Mauricio Cabrera

发表

Mutagenicity of N-oxide containing heterocycles and related compounds: experimental and theoretical studies.

Hugo Cerecetto, N. Campillo, Mercedes González, 2014, Current topics in medicinal chemistry.

Novel and Selective Rhipicephalus microplus Triosephosphate Isomerase Inhibitors with Acaricidal Activity

R. Pérez-Montfort, Rodrigo Nunes da Fonseca, J. Moraes, 2018, Veterinary sciences.

Discovery of Potent EGFR Inhibitors through the Incorporation of a 3D-Aromatic-Boron-Rich-Cluster into the 4-Anilinoquinazoline Scaffold: Potential Drugs for Glioma Treatment.

F. Teixidor, C. Viňas, Pablo Cabral, 2018, Chemistry.

Biotransformation of Phenazine 5,10-Dioxides under Hypoxic Conditions as an Example of Activation of Anticancer Prodrug: An Interdisciplinary Experiment for Biochemistry or Organic Chemistry

L. Thomson, H. Cerecetto, Mercedes González, 2013 .

Bioactive-guided Identification of Labdane Diterpenoids from Aerial Parts of Aristeguietia glutinosa as anti-Trypanosoma cruzi agents

H. Cerecetto, J. Varela, Mercedes González, 2012, Natural product communications.

Identification and characterization of human interferon alpha inhibitors through a WISH cell line-based reporter gene assay.

R. Kratje, M. Oggero, M. Bollati-Fogolín, 2019, Bioorganic chemistry.

3-Trifluoromethylquinoxaline N,N'-dioxides as anti-trypanosomatid agents. Identification of optimal anti-T. cruzi agents and mechanism of action studies.

A. López de Cerain, Diego Benítez, A. Monge, 2011, Journal of medicinal chemistry.

Study of benzo[a]phenazine 7,12-dioxide as selective hypoxic cytotoxin-scaffold. Identification of aerobic-antitumoral activity through DNA fragmentation.

M. Cascante, L. Pietrasanta, A. M. Bruno, 2010, Bioorganic & Medicinal Chemistry.

Identification of chalcones as in vivo liver monofunctional phase II enzymes inducers.

Marcelo Fernández, A. López de Cerain, A. Monge, 2010, Bioorganic & medicinal chemistry.

Synthetic chalcones, flavanones, and flavones as antitumoral agents: biological evaluation and structure-activity relationships.

E. Castellano, G. Seoane, A. Monge, 2007, Bioorganic & medicinal chemistry.

New copper-based complexes with quinoxaline N1,N4-dioxide derivatives, potential antitumoral agents.

Hugo Cerecetto, A. Costa-Filho, M. H. Torre, 2008, Journal of inorganic biochemistry.

Cytotoxic palladium complexes of bioreductive quinoxaline N1,N4-dioxide prodrugs.

B. Garat, P. Smircich, M. H. Torre, 2009, Bioorganic & medicinal chemistry.

Discovery of new orally effective analgesic and anti-inflammatory hybrid furoxanyl N-acylhydrazone derivatives.

L. M. Lima, E. Barreiro, M. Bollati-Fogolín, 2012, Bioorganic & medicinal chemistry.

Structural modifications on the phenazine N,N'-dioxide-scaffold looking for new selective hypoxic cytotoxins.

A. López de Cerain, A. Monge, H. Cerecetto, 2010, European journal of medicinal chemistry.

Differential enzymatic reductions governing the differential hypoxia-selective cytotoxicities of phenazine 5,10-dioxides.

H. Cerecetto, Mercedes González, Mauricio Cabrera, 2008, Chemical research in toxicology.

A serendipitous one-step conversion of 3H-1,2-dithiole-3-thione to (E)-3-[1-(alkylthio)alkylidene]-3H-1,2-dithiole: an experimental and theoretical study

H. Cerecetto, Mercedes González, G. Echeverría, 2014, Molecular Diversity.

Massive screening yields novel and selective Trypanosoma cruzi triosephosphate isomerase dimer-interface-irreversible inhibitors with anti-trypanosomal activity.

R. Pérez-Montfort, A. Gómez-Puyou, A. Merlino, 2010, European journal of medicinal chemistry.

Novel and selective inactivators of Triosephosphate isomerase with anti-trematode activity

D. Timson, C. Caffrey, Teresa Freire, 2020, Scientific Reports.

In vivo phase II-enzymes inducers, as potential chemopreventive agents, based on the chalcone and furoxan skeletons.

H. Cerecetto, Mercedes González, Mauricio Cabrera, 2016, Bioorganic & medicinal chemistry.

Drug Targets: Screening for Small Molecules that Inhibit Fasciola hepatica Enzymes.

Ileana Corvo, Guzmán Álvarez, Florencia Ferraro, 2020, Methods in molecular biology.

Cathepsin L Inhibitors with Activity against the Liver Fluke Identified From a Focus Library of Quinoxaline 1,4-di-N-Oxide Derivatives

A. Merlino, Ileana Corvo, H. Cerecetto, 2019, Molecules.

Identification of Chalcones as Fasciola hepatica Cathepsin L Inhibitors Using a Comprehensive Experimental and Computational Approach

J. Tort, A. Merlino, Ileana Corvo, 2016, PLoS neglected tropical diseases.

Novel and selective inactivators of Triosephosphate isomerase with anti-trematode activity

D. Timson, C. Caffrey, Teresa Freire, 2020, Scientific Reports.

Small-Molecule Kinase-Inhibitors-Loaded Boron Cluster as Hybrid Agents for Glioma-Cell-Targeting Therapy.

F. Teixidor, C. Viňas, Pablo Cabral, 2017, Chemistry.

Novel Phenazine 5,10-Dioxides Release •OH in Simulated Hypoxia and Induce Reduction of Tumour Volume In Vivo

M. Cascante, G. Pachón, A. López de Cerain, 2011, ISRN pharmacology.

Research Article Novel Phenazine 5,10-Dioxides ReleaseOH in Simulated Hypoxia and Induce Reduction of Tumour VolumeInVivo

M. Cascante, A. Monge, H. Cerecetto, 2011 .

3-H-[1,2]Dithiole as a New Anti-Trypanosoma cruzi Chemotype: Biological and Mechanism of Action Studies

R. Pérez-Montfort, A. Gómez-Puyou, Beatriz Aguirre-López, 2015, Molecules.

Searching phase II enzymes inducers, from Michael acceptor-[1,2]dithiolethione hybrids, as cancer chemopreventive agents.

H. Cerecetto, Mercedes González, Mauricio Cabrera, 2015, Future medicinal chemistry.

A serendipitous one-step conversion of 3H-1,2-dithiole-3-thione to (E)-3-[1-(alkylthio)alkylidene]-3H-1,2-dithiole: an experimental and theoretical study

H. Cerecetto, Mercedes González, G. Echeverría, 2014, Molecular Diversity.

Cytotoxic, mutagenic and genotoxic effects of new anti-T. cruzi 5-phenylethenylbenzofuroxans. Contribution of phase I metabolites on the mutagenicity induction.

A. Monge, A. Merlino, H. Cerecetto, 2009, Toxicology letters.

New hybrid bromopyridine-chalcones as in vivo phase II enzyme inducers: potential chemopreventive agents

H. Cerecetto, Mercedes González, Mauricio Cabrera, 2016 .

New hits as phase II enzymes inducers from a focused library with heteroatom–heteroatom and Michael-acceptor motives

D. Kawano, M. Bollati-Fogolín, V. Eifler-Lima, 2015, Future science OA.

Genetic toxicology and preliminary in vivo studies of nitric oxide donor tocopherol analogs as potential new class of antiatherogenic agents

A. Vettorazzi, H. Botti, H. Rubbo, 2011, Drug and chemical toxicology.

Morphological evidence of the protective effects of a synthetic chalcone against the striatal myelin damage induced by glutaric acid

J. C. Rosillo, H. Cerecetto, G. Casanova, 2023, International journal of developmental neuroscience : the official journal of the International Society for Developmental Neuroscience.

Synthesis and antitumoral evaluation of natural product‐like compounds based on tropolone and benzotropolone derivatives

G. Moyna, Mauricio Cabrera, Macarena Eugui, 2022, Archiv der Pharmazie.

Garbage in, garbage out: how reliable training data improved a virtual screening approach against SARS-CoV-2 MPro

Lucas N. Alberca, A. Talevi, C. Kunick, 2023, Frontiers in Pharmacology.