Y. Fukuda

发表

Synthesis and antibacterial activity of novel pyrido[1,2,3-de][1,4]benzoxazine-6-carboxylic acid derivatives carrying the 3-cyclopropylaminomethyl-4-substituted-1-pyrrolidinyl group as a C-10 substituent.

Tetsuya Kimura, M. Takei, Y. Asahina, 2008, Journal of medicinal chemistry.

Structure activity relationship of N-1 substituted 1,5-naphthyrid-2-one analogs of oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents (Part-9).

Akinori Nishimura, P. Meinke, D. Olsen, 2022, Bioorganic & medicinal chemistry letters.

Kibdelomycin Is a Bactericidal Broad-Spectrum Aerobic Antibacterial Agent

C. Garlisi, Carl J. Balibar, P. Dayananth, 2015, Antimicrobial Agents and Chemotherapy.

Synthesis and structure-activity relationship studies of highly potent novel oxazolidinone antibacterials.

A. Kojima, T. Komine, Y. Asahina, 2008, Journal of medicinal chemistry.

In Vitro and In Vivo Characterization of the Novel Oxabicyclooctane-Linked Bacterial Topoisomerase Inhibitor AM-8722, a Selective, Potent Inhibitor of Bacterial DNA Gyrase

Akinori Nishimura, Jin Wu, C. Garlisi, 2016, Antimicrobial Agents and Chemotherapy.

Synthetic studies on duocarmycin. 2. Synthesis and cytotoxicity of natural (+)-duocarmycin A and its three possible stereoisomers.

K. Nakatani, S. Terashima, Y. Fukuda, 1994 .

Synthetic studies on duocarmycin. 1. Total synthesis of dl-duocarmycin A and its 2-epimer

K. Nakatani, Y. Fukuda, Y. Itoh, 1994 .

Synthesis and cytotoxicity of enantiomeric pairs of duocarmycin a and its 2-epimer

K. Nakatani, S. Terashima, Y. Fukuda, 1992 .

DNA alkylation properties of the duocarmycins: (+)-duocarmycin A, epi-(+)-duocarmycin A, ent-(−)-duocarmycin A and epi,ent-(−)-duocarmycin A

D. Boger, K. Nakatani, S. Terashima, 1992 .

First total synthesis of dl-duocarmycin A

K. Nakatani, S. Terashima, Yoshio N Ito, 1990 .

Synthesis and Cytotoxicity of Various Structural Types of Novel Cyclopropapyrroloindole(CPI) Derivatives

H. Furuta, S. Terashima, Y. Oomori, 1998 .

Structures of kibdelomycin bound to Staphylococcus aureus GyrB and ParE showed a novel U-shaped binding mode.

N. Sharma, K. Lumb, Sangita Patel, 2014, ACS chemical biology.

A novel synthesis of (+)-duocarmycin SA

S. Terashima, Y. Fukuda, 1997 .

Stereoselective synthesis of cis-2-fluorocyclopropanecarboxylic acid.

Y. Fukuda, Taku Shibue, 2014, The Journal of organic chemistry.

Novel cyclopropapyrroloindole derivative (AT-3510) bearing methoxycarbonyl and trifluoromethyl groups.

H. Furuta, S. Terashima, Y. Oomori, 1999, Journal of medicinal chemistry.

Synthesis and antitumor activity of novel cyclopropapyrroloindole (CPI) derivatives bearing bis(methoxycarbonyl) groups

S. Terashima, Y. Oomori, Y. Fukuda, 1997 .

Synthetic Studies on Duocarmycin. Part 2. Synthesis and Cytotoxicity of Natural (+)-Duocarmycin A and Its Three Possible Stereoisomers.

K. Nakatani, S. Terashima, Y. Fukuda, 1994 .

The novel cyclopropapyrroloindole(CPI) bisalkylators bearing methoxycarbonyl and trifluoromethyl groups.

H. Furuta, S. Terashima, Y. Oomori, 1998, Bioorganic & medicinal chemistry letters.

Synthesis and antitumor activity of novel cyclopropapyrroloindole(CPI) derivatives bearing methoxycarbonyl and trifluoromethyl groups

H. Furuta, S. Terashima, F. Shiga, 1997 .

First Total Synthesis of dl‐Duocarmycin A (I).

K. Nakatani, S. Terashima, Yoshio N Ito, 1992 .

Synthetic Studies on Duocarmycin. Part 1. Total Synthesis of dl‐ Duocarmycin A and Its 2‐Epimer.

K. Nakatani, S. Terashima, Y. Fukuda, 1994 .

Studies on Conjugated Nitriles. VII. Lewis Acid-Promoted Reaction of Active Methylene Compounds with Diethyl Phosphorocyanidate; Preparation of α, β-Unsaturated α-Aminophosphonates

M. Sakamoto, T. Kawasaki, Y. Fukuda, 1994 .

Structure activity relationship of C-2 ether substituted 1,5-naphthyridine analogs of oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents (Part-5).

Akinori Nishimura, Jin Wu, P. Meinke, 2015, Bioorganic & medicinal chemistry letters.

Hydroxy tricyclic 1,5-naphthyridinone oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents-SAR of RHS moiety (Part-3).

R. Nargund, Akinori Nishimura, Jin Wu, 2015, Bioorganic & medicinal chemistry letters.

Tricyclic 1,5-naphthyridinone oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents-SAR of left-hand-side moiety (Part-2).

Leo A. Joyce, E. Sherer, R. Nargund, 2015, Bioorganic & medicinal chemistry letters.

Oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad spectrum antibacterial agents.

Sangita Patel, Jin Wu, P. Meinke, 2014, ACS medicinal chemistry letters.

C1–C2-linker substituted 1,5-naphthyridine analogues of oxabicyclooctane-linked NBTIs as broad-spectrum antibacterial agents (part 7)

Akinori Nishimura, Jin Wu, Xuanjia Peng, 2015 .

Structure activity relationship of pyridoxazinone substituted RHS analogs of oxabicyclooctane-linked 1,5-naphthyridinyl novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents (Part-6).

Akinori Nishimura, Jin Wu, Xuanjia Peng, 2015, Bioorganic & medicinal chemistry letters.

Efficient synthesis of cyclopropylhydrazine salts

Y. Fukuda, Taku Shibue, 2014 .

Hydroxy tricyclic 1,5-naphthyridinone oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents-SAR of RHS moiety (Part-3).

R. Nargund, Akinori Nishimura, Jin Wu, 2015, Bioorganic & medicinal chemistry letters.