Sean Riley

The novel sphingosine-1-phosphate receptors antagonist AD2900 affects lymphocyte activation and inhibits T-cell entry into the lymph nodes.

H. Rosen, S. Gatt, A. Dagan, 2017, Oncotarget.

Novel selective allosteric and bitopic ligands for the S1P(3) receptor.

Steven J Brown, S. Schürer, M. Guerrero, 2012, ACS chemical biology.

Design, Synthesis, and In Vitro and In Vivo Evaluation of an (18)F-Labeled Sphingosine 1-Phosphate Receptor 1 (S1P1) PET Tracer.

Steven J Brown, Hongjun Jin, Xuyi Yue, 2016, Journal of medicinal chemistry.

Bitopic Sphingosine 1-Phosphate Receptor 3 (S1P3) Antagonist Rescue from Complete Heart Block: Pharmacological and Genetic Evidence for Direct S1P3 Regulation of Mouse Cardiac Conduction

Steven J Brown, A. McCulloch, P. Gonzalez-Cabrera, 2016, Molecular Pharmacology.

Identification of Zika Virus Inhibitors Using Homology Modeling and Similarity-Based Screening to Target Glycoprotein E

R. Rizzo, T. D. McGee, A. Jacobs, 2020, Biochemistry.

A novel selective androgen receptor modulator (SARM) MK-4541 exerts anti-androgenic activity in the prostate cancer xenograft R–3327G and anabolic activity on skeletal muscle mass & function in castrated mice

H. Wilkinson, S. Alves, M. Gentile, 2016, The Journal of Steroid Biochemistry and Molecular Biology.

A novel high-throughput activity assay for the Trypanosoma brucei editosome enzyme REL1 and other RNA ligases

Rommie E. Amaro, A. Schnaufer, R. Amaro, 2015, Nucleic acids research.

Design and Synthesis of a Novel and Selective Kappa Opioid Receptor (KOR) Antagonist (BTRX-335140).

Steven J Brown, M. Urbano, M. Guerrero, 2019, Journal of medicinal chemistry.

Fluorometric High-Throughput Screening Assay for Secreted Phospholipases A2 Using Phospholipid Vesicles

Steven J Brown, M. Gelb, T. Spicer, 2016, Journal of biomolecular screening.