Melissa D'Ascenzio

发表

S. Carradori, D. Secci, A. Bolasco, 2012, Expert opinion on therapeutic patents.

An Activity‐Based Probe Targeting Non‐Catalytic, Highly Conserved Amino Acid Residues within Bromodomains

M. Schirle, S. Knapp, O. Fedorov, 2018, Angewandte Chemie.

Synthesis, anti-Candida activity, and cytotoxicity of new (4-(4-iodophenyl)thiazol-2-yl)hydrazine derivatives.

S. Carradori, L. Polletta, D. Secci, 2012, European journal of medicinal chemistry.

Selective MAO-B inhibitors: a lesson from natural products

S. Carradori, D. Secci, A. Bolasco, 2014, Molecular Diversity.

Conventional and Microwave-Assisted Synthesis of Benzimidazole Derivatives and Their In Vitro Inhibition of Human Cyclooxygenase

S. Carradori, D. Secci, M. Yáñez, 2012 .

Salen and tetrahydrosalen derivatives act as effective inhibitors of the tumor-associated carbonic anhydrase XII--a new scaffold for designing isoform-selective inhibitors.

C. De Monte, S. Carradori, C. Supuran, 2013, Bioorganic & medicinal chemistry letters.

Open saccharin-based secondary sulfonamides as potent and selective inhibitors of cancer-related carbonic anhydrase IX and XII isoforms

S. Carradori, A. Mollica, C. Supuran, 2016, Journal of enzyme inhibition and medicinal chemistry.

Discovery and optimization of pyrazoline derivatives as promising monoamine oxidase inhibitors.

S. Carradori, D. Secci, E. Maccioni, 2012, Current topics in medicinal chemistry.

Design, synthesis and biological characterization of thiazolidin-4-one derivatives as promising inhibitors of Toxoplasma gondii.

C. De Monte, S. Carradori, D. Secci, 2014, European journal of medicinal chemistry.

Synthesis and anti-Helicobacter pylori Activity of 4-(Coumarin-3-yl)thiazol-2-ylhydrazone Derivatives.

S. Carradori, D. Secci, F. Sisto, 2011 .

Synthesis and anti-Helicobacter pylori activity of 4-(coumarin-3-yl)thiazol-2-ylhydrazone derivatives

S. Carradori, D. Secci, F. Sisto, 2010 .

Microwave and ultrasound-assisted synthesis of thiosemicarbazones and their corresponding (4,5-substituted-thiazol-2-yl)hydrazines

S. Carradori, D. Secci, A. Bolasco, 2014 .

Recent advances in the development of selective human MAO-B inhibitors: (hetero)arylidene-(4-substituted-thiazol-2-yl)hydrazines.

S. Carradori, D. Secci, R. Nescatelli, 2012, European journal of medicinal chemistry.

Synthesis, biological evaluation and quantitative structure-active relationships of 1,3-thiazolidin-4-one derivatives. A promising chemical scaffold endowed with high antifungal potency and low cytotoxicity.

C. De Monte, S. Carradori, R. Grande, 2017, European journal of medicinal chemistry.

Synthesis and biological evaluation of novel 2,4-disubstituted-1,3-thiazoles as anti-Candida spp. agents.

S. Carradori, D. Secci, A. Granese, 2011, European journal of medicinal chemistry.

(Thiazol-2-yl)hydrazone derivatives from acetylpyridines as dual inhibitors of MAO and AChE: synthesis, biological evaluation and molecular modeling studies

C. De Monte, S. Carradori, R. Di Santo, 2015, Journal of enzyme inhibition and medicinal chemistry.

Selective MAO-B inhibitors: a lesson from natural products

S. Carradori, D. Secci, A. Bolasco, 2013, Molecular Diversity.

Evaluation of a large library of (thiazol-2-yl)hydrazones and analogues as histone acetyltransferase inhibitors: enzyme and cellular studies.

C. De Monte, S. Carradori, L. Altucci, 2014, European journal of medicinal chemistry.

4-(3-Nitrophenyl)thiazol-2-ylhydrazone derivatives as antioxidants and selective hMAO-B inhibitors: synthesis, biological activity and computational analysis

S. Carradori, G. Zengin, D. Secci, 2019, Journal of enzyme inhibition and medicinal chemistry.

Identification of the stereochemical requirements in the 4-aryl-2-cycloalkylidenhydrazinylthiazole scaffold for the design of selective human monoamine oxidase B inhibitors.

C. De Monte, S. Carradori, L. Mannina, 2014, Bioorganic & medicinal chemistry.

Synthesis and selective inhibition of human monoamine oxidases of a large scaffold of (4,5-substituted-thiazol-2-yl)hydrazones

S. Carradori, D. Secci, M. Yáñez, 2010 .

Exploring 4-substituted-2-thiazolylhydrazones from 2-, 3-, and 4-acetylpyridine as selective and reversible hMAO-B inhibitors.

S. Carradori, R. Silvestri, D. Secci, 2013, European journal of medicinal chemistry.

Synthesis and Selective Human Monoamine Oxidase B Inhibition of Heterocyclic Hybrids Based on Hydrazine and Thiazole Scaffolds

C. De Monte, S. Carradori, D. Secci, 2013, Archiv der Pharmazie.

Design, synthesis and evaluation of N-substituted saccharin derivatives as selective inhibitors of tumor-associated carbonic anhydrase XII.

C. De Monte, S. Carradori, C. Supuran, 2014, Bioorganic & medicinal chemistry.

A Combined Crystallographic and Theoretical Study Explains the Capability of Carboxylic Acids to Adopt Multiple Binding Modes in the Active Site of Carbonic Anhydrases.

E. Langella, S. Carradori, C. Supuran, 2016, Chemistry.

1,3-Dipolar cycloaddition, HPLC enantioseparation and docking studies of saccharin/isoxazole and saccharin/isoxazoline derivatives as selective carbonic anhydrase IX and XII inhibitors.

S. Carradori, C. Supuran, T. Tuccinardi, 2020, Journal of medicinal chemistry.

Selective inhibition of human carbonic anhydrases by novel amide derivatives of probenecid: synthesis, biological evaluation and molecular modelling studies.

S. Carradori, C. Supuran, D. Vullo, 2014, Bioorganic & medicinal chemistry.

New amide derivatives of Probenecid as selective inhibitors of carbonic anhydrase IX and XII: biological evaluation and molecular modelling studies.

C. De Monte, S. Carradori, A. Mollica, 2015, Bioorganic & medicinal chemistry.

Synthesis and pharmacological screening of a large library of 1,3,4-thiadiazolines as innovative therapeutic tools for the treatment of prostate cancer and melanoma.

C. De Monte, S. Carradori, A. Mollica, 2015, European journal of medicinal chemistry.

Cyclic tertiary sulfamates: selective inhibition of the tumor-associated carbonic anhydrases IX and XII by N- and O-substituted acesulfame derivatives.

C. De Monte, S. Carradori, C. Supuran, 2014, European journal of medicinal chemistry.

Synthesis and pharmacological screening of a large library of 1,3,4-thiadiazolines as innovative therapeutic tools for the treatment of prostate cancer and melanoma.

S. Carradori, A. Mollica, D. Secci, 2015, European journal of medicinal chemistry.