P. S. Watson

发表

A diastereoselective synthesis of 2,4-disubstituted piperidines: scaffolds for drug discovery.

B. Jiang, B. Jiang, P. S. Watson, 2000, Organic letters.

Lipophilic modifications to dinucleoside polyphosphates and nucleotides that confer antagonist properties at the platelet P2Y12 receptor.

J. Boyer, J. Douglass, C. Redick, 2008, Journal of medicinal chemistry.

CCR3 antagonists: a potential new therapy for the treatment of asthma. Discovery and structure-activity relationships.

G. Trainor, M. Covington, C. Decicco, 2002, Bioorganic & medicinal chemistry letters.

Adenosine analogues as inhibitors of P2Y12 receptor mediated platelet aggregation.

J. Boyer, S. Mahanty, J. Douglass, 2008, Bioorganic & medicinal chemistry letters.

2,4-Disubstituted piperidines as selective CC chemokine receptor 3 (CCR3) antagonists: synthesis and selectivity.

G. Trainor, M. Covington, C. Decicco, 2006, Bioorganic & medicinal chemistry letters.

Discovery of N-propylurea 3-benzylpiperidines as selective CC chemokine receptor-3 (CCR3) antagonists.

G. Trainor, M. Covington, C. Decicco, 2004, Bioorganic & medicinal chemistry letters.

Examination of the olefin–olefin ring closing metathesis to prepare Latrunculin B

J. Lampe, J. She, P. S. Watson, 2009 .

Synthesis and intramolecular photocycloadditions of 2-acyloxy-3-hexenoyl cyclohexenones: Diastereoselectivity in the intramolecular [2+2] photocycloadditions of alkenes and cyclohexenones tethered by four atoms

B. W. King, M. Crimmins, L. E. Guise, 1997 .

Nonconventional Stereochemical Issues in the Design of the Synthesis of the Vancomycin Antibiotics: Challenges Imposed by Axial and Nonplanar Chiral Elements in the Heptapeptide Aglycons.

T. I. Richardson, Davidr . Evans, C. Dinsmore, 1998, Angewandte Chemie.

Strategy for the enantioselective synthesis of trans-2,4-disubstituted piperidines: application to the CCR3 antagonist IS811.

W. A. Nugent, P. S. Watson, G. Kauffman, 2006, The Journal of organic chemistry.

Addition of Zinc Homoenolates to Acetylenic Esters and Amides: A Formal [3 + 2] Cycloaddition

P. Nantermet, M. Crimmins, A. Cheung, 1993 .

Indazoles: regioselective protection and subsequent amine coupling reactions.

J. Lampe, W. Bodnar, David J. Slade, 2009, The Journal of organic chemistry.

Synthesis and Intramolecular Photocycloadditions of 2-Acyloxy-3-hexenoyl Cyclohexenones: Diastereoselectivity in the Intramolecular [2 + 2] Photocycloadditions of Alkenes and Cyclohexenones Tethered by Four Atoms.

B. W. King, M. Crimmins, L. E. Guise, 2010 .

Stereoselective intramolecular enone-olefin photocycloadditions of 1,7-dienes: Model studies on the synthesis of lycopodium alkaloids

M. Crimmins, P. S. Watson, 1993 .

Synthesis of the orienticin C M(2–4) macrocycle utilizing a nucleophilic aromatic substitution strategy

Davidr . Evans, P. S. Watson, 1996 .

Discovery of N-propylurea 3-benzylpiperidines as selective CC chemokine receptor-3 (CCR3) antagonists.

G. Trainor, M. Covington, C. Decicco, 2004, Bioorganic & medicinal chemistry letters.

From rigid cyclic templates to conformationally stabilized acyclic scaffolds. Part I: the discovery of CCR3 antagonist development candidate BMS-639623 with picomolar inhibition potency against eosinophil chemotaxis.

I. Kariv, S. Mandlekar, A. Tebben, 2008, Bioorganic & medicinal chemistry letters.

Approaches to the Synthesis of the Vancomycin Antibiotics. Synthesis of Orienticin C (Bis-dechlorovancomycin) Aglycon

J. Barrow, Davidr . Evans, J. Ellman, 1997 .

Approaches to the Synthesis of the Vancomycin Antibiotics. Synthesis of Orienticin C (Bis-dechlorovancomycin) Aglycon (I).

J. Barrow, Davidr . Evans, J. Ellman, 1997 .