G. Raidaru

发表

Fluorescent photoaffinity probes for mitotic protein kinase Aurora A.

A. Uri, Darja Lavogina, Katariina Kisand, 2015, Bioorganic & medicinal chemistry letters.

Selective Bisubstrate Inhibitors with Sub‐nanomolar Affinity for Protein Kinase Pim‐1

S. Knapp, E. Enkvist, A. Uri, 2013, ChemMedChem.

Bisubstrate inhibitor approach for targeting mitotic kinase Haspin.

S. Knapp, A. Chaikuad, A. Uri, 2015, Bioconjugate chemistry.

Liquid-phase synthesis of a pegylated adenosine-oligoarginine conjugate, cell-permeable inhibitor of cAMP-dependent protein kinase.

M. Pooga, K. Padari, J. Subbi, 2003, Bioorganic & medicinal chemistry letters.

Synthesis of Potential Purinoceptor Antagonists: Application of P1-tBu Phosphazene Base for Alkylation of Adenine in Solution and on Solid Phase

J. Boyer, J. Subbi, E. Enkvist, 2006, Nucleosides, nucleotides & nucleic acids.

Adenosine-derived non-phosphate antagonists for P2Y(1) purinoceptors.

J. Järv, M. Kelve, J. Subbi, 2000, Biochemical and biophysical research communications.

P 5 Calpain-mediated activation of cyclin dependent kinase 5 is critical for alpha-synuclein toxicity in vitro

O. Issinger, Lawrence W. Miller, K. Niefind, 2012 .

Synthesis of N-protected erythro-phenylalanylepoxides

J. Järv, Ü. Langel, M. Zetterström, 1995 .

Synthesis of 4,4′-Dibromobenzilic Acid

U. Mäeorg, U. Soomets, A. Perkson, 1994 .

[35S]GTPγS autoradiography reveals a wide distribution of Gi/o‐linked ADP receptors in the nervous system: close similarities with the platelet P2YADP receptor

J. Laitinen, R. Miettinen, A. Uri, 2001 .

Kinetic analysis of inhibition of cAMP-dependent protein kinase catalytic subunit by the peptide-nucleoside conjugate AdcAhxArg6.

J. Järv, A. Kuznetsov, A. Uri, 2004, Bioorganic chemistry.

Adenosine-5'-carboxylic acid peptidyl derivatives as inhibitors of protein kinases.

J. Järv, M. Loog, A. Uri, 1999, Bioorganic & medicinal chemistry letters.

Carbocyclic 3'-deoxyadenosine-based highly potent bisubstrate-analog inhibitor of basophilic protein kinases.

E. Enkvist, A. Uri, T. Pehk, 2007, Bioorganic & medicinal chemistry letters.

Adenosine analogue-oligo-arginine conjugates (ARCs) serve as high-affinity inhibitors and fluorescence probes of type I cGMP-dependent protein kinase (PKGIalpha).

C. Nickl, W. Dostmann, E. Enkvist, 2010, Biochimica et biophysica acta.

High-affinity bisubstrate probe for fluorescence anisotropy binding/displacement assays with protein kinases PKA and ROCK.

E. Enkvist, A. Uri, Kaido Viht, 2009, Analytical biochemistry.

Structural analysis of ARC-type inhibitor (ARC-1034) binding to protein kinase A catalytic subunit and rational design of bisubstrate analogue inhibitors of basophilic protein kinases.

D. Bossemeyer, E. Enkvist, A. Uri, 2009, Journal of medicinal chemistry.

Surface-plasmon-resonance-based biosensor with immobilized bisubstrate analog inhibitor for the determination of affinities of ATP- and protein-competitive ligands of cAMP-dependent protein kinase.

F. Herberg, A. Uri, Kaido Viht, 2007, Analytical biochemistry.

Conjugation of adenosine and hexa-(D-arginine) leads to a nanomolar bisubstrate-analog inhibitor of basophilic protein kinases.

E. Enkvist, A. Uri, Kaido Viht, 2006, Journal of medicinal chemistry.

Protein-induced long lifetime luminescence of nonmetal probes.

E. Enkvist, A. Uri, G. Raidaru, 2011, ACS chemical biology.

Effect of the structure of adenosine mimic of bisubstrate-analog inhibitors on their activity towards basophilic protein kinases.

E. Enkvist, A. Uri, G. Raidaru, 2009, Bioorganic & medicinal chemistry letters.

Fluorometric TLC assay for evaluation of protein kinase inhibitors.

E. Enkvist, A. Uri, Kaido Viht, 2005, Analytical biochemistry.

Acetoxymethyl Ester of Tetrabromobenzimidazole-Peptoid Conjugate for Inhibition of Protein Kinase CK2 in Living Cells.

O. Issinger, B. Guerra, E. Enkvist, 2015, Bioconjugate chemistry.

A subnanomolar fluorescent probe for protein kinase CK2 interaction studies.

O. Issinger, K. Niefind, E. Enkvist, 2012, Organic & biomolecular chemistry.

Conjugates of 5-isoquinolinesulfonylamides and oligo-D-arginine possess high affinity and selectivity towards Rho kinase (ROCK).

E. Enkvist, A. Uri, Darja Lavogina, 2012, Bioorganic & medicinal chemistry letters.

Identification of the ability of highly charged nanomolar inhibitors of protein kinases to cross plasma membranes and carry a protein into cells.

M. Pooga, K. Padari, J. Subbi, 2002, Bioorganic & medicinal chemistry letters.

Phosphate-substituted ATP analogs are antagonists at human P2Y1 purinoceptors.

J. Järv, K. Sak, G. Raidaru, 2000, Archives of biochemistry and biophysics.

Bifunctional Ligands for Inhibition of Tight-Binding Protein-Protein Interactions.

M. Zaccolo, R. Engh, K. A. Alam, 2016, Bioconjugate chemistry.

D2 dopamine receptor-G protein coupling. Cross-regulation of agonist and guanosine nucleotide binding sites

K. Fuxe, A. Terasmaa, A. Rinken, 2001, Neuroscience Letters.

[(35)S]GTPgammaS autoradiography reveals a wide distribution of G(i/o)-linked ADP receptors in the nervous system: close similarities with the platelet P2Y(ADP) receptor.

J. Laitinen, R. Miettinen, A. Uri, 2001, Journal of Neurochemistry.