U. Dolling

发表

An expedient one-pot synthesis for protected 2-thia-5-azabicyclo[2.2.1]heptan-3-ones. Versatile intermediates in the synthesis of carbapenem sidechains

P. Reider, K. Brands, G. Marchesini, 1996 .

The conformational bias of aryl, arylsulfonyl geminally substituted tertiary carbon centers: applications in substrate-based stereocontrol.

Jeremy P. Scott, Jennifer R. Chilenski, S. Oliver, 2006, Organic & biomolecular chemistry.

Intramolecular Aromatic 1,5-Hydrogen Transfer in Free Radical Reactions 1. Unprecedented Rearrangements in Pschorr Cyclization, Sandmeyer, and Hydro-, Hydroxy-, and Iododediazoniation Reactions

A. W. Douglas, N. L. Abramson, S. Karady, 1995 .

Stereoselective synthesis of 2-aryloxy acids from lactamide derived esters of racemic α-halo carboxylic acids

Paul N. Devine, R. Heid, D. Tschaen, 1996 .

A new general method for preparation of N-methoxy-N-methylamides. Application in direct conversion of an ester to a ketone

E. Grabowski, N. Yasuda, J. M. Williams, 1995 .

Asymmetric reduction of keto oxime ethers using oxazaborolidine reagents. The enantioselective synthesis of cyclic amino alcohols

P. Reider, R. Tillyer, D. Tschaen, 1995 .

Copper-mediated reaction of 2-halopyridines with ethyl bromodifluoroacetate

D. J. Wallace, Cameron J. Cowden, A. Davies, 2002 .

Preparation of 2-aryl- and 2-alkenyl-substituted carbapenems under mild suzuki cross-coupling conditions

Yulan Li, L. Xavier, N. Yasuda, 1993 .

Efficient Synthesis of α-Chloro Ketones via Reaction of Organometallic Reagents with N-Methoxy-N-Methylchloroacetamide

R. Tillyer, L. Frey, D. Tschaen, 1996 .

Observations on the DDQ Oxidation of 1-Acyldihydropyridines - A Synthetic Application

D. J. Wallace, Andrew D. Gibb, K. Brands, 2001 .

Asymmetric Synthesis of MK-0499

D. Cai, L. Frey, S. Karady, 1995 .

An efficient one-pot synthesis of annulated pyridines utilising a directed ortho-metallation/transmetallation approach

Cameron J. Cowden, A. Davies, D. Lieberman, 2004 .

Practical Asymmetric Synthesis of a Non-Peptidic αvβ3 Antagonist

Cameron J. Cowden, A. Davies, Gavin W. Stewart, 2005 .

Synthesis of N-arylated sultams: palladium- and copper-catalyzed cross coupling of aryl halides with 1,4-butane and 1,3-propanesultams

M. Palucki, D. Steinhuebel, D. Askin, 2004 .

An improved preparation of 3,5-bis(trifluoromethyl)acetophenone and safety considerations in the preparation of 3,5-bis(trifluoromethyl)phenyl Grignard reagent.

Donald C. Bachert, R. Cvetovich, J. Leazer, 2003, The Journal of organic chemistry.

Unprecedented Catalytic Three Component One-Pot Condensation Reaction: An Efficient Synthesis of 5-Alkoxycarbonyl- 4-aryl-3,4-dihydropyrimidin-2(1H)-ones

E. Hu, D. Sidler, U. Dolling, 1998 .

Unprecedented Catalytic Three Component One-Pot Condensation Reaction: An Efficient Synthesis of 5-Alkoxycarbonyl-4-aryl-3,4-dihydropyrimidin-2(1H)-ones.

D. Sidler, U. Dolling, H. HuEssa, 1998 .

Practical synthesis of the new carbapenem antibiotic ertapenem sodium.

D. Sidler, T. Novak, R. Skerlj, 2005, The Journal of organic chemistry.

2,3-Dichloro-5,6-dicyano-1,4-benzoquinone (DDQ) oxidation of silyl enol ethers to enones via DDQ-substrate adducts

E. Grabowski, A. Bhattacharya, L. Dimichele, 1989 .

Efficient catalytic asymmetric alkylations. 1. Enantioselective synthesis of (+)-indacrinone via chiral phase-transfer catalysis

E. Grabowski, U. Dolling, Paul Davis, 1984 .

Stereoselective Conjugate Addition Reactions of α,β-Unsaturated tert-Butyl Esters with Aryllithium Reagents†

A. Caillé, P. Reider, E. Grabowski, 1998 .

MILD ARYL ETHER FORMATION IN THE SEMISYNTHESIS OF THE NOVEL MACROLIDE IMMUNOSUPPRESSANT L-732,531

J. M. Williams, K. Brands, G. Marchesini, 1998 .

Stereoselective Double Ring Closing Metathesis Reactions in the Synthesis of Spirocyclic Compounds.

P. Bulger, D. J. Wallace, U. Dolling, 2000 .

Efficient catalytic asymmetric alkylations. 3. A kinetic and mechanistic study of the enantioselective phase-transfer methylation of 6,7-dichloro-5-methoxy-2-phenyl-1-indanone

E. Grabowski, D. Hughes, U. Dolling, 1987 .

An investigation into the alkylation of 1,2,4-triazole

P. Bulger, Cameron J. Cowden, A. Davies, 2000 .

METHOXYMETHYLATION OF ALCOHOLS, PHENOLS, AND AVERMECTIN AGLYCONES USING MOM-2-PYRIDYLSULFIDE

T. Novak, S. Karady, Benjamin F Marcune, 1999 .

Practical synthesis of aryl triflates under aqueous conditions.

D. Frantz, M. H. Kress, U. Dolling, 2002, Organic letters.

Practical synthesis of a highly functionalized thiazole ketone

L. Tan, E. Grabowski, Cheng-yi Chen, 2003 .

Efficient one-pot synthesis of the 2-aminocarbonylpyrrolidin-4-ylthio-containing side chain of the new broad-spectrum carbapenem antibiotic ertapenem.

P. Reider, R. Reamer, K. Conrad, 2002, The Journal of organic chemistry.

Acylimidazolides as Versatile Synthetic Intermediates for the Preparation of Sterically Congested Amides and Ketones: A Practical Synthesis of Proscar®

E. Grabowski, J. Amato, A. Bhattacharya, 1990 .

Convenient Synthesis and Isolation of 1-Aminocyclopropane-1-carboxylic Acid (ACC) and N-Protected ACC Derivatives

S. Allwein, Andrew Martins, T. Nelson, 2004 .

Practical and efficient synthesis of N-halo compounds

Hua Zhou, R. Volante, D. Gauthier, 2005 .

An improved method for chiral oxazaborolidine-catalyzed reduction of 4-chromanone analogs and MK-0499

A. W. Douglas, D. Cai, D. Tschaen, 1994 .

A double ring closing metathesis reaction in the rapid, enantioselective synthesis of NK-1 receptor antagonists.

J. Goodman, P. Reider, D. J. Wallace, 2001, Organic letters.

7-Norbornenylidene - a potentially nonclassical carbene

R. Moss, U. Dolling, Joanne R. Whittle, 1971 .

Development of a Phase Transfer Catalyzed Asymmetric Synthesis for an Estrogen Receptor Beta Selective Agonist

Jeremy P. Scott, S. Oliver, Khateeta M. Emerson, 2008 .

Enantioselective Robinson Annelations via Phase‐Transfer Catalysis

E. Grabowski, S. Karady, A. Bhattacharya, 1986 .

Silylation-mediated oxidation of 4-aza-3-ketosteroids with DDQ proceeds via DDQ-substrate adducts

A. W. Douglas, E. Grabowski, A. Bhattacharya, 1988 .

An efficient and general synthesis of 3-substituted propionaldehydes using the Suzuki-Miyaura coupling

Cameron J. Cowden, Sarah E. Brewer, A. Davies, 2004 .

Stereoselective synthesis of a potent thrombin inhibitor by a novel P2-P3 lactone ring opening.

Jeffrey C. Moore, M. Sturr, K. Gbewonyo, 2004, The Journal of organic chemistry.

Photolysis of phenyldiazomethane in olefinic matrices. Chemistry of triplet phenylcarbene

R. Moss, U. Dolling, 1971 .

A new synthesis of 1,2,4-triazolin-5-ones: application to the convergent synthesis of an NK1 antagonist

Cameron J. Cowden, A. Davies, Robert D. Wilson, 2000 .

A New Synthesis of 1,2,4-Triazolin-5-ones: Application to the Convergent Synthesis of an NK1 Antagonist.

Cameron J. Cowden, A. Davies, Robert D. Wilson, 2001 .

Preparation of 2-Aryl- and 2-Alkenyl-Substituted Carbapenems Under Mild Suzuki Cross-Coupling Conditions.

Yulan Li, L. Xavier, N. Yasuda, 1993 .

Regioselective synthesis of N-substituted-4-substituted isothiazolidine-1,1-dioxides

Faye J. Sheen, Ed Cleator, M. Bio, 2006 .

Regioselective Synthesis of N-Substituted-4-substituted Isothiazolidine-1,1-dioxides.

Faye J. Sheen, Ed Cleator, M. Bio, 2006 .

Practical Synthesis of Anti-Methicillin-Resistant Staphylococcus Aureus (MRSA) Carbapenem L-742,728

A. W. Douglas, Yulan Li, D. Mathre, 1998 .

Practical asymmetric synthesis of aprepitant, a potent human NK-1 receptor antagonist, via a stereoselective Lewis acid-catalyzed trans acetalization reaction.

P. Reider, E. Grabowski, Guojie Ho, 2002, The Journal of organic chemistry.

Synthesis and resolution of 3-fluoro-D,L-alanine-2-d: a selective deuteration via reductive amination with sodium borodeuteride

A. W. Douglas, E. Grabowski, M. Sletzinger, 1978 .

A Practical Synthesis of a ?-Secretase Inhibitor

Jeremy P. Scott, C. McWilliams, A. Davies, 2007 .

Expedient Diels–Alder assembly of 4-aryl-4-phenylsulfonyl cyclohexanones ☆

Jeremy P. Scott, E. M. Beck, A. Davies, 2004 .

Practical asymmetric synthesis of a gamma-secretase inhibitor exploiting substrate-controlled intramolecular nitrile oxide-olefin cycloaddition.

Jeremy P. Scott, R. Reamer, S. Oliver, 2006, The Journal of organic chemistry.

Asymmetric Reduction of Keto Oxime Ethers Using Oxazaborolidine Reagents. The Enantioselective Synthesis of Cyclic Amino Alcohols.

P. Reider, R. Tillyer, D. Tschaen, 1995 .

Sequential Dehydrogenation of 3-Keto-4-azasteroids. The Reaction of Ene-Lactams with 2,3-Dichloro-5,6-dicyano-1,4-benzoquinone (DDQ)

E. Grabowski, R. Reamer, J. M. Williams, 1995 .

Development of a Scaleable Synthesis of a 3-Aminopyrazinone Acetamide Thrombin Inhibitor

D. Hands, Khateeta M. Emerson, A. Davies, 2004 .