H. van de Langemheen

发表

Highly tunable thiosulfonates as a novel class of cysteine protease inhibitors with anti-parasitic activity against Schistosoma mansoni.

A. Kreidenweiss, R. J. Liskamp, E. Koehne, 2019, Bioorganic & medicinal chemistry.

Potential peptidic proteasome inhibitors by incorporation of an electrophilic trap based on amino acid derived α-substituted sulfonyl fluorides.

Arwin J. Brouwer, R. Liskamp, A. J. Brouwer, 2017, Bioorganic & medicinal chemistry.

Proteasome inhibition by new dual warhead containing peptido vinyl sulfonyl fluorides.

Arwin J. Brouwer, R. Liskamp, A. Ciaffoni, 2016, Bioorganic & medicinal chemistry.

Synthesis of tris-tertiary amine CycloTriVeratrilene (TACTV) derivatives as water soluble pre-organized three aromatic ring containing molecular scaffolds for the construction of protein mimics

Susan Gannon, D. Ward, H. van de Langemheen, 2019, Tetrahedron Letters.

Synthesis of cyclic peptides containing a thioester handle for native chemical ligation.

Arwin J. Brouwer, R. Liskamp, J. Kruijtzer, 2012, The Journal of organic chemistry.

An orthogonally protected CycloTriVeratrylene (CTV) as a highly pre-organized molecular scaffold for subsequent ligation of different cyclic peptides towards protein mimics.

H. van de Langemheen, R. Liskamp, Ondřej Longin, 2017, Bioorganic & medicinal chemistry.

Polar Hinges as Functionalized Conformational Constraints in (Bi)cyclic Peptides

Claire Wilson, C. Heinis, J. Bijl, 2017, Chembiochem : a European journal of chemical biology.

Synthesis of the TACO scaffold as a new selectively deprotectable conformationally restricted triazacyclophane based scaffold.

R. Liskamp, A. Ciaffoni, A. J. Brouwer, 2014, Organic letters.

Efficient synthesis of protein mimics by sequential native chemical ligation.

R. Liskamp, J. Kruijtzer, H. van de Langemheen, 2014, Organic letters.

Synthetic antibody protein mimics of infliximab by molecular scaffolding on novel CycloTriVeratrilene (CTV) derivatives.

M. Hezwani, H. van de Langemheen, R. Liskamp, 2018, Organic & biomolecular chemistry.

Immobilization by Surface Conjugation of Cyclic Peptides for Effective Mimicry of the HCV-Envelope E2 Protein as a Strategy toward Synthetic Vaccines.

Arvind H. Patel, R. Liskamp, J. Dunlop, 2018, Bioconjugate chemistry.

Dual role of isocitrate lyase 1 in the glyoxylate and methylcitrate cycles in Mycobacterium tuberculosis

James C Sacchettini, J. Sacchettini, E. Muñoz-Elías, 2006, Molecular microbiology.

Design, Synthesis, and Evaluation of a Diazirine Photoaffinity Probe for Ligand-Based Receptor Capture Targeting G Protein–Coupled Receptors

G. Milligan, A. Tobin, R. Liskamp, 2018, Molecular Pharmacology.

Scaffolded multiple cyclic peptide libraries for protein mimics by native chemical ligation.

R. Liskamp, J. Kruijtzer, H. van de Langemheen, 2014, Organic & biomolecular chemistry.

Potent and Highly Selective Inhibitors of the Proteasome Trypsin-like Site by Incorporation of Basic Side Chain Containing Amino Acid Derived Sulfonyl Fluorides.

Arwin J. Brouwer, R. Liskamp, A. J. Brouwer, 2018, Journal of medicinal chemistry.