T. Bardos

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Oligonucleotides containing modified bases. I. Inhibition of DNA and RNA polymerases by partially thiolated oligocytidylic acids.

M. Kung, Y. Ho, T. Bardos, 1976, Biochemical and biophysical research communications.

Modified telomeric repeat amplification protocol: a quantitative radioactive assay for telomerase without using electrophoresis.

I. Szatmári, J. Aradi, T. Bardos, 2000, Analytical biochemistry.

Antimetabolites: molecular design and mode of action.

T. Bardos, 1974, Topics in current chemistry.

Structure-activity relationships and mode of action of 5-mercapto-substituted oligo- and polynucleotides as antitemplates inhibiting replication of human immunodeficiency virus type 1

R. Schinazi, K. H. Ling, T. Bardos, 1992, Antimicrobial Agents and Chemotherapy.

Anti-Tumour Activity of 5-Mercaptouracil

J. Ambrus, A. Segaloff, T. Bardos, 1959, Nature.

Cyclophosphamide, 2,2-dimethylaziridines and other alkylating agents as inhibitors of serum cholinesterase.

D. Lalka, T. Bardos, 1975, Biochemical pharmacology.

CHEMICAL AND ENZYMATIC METHODS IN THE SYNTHESIS OF MODIFIED POLYNUCLEOTIDES

Y. Ho, T. Bardos, 1978 .

Effects of 5-mercapto-2'-deoxyuridine on the incorporation of nucleosides into RNA and DNA in a primary lymphocyte culture system.

T. Bardos, D. Bogyo, Z. Chmielewicz, 1976, Cancer research.

Uptake of partially thiolated DNA by ascites tumor cells.

V. Paffenholz, Y. Ho, T. Bardos, 1976, Cancer research.

Uptake of PartiallyThiolated DNA by AscitesTumor Cells1

V. Paffenholz, Y. Ho, T. Bardos, 1976 .

Synthetic porphyrins. I. Synthesis and spectra of some para‐substituted meso ‐ Tetraphenylporphines

N. Datta-Gupta, T. Bardos, N. Datta-gupta, 1966 .

Structural characterization of partially thiolated poly(cytidylic acid).

R. Fiel, J. Aradi, Y. Ho, 1979, Biochemistry.

Synthesis of 5-Ethyl-2-pyrimidinone-2′-deoxyriboside as a New Potential Antiviral Agent

S. Trehan, T. Bardos, J. Macdiarmid, 1994 .

Chapter 28. Nucleosides and Nucleotides

T. Bardos, 1968 .

Crystal and molecular structure of 5-[1-(2′-deoxy-α-d-ribofuranosyl)uracilyl] disulfide

E. Shefter, T. Bardos, M. Kotick, 1967 .

Pyrimido[5,4-b]quinolines. III. Synthesis of 10-alkyl-substituted 10-deazaalloxazines

C. K. Chu, T. Bardos, 1977 .

Synthesis and properties of bis(2,2-dimethylaziridinyl)phosphinic amides: a series of new antineoplastic agents.

W. Rose, J. Ambrus, M. Perlman, 1985, Journal of medicinal chemistry.

Synthesis of some 1,3,8-trisubstituted pyrimido[4,5-c][2,7]-naphthyridin-6-ones as potential antitumor agents

A. Gangjee, T. Kalman, T. Bardos, 1984 .

SYNTHESIS OF POTENTIAL "DUAL ANTAGONISTS." I. SOME BIS(1-AZIRIDINYL)PHOSPHINYL CARBAMATES AND THEIR STRUCTURAL ANALOGS.

T. Bardos, Z. B. Papanastassiou, 1962, Journal of medicinal and pharmaceutical chemistry.

A STUDY OF COMPARATIVE CHEMICAL AND BIOLOGICAL ACTIVITIES OF ALKYLATING AGENTS.

D. Triggle, T. Bardos, N. Datta-gupta, 1965, Journal of medicinal chemistry.

Synthesis of 5-S-substituted 2'-deoxyuridines. Study of the factors influencing stereoselectivity of the silyl modification of the Hilbert-Johnson reaction.

C. Szántay, T. Bardos, M. Kotick, 1969, The Journal of organic chemistry.

Measurement of the Inversion Rate of a Secondary Amine and Its N-Deuterio Analog by Nuclear Magnetic Resonance Spectroscopy1

C. Szántay, T. Bardos, C. Navada, 1965 .

Synthesis, molecular symmetry, and chemical reactivity of C-aryl-substituted phosphoraziridines

M. Perlman, T. Bardos, 1988 .

5-mercaptodeoxyuridine--its enzymatic synthesis and mode of action in microbiological systems.

T. Kalman, A. Bloch, T. Bardos, 1969, Biochemical pharmacology.

Mechanisms of reactions of ring-substituted bis(1-aziridinyl)phosphinyl urethan antineoplastic agents.

T. Bardos, Z. Chmielewicz, C. Navada, 1970, Journal of pharmaceutical sciences.

Synthesis of Potential Dual Antagonists III

T. Bardos, A. K. Barua, Z. B. Papanastassiou, 1965 .

SYNTHESIS OF POTENTIAL DUAL ANTAGONISTS. 3. RING-SUBSTITUTED ETHYL (BIS(1-AZIRIDINYL)PHOSPHINYL)CARBAMATES.

T. Bardos, A. K. Barua, Z. B. Papanastassiou, 1965, Journal of pharmaceutical sciences.

Chapter 31. Nucleosides and Nucleotides

T. Bardos, 1970 .

Synthesis of 5-Mercaptocytosine Nucleosides and Nucleotides

G. Szekeres, Y. Ho, T. Bardos, 1983 .

Biochemical parameters of neoplasia. II. Some macromolecular properties of deoxyribonucleic acid from normal and neoplastic human tissue.

R. Fiel, J. Ambrus, T. Bardos, 1965, Cancer research.

Synthetic porphyrins. II. Preparation and spectra of some metal chelates of para-substituted-meso-tetraphenylporphines.

T. Bardos, N. Datta-gupta, 1968, Journal of pharmaceutical sciences.

Ionic inhibition of growth in Lactobacillus leichmannii 313 and its reversal with vitamin B12.

T. Bardos, H. L. Gordon, 1953 .

Potent inhibition of HIV-1 entry by (s4dU)35.

J. Szöllősi, L. Fésüs, K. Watson, 2005, Virology.

A Synthetic Compound with Folinic Acid Activity

W. Shive, T. Bardos, E. H. Flynn, 1951 .

Synthetic'members of the folinic acid group.

W. Shive, T. Bardos, L. Rogers, 1950 .

INTERACTION OF LASER RADIATION WITH BIOLOGIC SYSTEMS. 3. STUDIES ON BIOLOGIC SYSTEMS IN VITRO.

E. Neter, S. Fine, J. Ambrus, 1965, Federation proceedings.

Synthesis and inhibition analysis of 2(4)-imino-4(2)-amino-2,4-dideoxyriboflavin, a dual antagonist of riboflavin and folinic acid.

C. K. Chu, T. Bardos, 1977, Journal of medicinal chemistry.

Synthetic and Degradative Investigations of the Structure of Folinic Acid-SF

W. Shive, J. Ravel, M. May, 1951 .

The folinic acid group, a series of new vitamins related to folic acid.

W. Shive, T. Bardos, Margaret E. Sibley, 1949 .

Comparative study of the thymidine kinase and thymidylate kinase activities and of the feedbach inhibition of thymidine kinase in normal and neoplastic human tissue.

J. Ambrus, T. Bardos, Z. Chmielewicz, 1968, Cancer research.

MOLECULAR APPROACHES TO INHIBIT ONCOGENESIS BY RNA TUMOR VIRUSES

P. Chandra, A. Götz, B. Mildner, 1977, Annals of the New York Academy of Sciences.

Action of partially thiolated polynucleotides on the DNA polymerase alpha from regenerating rat liver.

M. Kung, Y. Ho, T. Bardos, 1976, Cancer research.

POLYNUCLEOTIDES CONTAINING 5‐MERCAPTO‐SUBSTITUTED PYRIMIDINES: INHIBITION OF VIRAL DNA POLYMERASES AND THE BIOLOGICAL IMPLICATION *

P. Chandra, A. Mikulski, U. Ebener, 1975, Annals of the New York Academy of Sciences.

Synthesis of Deoxyalloxazines (Benzopteridines)1

T. Bardos, D. B. Olsen, T. Enkoji, 1957 .

Synthesis of new nucleoside phosphoraziridines as potential site-directed antineoplastic agents.

W. Rose, J. A. Dunn, T. Bardos, 1990, Journal of medicinal chemistry.

Comparative chemical and biological studies of four prototype phosphoraziridine antineoplastic agents.

J. A. Dunn, T. Bardos, 1991, Biochemical pharmacology.

Synthesis of New Nucleoside Phosphoraziridines as Potential Site- Directed Antineoplastic Agents.

W. Rose, J. A. Dunn, T. Bardos, 1991 .

Synthesis and testing of quinone-based bis(2,2-dimethyl-1-aziridinyl)phosphinyl carbamates as radiation-potentiating antitumor agents.

T. Bardos, J. Macdiarmid, J. Earle, 1988, Journal of Medicinal Chemistry.

Synthesis of 5'-thymidinyl bis(1-aziridinyl)phosphinates as antineoplastic agents.

T. Bardos, L. Hsiao, 1981, Journal of Medicinal Chemistry.

Chemical mechanism of the radiation potentiating effects of 2,2-dimethylaziridine-type antitumor agents.

J. A. Dunn, M. Perlman, T. Bardos, 1979, International journal of radiation oncology, biology, physics.

Synthfsis of bis(aziridinyl)phosphinyl-N-hydroxyurethane derivatives as antineoplastic agents.

G. Wampler, W. Regelson, T. Bardos, 1975, Journal of medicinal chemistry.

Reactions of 2,2-dimethylaziridine-type alkylating agents in biological systems. I. Colorimetric estimation and stability in physiological media.

D. Lalka, T. Bardos, 1973, Journal of pharmaceutical sciences.

Combination of chemotherapy with dual antagonists and radiotherapy in the treatment of neoplastic disease

C. Ambrus, T. Bardos, J. L. Ambrus, 1971, Journal of surgical oncology.

Synthesis and chemotherapeutic effects of ethyl bis-(2,2-dimethyl)-ethylenamido phosphate. A preliminary report.

A. Munson, J. Ambrus, T. Bardos, 1967, Journal of pharmaceutical sciences.

Consideration of chemical reaction mechanisms in relationship to the biological action of "dual antagonists".

T. Bardos, 1962, Biochemical pharmacology.

‘Dual Antagonists’; Alkyl N-(bis-(ethylenimido)phosphoro)-carbamates; a New Series of Anti-Tumour Agents

A. Segaloff, T. Bardos, J. L. Ambrus, 1959, Nature.

Synthesis of potential dual-acting radiation sensitizer antineoplastic agents: 2,2-dimethylphosphoraziridines containing 2-nitroimidazoles or other electron-affinic moieties.

G. Wampler, W. Rose, J. A. Dunn, 1991, Journal of Medicinal Chemistry.

Reactions of 2,2-dimethylaziridine-type alkylating agents in biological systems II: comparative pharmacokinetics in dogs.

W. Jusko, D. Lalka, T. Bardos, 1975, Journal of Pharmacy and Science.

STRUCTURE‐ACTIVITY RELATIONSHIPS OF ALKYLATING AGENTS IN CANCER CHEMOTHERAPY *

T. Bardos, Z. Chmielewicz, P. Hebborn, 1969 .

Synthesis and biological activities of 2-Pyrimidinone Nucleosides. III.1,2 5-Alkynyl-2-Pyrimidinone 2′-Deoxyribosides

S. Efange, T. Bardos, Yung‐chi Cheng, 1985 .

Synthesis of 5‐methylmercaptopyrimidine nucleosides

T. Bardos, E. Ryu, 1979 .

Stereoselective synthesis of the anomeric 5-mercapto-2′-deoxyuridines and of some other α- and β-deoxyribonucleosides

C. Szántay, T. Bardos, M. Kotick, 1966 .

Differential Effects of 5-Methylmercapto-2′-Deoxyuridine on the Replication of Herpes Simplex Virus Type 1 in Two Cell Systems

K. Chadha, R. Hughes, Y. Ho, 1976, Antimicrobial Agents and Chemotherapy.

Methylation of 4-thio-2'-deoxyuridylate by thymidylate synthetase.

G. Szekeres, T. Kalman, A. Bloch, 1973, Biochemical and biophysical research communications.

Calvacin: A New Antitumor Agent.

R. U. Byerrum, J. Luck, C. Stock, 1960, Science.

PTERIDINOSTEROIDS. II. SYNTHESIS OF 17-BETA-ACETOXY-5-ALPHA-ANDROSTANO(2,3-G)-2',4'-DIAMINOPTERIDINE.

T. Bardos, Z. Chmielewicz, S. Raman, 1964, Journal of medicinal chemistry.

Anti-herpes simplex virus activity of 5-substituted 2-pyrimidinone nucleosides

Y. Cheng, M. Fisher, S. Efange, 1989, Antimicrobial Agents and Chemotherapy.

Simplified synthesis of 5-mercaptouracil riboside derivatives

F. J. Dinan, J. Barren, T. Bardos, 1982 .

The autoxidation of 5-mercaptouracil and 5-mercaptodeoxyuridine.

T. Kalman, T. Bardos, 1967, Journal of the American Chemical Society.

Synthesis of Compounds Related to Thymine. I. 5-Mercaptouracil and Some S-Substituted Derivatives

T. Bardos, R. R. Herr, T. Enkoji, 1955 .

The reaction of 5-bromouracil derivatives with sulfur nucleophiles, and a novel synthetic route to 5-sulfur-substituted uracils and nucleotides.

T. Kalman, T. Bardos, L. Szabo, 1970, The Journal of organic chemistry.

Diazoketone and chloromethylketone analogs of methotrexate as potential antitumor agents.

A. Gangjee, T. Kalman, T. Bardos, 1982, Journal of pharmaceutical sciences.

Synthesis of 1,2-dihydro-1-(2-deoxy- -D-erythro-pentofuranosyl)-2-oxopyrazine 4-oxide, a potent analog of deoxyuridine.

A. Bloch, T. Bardos, P. Berkowitz, 1973, Journal of medicinal chemistry.

Alterations of some macromolecular and biochemical properties of calf thymus DNA caused by "dual antagonists" and nitrogen mustard.

R. Fiel, J. Ambrus, T. Bardos, 1967, Cancer research.

Effect of increasing thiolation of the polycytidylic acid strand of poly I: poly C on the α, β and γ interferon-inducing properties, antiviral and antiproliferative activities

J. A. Dunn, J. Ambrus, K. Chadha, 2004 .

Studies on the chemistry, antitumor activity, and pharmacology of ethyl Di‐(2,2 ‐dimethyl)ethylenamido phosphate (AB‐163)

A. Munson, J. Ambrus, T. Bardos, 1969, Journal of surgical oncology.

SYNTHESIS OF POTENTIAL DUAL ANTAGONISTS IV. EFFECT OF RING SUBSTITUENTS ON THE ALKYLATING AND HYDROLYTIC PROPERTIES OF BIS-(1-AZIRIDINYL)PHOSPHINYL CARBAMATES.

T. Bardos, Z. Chmielewicz, C. Navada, 1965, Journal of pharmaceutical sciences.

STUDIES ON THE MECHANISM OF ACTION OF CYCLOPHOSPHAMIDE AND AB-132 WITH THE AID OF RADIOPROTECTIVE AGENTS.

A. Munson, N. Back, E. Achter, 1964, Life sciences.

Studies in the pharmacodynamics of mechlorethamine and AB 100.

R. Ausman, H. Hagedorn, J. Ambrus, 1961, JAMA.

Absence of cross-resistance to alkylating agents in cyclophosphamide-resistant L1210 leukemia.

G. Wampler, W. Regelson, T. Bardos, 1978, European journal of cancer.

SYNTHESIS OF BIS-(AZIRIDINYL)PHOSPHINYL-N-HYDROXYURETHANE DERIVATIVES AS ANTINEOPLASTIC AGENTS

G. Wampler, W. Regelson, T. Bardos, 1975 .

SYNTHESIS OF 5′-THYMIDINYL BIS(1-AZIRIDINYL)PHOSPHINATES AS ANTINEOPLASTIC AGENTS

T. Bardos, L. Hsiao, 1981 .

Radiation sensitizing agents in clinical radiation and chemotherapy.

J. Ambrus, C. Ambrus, T. Bardos, 1980, Journal of medicine.

Synthesis and Testing of Quinone-Based Bis(2,2-dimethyl-1-aziridinyl)phosphoryl Carbamates as Radiation-Potentiating Antitumor Agents.

T. Bardos, J. Macdiarmid, J. Earle, 1988 .

Laboratory and clinical evaluation of the radiation-potentiating activity of ethyl-N-bis (2,2-dimethylethylamidinophosphoro) carbamate (AB-132).

W. Regelson, J. Ambrus, C. Ambrus, 1975, Journal of medicine.

Synthesis of some new S-alkylated derivatives of 5-mercapto-2'-deoxyuridine as potential antiviral agents.

F. J. Dinan, T. Bardos, 1980, Journal of medicinal chemistry.

Synthesis and biological activities of 2-pyrimidinone nucleosides. 2. 5-Halo-2-pyrimidinone 2'-deoxyribonucleosides.

Y. Cheng, S. Efange, H. Shih, 1985, Journal of medicinal chemistry.

Synthesis and antiviral activity of 1-(2-deoxy-beta-D-ribofuranosyl)-5-(methylmercapto)-2-pyrimidinone.

Y. Cheng, A. Schroeder, T. Bardos, 1981, Journal of medicinal chemistry.

Spectrophotometric and chemical studies of 5-mercaptouracil, 5-mercaptodeoxyuridine, and their S-substituted derivatives.

T. Kalman, T. Bardos, 1966, Journal of pharmaceutical sciences.

Synthesis of Compounds Related to Thymine. II. Effect of Thymine Antagonists on the Biosynthesis of DNA

G. M. Levin, T. Bardos, R. R. Herr, 1955 .

Differential responses of DNA and RNA polymerase to modifications of the template rat liver DNA caused by action of the carcinogen acetylaminofluorene in vivo and in vitro.

S. Belman, J. Ambrus, W. Troll, 1968, Biochimica et biophysica acta.

Pyrazine nucleoside analogs. Synthesis and reactions of some 5-thio-substituted pyrazines

M. Bobek, P. Tuntiwachwuttikul, T. Bardos, 1991 .

Pyrazine Nucleoside Analogs. Synthesis and Reactions of Some 5‐ Thiosubstituted Pyrazines.

M. Bobek, P. Tuntiwachwuttikul, T. Bardos, 1991 .

Inhibition of DNA polymerase alpha from leukemic and normal human cells by partially thiolated human deoxyribonucleic acids.

J. Minowada, J. Aradi, Y. Ho, 1985, Cancer biochemistry biophysics.

Pteridinosteroids. A new type of folic acid antagonist with lipid solubility

A. Segaloff, T. Bardos, Z. Chmielewicz, 1963 .

SYNTHESIS AND ANTIVIRAL ACTIVITY OF 1-(2-DEOXY-β-D-RIBOFURANOSYL)-5-(METHYLMERCAPTO)-2-PYRIMIDINONE

A. Schroeder, T. Bardos, Yung‐chi Cheng, 1981 .

The nitration of 6-chloro-1-naphthoic acid.

C. Price, T. Bardos, H. I. Enos, 1948, Journal of the American Chemical Society.

Inhibition of DNA-dependent RNA polymerase with partially thiolated polynucleotides.

A. Mikulski, T. Kalman, T. Bardos, 1973, Biochimica et biophysica acta.

Enzymatic studies relating to the mode of action of 5-mercapto-2'-deoxyuridine.

T. Kalman, T. Bardos, 1970, Molecular pharmacology.

Plasma clearance and tissue distribution of partially thiolated polycytidylic acid and its degradation products in rodents.

M. Kung, D. Lalka, Y. Ho, 1984, Cancer research.

The activation of murine macrophages and natural killer cells by the partially thiolated double stranded RNA poly(I)-mercapto poly(C).

P. Cavanaugh, Y. Ho, T. Bardos, 1996, Research communications in molecular pathology and pharmacology.

Inhibition of some DNA polymerase activities from cultured Burkitt cells by thiolated ribonucleic acids.

T. Bardos, B. Srivastava, 1973, Life sciences.

A systematic investigation of the presence of growth-inhibitory substances in animal tissues.

M. V. Nadkarni, T. Bardos, Z. Chmielewicz, 1968, Cancer research.

Biochemical parameters of neoplasis. I. "Priming" activity of deoxyribonucleic acid from normal and neoplastic human tissues in a deoxyribonucleic acid polymerase system.

J. Ambrus, C. Ambrus, T. Bardos, 1965, Cancer research.

Enzymatic synthesis of polyuridylic acid containing modified bases.

J. Aradi, Y. Ho, T. Bardos, 1980, Nucleic acids research.

Effects of partially thiolated polycytidylic acid on the clonogenicity of murine leukemic stem cells.

H. Preisler, Y. Ho, T. Bardos, 1979, Cancer research.

Use of AB‐103 (a “dual antagonist”) in the treatment of bronchogenic carcinoma

J. Sokal, L. Stutzman, T. Bardos, 1961, Cancer.