. Hamm, G. Ferry, J. Boutin, 2018, Proceedings of the National Academy of Sciences.

Allosteric modulation of ghrelin receptor signaling by lipids

P. Bisch, S. Cantel, L. Catoire, 2021, Nature Communications.

α-tocopherol and α-tocopheryl phosphate interact with the cannabinoid system in the rodent hippocampus.

J. Guiramand, M. Vignes, C. Cohen‐Solal, 2011, Free radical biology & medicine.

Conditional and Reversible Activation of Class A and B G Protein-Coupled Receptors Using Tethered Pharmacology

D. Trauner, D. Hodson, J. Banères, 2018, ACS central science.

New trisubstituted 1,2,4-triazoles as ghrelin receptor antagonists.

A. Blayo, Jean Martinez, J. Fehrentz, 2015, Bioorganic & medicinal chemistry letters.

Homogeneous time-resolved fluorescence-based assay to screen for ligands targeting the growth hormone secretagogue receptor type 1a.

T. Roux, Emmanuel Bourrier, L. Lamarque, 2011, Analytical biochemistry.

Activation of the ghrelin receptor is described by a privileged collective motion: a model for constitutive and agonist-induced activation of a sub-class A G-protein coupled receptor (GPCR).

David Perahia, Nicolas Floquet, D. Pérahia, 2010, Journal of molecular biology.

The novel nonapeptide acein targets angiotensin converting enzyme in the brain and induces dopamine release

M. Kemel, P. Marin, S. Cantel, 2016, British journal of pharmacology.

Detergent-free Isolation of Functional G Protein-Coupled Receptors into Nanometric Lipid Particles.

O. Nosjean, G. Ferry, J. Boutin, 2016, Biochemistry.

The 1,2,4-triazole as a scaffold for the design of ghrelin receptor ligands: development of JMV 2959, a potent antagonist

A. Moulin, Jean Martinez, J. Fehrentz, 2013, Amino Acids.

Development of a novel fluorescent ligand of growth hormone secretagogue receptor based on the N-Terminal Leap2 region

S. Cantel, J. Fehrentz, S. Denoyelle, 2019, Molecular and Cellular Endocrinology.

Evidence Supporting a Role for Constitutive Ghrelin Receptor Signaling in Fasting-Induced Hyperphagia in Male Mice

J. Fehrentz, M. Perelló, J. Epelbaum, 2018, Endocrinology.

Structure and dynamics of G protein-coupled receptor–bound ghrelin reveal the critical role of the octanoyl chain

S. Cantel, A. Milon, J. Fehrentz, 2019, Proceedings of the National Academy of Sciences.

Quantitative MALDI‐MS Binding Assays: An Alternative to Radiolabeling

C. Enjalbal, S. Cantel, Jean Martínez, 2016, ChemMedChem.

Ghrelin receptor conformational dynamics regulate the transition from a preassembled to an active receptor:Gq complex

D. Pérahia, E. Trinquet, B. Mouillac, 2015, Proceedings of the National Academy of Sciences.

Concerted conformational dynamics and water movements in the ghrelin G protein-coupled receptor

P. Bisch, D. Pérahia, S. Cantel, 2021, eLife.

Agonism, Antagonism, and Inverse Agonism Bias at the Ghrelin Receptor Signaling*

Jean Martinez, J. Fehrentz, S. Denoyelle, 2015, The Journal of Biological Chemistry.

Design and Characterization of a Triazole-Based Growth Hormone Secretagogue Receptor Modulator Inhibiting the Glucoregulatory and Feeding Actions of Ghrelin.

S. Cantel, J. Fehrentz, S. Denoyelle, 2022, Biochemical pharmacology.