D. L. Dyer

Efficacious, orally bioavailable thrombin inhibitors based on 3-aminopyridinone or 3-aminopyrazinone acetamide peptidomimetic templates.

J. Vacca, J. Shafer, Z. Chen, 1998, Journal of medicinal chemistry.

Antithrombotic efficacy of thrombin inhibitor L-374,087: intravenous activity in a primate model of venous thrombus extension and oral activity in a canine model of primary venous and coronary artery thrombosis.

J. Vacca, J. Shafer, S. Gardell, 1999, The Journal of pharmacology and experimental therapeutics.

L-374,087, an efficacious, orally bioavailable, pyridinone acetamide thrombin inhibitor.

J. Vacca, J. Shafer, Z. Chen, 1998, Bioorganic & medicinal chemistry letters.

Small, low nanomolar, noncovalent thrombin inhibitors lacking a group to fill the 'distal binding pocket'.

Youwei Yan, L. Kuo, S. D. Lewis, 2003, Bioorganic & medicinal chemistry letters.

Small, Low Nanomolar, Noncovalent Thrombin Inhibitors Lacking a Group to Fill the “Distal Binding Pocket”.

Youwei Yan, L. Kuo, S. D. Lewis, 2003 .

L-373,890, An achiral, noncovalent, subnanomolar thrombin inhibitor

J. Vacca, S. Gardell, A. Mulichak, 1997 .

L‐373,890, an Achiral, Noncovalent, Subnanomolar Thrombin Inhibitor.

J. Vacca, S. Gardell, A. Mulichak, 1997 .